Anti-bacterial agents based upon oxoanion binding
    3.
    发明授权
    Anti-bacterial agents based upon oxoanion binding 失效
    基于氧阴离子结合的抗菌剂

    公开(公告)号:US06737415B2

    公开(公告)日:2004-05-18

    申请号:US10227327

    申请日:2002-08-22

    Abstract: Compounds of the structure I: are useful for treating bacterial growth, wherein E is selected from the group consisting of B, P, and S, T1, and T2 are each independently selected from the group consisting of O, NR, and CH2, where R=H or C1-C8 alkyl, or C1-C8 oxoalkyl, and L is selected from the group consisting of ethylene, propylene, and four to six-membered alicyclic and aromatic rings, provided that structure I does not include AI-2-borate. The compounds may be used to treat bacterial infections in human beings and to regulate biofilm formation. Pharmaceutical compositions comprising one or more such compounds are useful for treating bacterial infections in human beings.

    Abstract translation: 结构I的化合物可用于治疗细菌生长,其中E选自B,P和S,T1和T2各自独立地选自O,NR和CH 2,其中 R = H或C 1 -C 8烷基或C 1 -C 8氧代烷基,L选自乙烯,丙烯和四至六元脂环和芳环,条件是结构I不包括AI-2- 硼酸盐 该化合物可用于治疗人类的细菌感染并调节生物膜形成。 包含一种或多种这样的化合物的药物组合物可用于治疗人类的细菌感染。

    Pest controlling compositions
    4.
    发明授权
    Pest controlling compositions 失效
    害虫控制组合物

    公开(公告)号:US4902690A

    公开(公告)日:1990-02-20

    申请号:US218491

    申请日:1988-07-06

    CPC classification number: A01N57/36 A01N43/90 A01N61/00 Y10S424/08 Y10S424/10

    Abstract: A pest-controlling composition which comprises:(A) a first compound capable of substantially inhibiting a phosphodiesterase enzyme (PDE) of said pest; and(B) a second compound having pest-dontrolling activity towards said pest, selected from the group consisting of(1) a substantial octopamine agonist toward an octopamine receptor present in said pest;(2) a compound directly and substantially stimulating the enzyme, adenylate cyclase; and(3) a cyclic adenosine monophosphate (cAMP) analogue.

    Abstract translation: 一种害虫控制组合物,其包含:(A)能够基本上抑制所述害虫的磷酸二酯酶(PDE)的第一化合物; 和(B)对所述有害生物具有害虫控制活性的第二化合物,其选自(1)对所述害虫中存在的章鱼胺受体的基本章鱼酚激动剂; (2)化合物直接且基本上刺激酶,腺苷酸环化酶; 和(3)环磷酸腺苷(cAMP)类似物。

    Benzoxaphospholes
    5.
    发明授权
    Benzoxaphospholes 失效
    苯并磷杂酚

    公开(公告)号:US4219510A

    公开(公告)日:1980-08-26

    申请号:US55429

    申请日:1979-07-06

    Applicant: James A. Miles

    Inventor: James A. Miles

    CPC classification number: C07F9/657172 A01N57/36 C07F9/657181

    Abstract: This disclosure relates to a class of bicyclic hetero compounds. More particularly, this disclosure relates to novel substituted benzoxaphospholes which are useful as herbicides. This disclosure further relates to herbicidal compositions containing such benzoxaphospholes and to herbicidal methods employing such compounds and compositions.

    Abstract translation: 本公开涉及一类双环杂化合物。 更具体地说,本公开涉及可用作除草剂的新型取代的苯并二磷杂磷素。 本公开进一步涉及含有这些苯并磷杂环的除草组合物和使用这种化合物和组合物的除草方法。

    Plant-growth-regulating compositions containing phospholanium salts
    7.
    发明授权
    Plant-growth-regulating compositions containing phospholanium salts 失效
    含有磷酸盐的植物生长调节组合物

    公开(公告)号:US4021221A

    公开(公告)日:1977-05-03

    申请号:US581527

    申请日:1975-05-28

    CPC classification number: C07F9/65688 A01N57/36

    Abstract: Compositions for regulating the growth of plants containing phospholanium salts of the formula: ##STR1## in which R.sup.1 is optionally substituted alkyl, alkenyl, alkynyl or cycloalkyl, or aralkyl which is optionally substituted in the aryl part,R.sup.2 is optionally substituted alkyl, alkenyl, alkynl or cycloalkyl, or aralkyl which is optionally substituted in the aryl part,R.sup.3 is halogen or alkyl,n is 0, 1 or 2, andA.sup.- is one equivalent of an anion of a nonphytotoxic acidAre outstandingly useful to inhibit, enhance, or modify the growth of plants, even at relatively low dosages.

    Abstract translation: 用于调节含有下式的磷酸盐的植物的生长的组合物:其中R 1是任选取代的烷基,烯基,炔基或环烷基或在芳基部分任选被取代的芳烷基,R 2是任选取代的 烷基,烯基,炔烃或环烷基,或在芳基部分任选被取代的芳烷基,R 3是卤素或烷基,N IS 0,1 OR 2,和A 1是非鸟苷酸的阴离子的1当量ARE OUTSTANDLYLY 有用的是抑制,增强或修改植物的生长,即使是相对低的量。

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