SUBSTITUTED PHENOXYETHYL (ISOPROPYL) ACYLOXYALKYL PHOSPHONATE COMPRISING PHOSPHORUSHETEROCYCLIC RING AND HAVING HERBICIDAL ACTIVITY, AND PREPARATION THEREFOR
    2.
    发明申请
    SUBSTITUTED PHENOXYETHYL (ISOPROPYL) ACYLOXYALKYL PHOSPHONATE COMPRISING PHOSPHORUSHETEROCYCLIC RING AND HAVING HERBICIDAL ACTIVITY, AND PREPARATION THEREFOR 有权
    取代的含有磷杂环戊烯的环氧乙烷(异丙基)乙酰氧基磷酸酯,并具有除草活性及其制备方法

    公开(公告)号:US20140171644A1

    公开(公告)日:2014-06-19

    申请号:US14185721

    申请日:2014-02-20

    CPC classification number: A01N57/36 C07F9/657118 C07F9/65742 C07F9/65748

    Abstract: A substituted phenoxyethyl(isopropyl)acyloxyalkyl phosphonate having phosphorusheterocyclic ring and having herbicidal activity, with a general formula of I, wherein R represents 5,5-dimethyl-1,3,2-dioxaphosphorinan-2-one-2-yl, or 1-oxo-1-phospha-2,6,7-trioxabicyclo[2,2,2]octan-4-yl, or 1-sulfo-1-phospha-2,6,7-trioxabicyclo 2,6,7-trioxabicyclo[2,2,2]octan-4-yl; R1 represents H, C1-C4 alkyl, phenyl, furyl, pyridyl, or phenyl substituted with methyl, methoxyl, nitro or chloro; R2 represents H, methyl, and methyl only if R in the general formula I is 1-sulfo-1-phospha-2,6,7-trioxabicyclo[2,2,2]octan-4-yl as phosphorusheterocyclic ring; X and Y represent H, halogen, C1-C4 alkyl or trifluoromethyl, and X and Y are the same or different. The compounds according to the present invention may be used as active component of dicotyledonous broadleaf weed herbicides.

    Abstract translation: 具有磷杂环并具有除草活性的取代的苯氧基乙基(异丙基)酰氧基烷基膦酸酯,具有通式I,其中R表示5,5-二甲基-1,3,2-二氧杂磷杂环己烷-2-酮-2-基或1 - 氧代-1-磷杂-2,6,7-三氧杂双环[2,2,2]辛-4-基或1-磺基-1-磷杂-2,6,7-三氧杂双环2,6,7-三氧杂双环 [2,2,2]辛-4-基; R 1表示H,C 1 -C 4烷基,苯基,呋喃基,吡啶基或被甲基,甲氧基,硝基或氯取代的苯基; 只有通式Ⅰ中的R是作为磷杂环的1-磺基-1-磷杂-2,6,7-三氧杂双环[2,2,2]辛-4-基,R2表示H,甲基和甲基。 X和Y表示H,卤素,C 1 -C 4烷基或三氟甲基,X和Y相同或不同。 根据本发明的化合物可以用作双子叶阔叶杂草除草剂的活性组分。

    Anti-bacterial agents based upon oxoanion binding
    4.
    发明授权
    Anti-bacterial agents based upon oxoanion binding 失效
    基于氧阴离子结合的抗菌剂

    公开(公告)号:US07326695B2

    公开(公告)日:2008-02-05

    申请号:US11435978

    申请日:2006-05-17

    Abstract: Compounds of the structure I: are useful for treating bacterial growth, wherein E is selected from the group consisting of B, P, and S, T1 and T2 are each independently selected from the group consisting of O, NR, and CH2, where R=H or C1-C8 alkyl, or C1-C8 oxoalkyl, and L is selected from the group consisting of ethylene, propylene, and four to six-membered alicyclic and aromatic rings, provided that structure I does not include AI-2-borate. The compounds may be used to treat bacterial infections in human beings and to regulate biofilm formation. Pharmaceutical compositions comprising one or more such compounds are useful for treating bacterial infections in human beings.

    Abstract translation: 结构I的化合物可用于治疗细菌生长,其中E选自B,P和S,T 1和T 2各自为 独立地选自O,NR和CH 2,其中R = H或C 1 -C 8烷基,或C 1个C 1 -C 8氧代烷基,L选自乙烯,丙烯和四至六元脂环和芳环,条件是结构I不 包括AI-2-硼酸盐。 该化合物可用于治疗人类的细菌感染并调节生物膜形成。 包含一种或多种这样的化合物的药物组合物可用于治疗人类的细菌感染。

    Pyrimidinetrione derivatives, agents containing them and their use as
agents for combating pests
    6.
    发明授权
    Pyrimidinetrione derivatives, agents containing them and their use as agents for combating pests 失效
    衍生物衍生物,包含它们的试剂及其用作组合物的试剂

    公开(公告)号:US5162327A

    公开(公告)日:1992-11-10

    申请号:US474379

    申请日:1990-02-02

    Abstract: Pyrimidinetrione derivatives, processes for their preparation, agents containing them and their use as agents for combating pests.Compounds of the formula I, tautomeric forms thereof of the formula Ia, stereoisomers thereof and the mixtures of these forms ##STR1## wherein R.sup.1 and R.sup.2 denote unsubstituted or substituted alkyl, alkenyl, alkynyl; alkoxy, alkylsulfonyl, alkylcarbonyl or cyano or optionally substituted phenyl, phenylsulfonyl or phenylcarbonyl,R.sup.3 denotes hydrogen, alkyl or optionally substituted phenyl,R.sup.4 denote H, OH, unsubstituted or substituted alkyl, alkenyl, alkynyl, phenylsulfonyl, phenylcarbonyl, phenylcarbamoyl or phenyl; alkylsulfonyl or alkylcarbonyl, which can be halogenated, alkylcarbamoyl or cyano,R.sup.5 and R.sup.6 denote halogen, alkoxy, alkylcarbonyl, alkoxycarbonyl, alkylsulfenyl, -sulfinyl or -sulfonyl, haloalkoxy, alkylamino, cyano, sulfo or nitro,A,X,Z and L denote oxygen, sulfur, sulfinyl, sulfonyl or nitrogen, which can be substituted by alkyl, or L denotes a double bond,M,D,E,Q and G denote carbon or nitrogen,V denotes carbon or substituted phosphorus,W denotes alkylene or haloalkylene, both of which can be substituted,Y.sup.1 denotes H, halogen, alkyl, alkylamino or hydroxyl,Y.sup.2 denotes oxygen, sulfur or nitrogen which is optionally substituted by alkyl andn amd m denote 0-4, and salts thereof which can be employed in agriculture or are physiologically tolerated, have advantageous actions against a broad spectrum or animal pests in agriculture and animal breeding.

    Abstract translation: 嘧啶四酮衍生物,其制备方法,含有它们的试剂及其作为防治害虫的试剂的用途。 (Ⅰ)的化合物,式Ia的互变异构体,其立体异构体和这些形式的混合物,其中R 1和R 2表示未取代或取代的烷基,烯基,炔基; 烷氧基,烷基磺酰基,烷基羰基或氰基或任选取代的苯基,苯基磺酰基或苯基羰基,R 3表示氢,烷基或任选取代的苯基,R 4表示H,OH,未取代或取代的烷基,烯基,炔基,苯基磺酰基,苯基羰基,苯基氨基甲酰基或苯基; 烷基磺酰基或烷基羰基,其可以被卤化,烷基氨基甲酰基或氰基,R5和R6表示卤素,烷氧基,烷基羰基,烷氧基羰基,烷基亚磺酰基, - 亚磺酰基或 - 磺酰基,卤代烷氧基,烷基氨基,氰基,磺基或硝基,A,X,Z和L 表示可被烷基取代的氧,硫,亚磺酰基,磺酰基或氮,或L表示双键,M,D,E,Q和G表示碳或氮,V表示碳或取代的磷,W表示亚烷基或 卤代亚烷基,它们都可以被取代,Y1表示H,卤素,烷基,烷基氨基或羟基,Y2表示氧,硫或氮,任选被烷基取代,n表示0-4,可以使用其盐 在农业中或具有生理上的耐受性,对农业和动物育种中的广谱或动物害虫具有有利的作用。

Patent Agency Ranking