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公开(公告)号:US5326755A
公开(公告)日:1994-07-05
申请号:US923970
申请日:1992-09-10
IPC分类号: A01N37/18 , A01N37/28 , A01N43/40 , A01N49/00 , A01N55/10 , A01P7/02 , A01P7/04 , C07C233/09 , C07C233/13 , C07C233/22 , C07C233/91 , C07C313/28 , C07D213/71 , C07F7/10 , A01N55/00 , C07C233/12 , C07C222/47
CPC分类号: A01N49/00 , C07C233/91 , C07C313/28 , C07D213/71 , C07C2101/02
摘要: The present application discloses pesticidally active compounds of formula I:QQ.sup.1 CR.sup.1 .dbd.CR.sup.2 CR.sup.3 .dbd.CR.sup.4 C(.dbd.X.sup.1)NR.sup.5 R.sup.6or a salt thereof, wherein Q is an monocyclic aromatic ring, or Q is a dihalovinyl group or a group R.sup.7 --C.dbd.C-- where R.sup.7 is C.sub.1-4 alkyl, tri C.sub.1-4 alkylsilyl, halogen or hydrogen; Q.sup.1 is a 1,2-cyclopropyl ring optionally substituted by one or more groups selected from C.sub.1-3 alkyl, halo, C.sub.1-3 haloalkyl, alkynyl, or cyano; R.sup.1, R.sup.2, R.sup.3 and R.sup.4 are the same or different with at least one being hydrogen and the others being independently selected from hydrogen, halo, C.sub.1-4 alkyl or C.sub.1-4 haloalkyl; X.sup.1 is oxygen or sulphur; R.sup.5 is C.sub.1-8 hydrocarbyl optionally substituted, halo, cyano, trifluoromethyl, trifluoromethylthio or C.sub.1-6 alkoxy; and R.sup.6 is selected from:(A) --Y.dbd.X.sup.2 --(R.sup.8).sub.a where X.sup.2 is O or S, Y is carbon, R.sup.8 is hydrogen, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, C.sub.1-5 alkylcarbonyl or aryl or CO.sub.2 R.sup.9 where R.sup.9 is an C.sub.1-4 alkyl or aryl, and a is 1 or 2;(B) --CR.sup.15 R.sup.16 X.sup.3 R.sup.17 where R.sup.15 and R.sup.16 are hydrogen or C.sub.1-4 alkyl, X.sup.3 is oxygen or sulphur and R.sup.17 is C.sub.1-4 alkyl, C.sub.1-5 alkylcarbonyl or aralkylcarbonyl R.sup.17,R.sup.15 X.sup.3, their preparation, pesticidal compositions containing them and their use against pests.
摘要翻译: PCT No.PCT / GB91 / 00539 Sec。 371日期:1992年9月10日 102(e)日期1992年9月10日PCT 1991年4月8日PCT PCT。 WO91 / 16301 PCT出版物 1991年10月31日。本申请公开了式I的杀虫活性化合物:QQ1CR1 = CR2CR3 = CR4C(= X1)NR5R6或其盐,其中Q为单环芳环,或Q为二卤代乙烯基或基团 R7-C = C-,其中R7是C1-4烷基,三C1-4烷基甲硅烷基,卤素或氢; Q1是任选被一个或多个选自C 1-3烷基,卤素,C 1-3卤代烷基,炔基或氰基的基团取代的1,2-环丙基环; R 1,R 2,R 3和R 4相同或不同,至少一个为氢,其余独立地选自氢,卤素,C 1-4烷基或C 1-4卤代烷基; X1是氧或硫; R 5为任选取代的C 1-8烃基,卤素,氰基,三氟甲基,三氟甲硫基或C 1-6烷氧基; 并且R 6选自:(A)-Y = X 2 - (R 8)a,其中X 2为O或S,Y为碳,R 8为氢,C 1-4烷基,C 1-4烷氧基,C 1-5烷基羰基或芳基或 CO 2 R 9,其中R 9为C 1-4烷基或芳基,a为1或2; (B)-CR15R16X3R17其中R15和R16为氢或C1-4烷基,X3为氧或硫,R17为C1-4烷基,C1-5烷基羰基或芳烷基羰基R17,R15X3,其制备方法,含有它们的杀虫组合物及其用途 反对有害生物
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2.
公开(公告)号:US5380733A
公开(公告)日:1995-01-10
申请号:US991239
申请日:1992-12-16
IPC分类号: A01N37/18 , A01N43/08 , A01N43/40 , A01N43/46 , A01N43/54 , A01N43/56 , A01N43/78 , A01N43/80 , A01N43/82 , C07C235/22 , C07C235/24 , C07D211/06 , C07D213/30 , C07D213/75 , C07D213/81 , C07D231/38 , C07D231/40 , C07D239/26 , C07D239/42 , C07D261/14 , C07D263/48 , C07D277/20 , C07D277/44 , C07D277/46 , C07D285/12 , C07D285/135 , C07D295/18 , C07D295/32 , C07D307/33 , C07D417/12 , C07F9/24 , C07D405/10
CPC分类号: C07D213/75 , A01N37/18 , A01N43/08 , A01N43/40 , A01N43/46 , A01N43/54 , A01N43/56 , A01N43/78 , A01N43/80 , A01N43/82 , C07D231/38 , C07D239/42 , C07D261/14 , C07D277/46 , C07D285/135 , C07D295/32 , C07D307/33
摘要: Compounds of the formula:Q(CH.sub.2).sub.a (O).sub.b Q.sub.1 CR.sub.2 .dbd.CR.sub.3 CR.sub.4 .dbd.CR.sub.5 CX.sub.1 NHR.sub.1wherein the terms Q, Q.sub.1, R.sub.1, R.sub.2, R.sub.3, R.sub.4, R.sub.5, X.sub.1 and the integers a and b are defined in the specification, or salts thereof. Said compounds are useful as pesticides.
摘要翻译: 化合物Q(CH2)a(O)bQ1CR2 = CR3CR4 = CR5CX1NHR1其中术语Q,Q1,R1,R2,R3,R4,R5,X1和整体a和b在本说明书中定义,或盐 其中。 所述化合物可用作杀虫剂。
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公开(公告)号:US5229424A
公开(公告)日:1993-07-20
申请号:US835683
申请日:1992-02-14
IPC分类号: A01N37/18 , A01N49/00 , C07C45/00 , C07C45/29 , C07C45/44 , C07C45/54 , C07C47/24 , C07C47/457 , C07C47/546 , C07C47/55 , C07C49/237 , C07C57/60 , C07C63/33 , C07C63/72 , C07C233/10 , C07C233/11 , C07C233/22 , C07C235/34 , C07C327/44 , C07D213/61 , C07D317/28 , C07F7/08 , C07F9/24
CPC分类号: C07F9/247 , A01N37/18 , A01N49/00 , C07C233/10 , C07C233/11 , C07C233/22 , C07C235/34 , C07C327/44 , C07C45/00 , C07C45/29 , C07C45/292 , C07C45/44 , C07C45/54 , C07C47/24 , C07C47/457 , C07C47/546 , C07C47/55 , C07C49/237 , C07C57/60 , C07C63/33 , C07C63/72 , C07D213/61 , C07D317/28 , C07F7/0818 , C07C2101/02
摘要: The present invention discloses pesticidally active compounds of formula (II) ##STR1## or a salt thereof, wherein Q is a monocylcic aromatic ring, or fused bicyclic ring system of which at least one ring is aromatic containing 9 or 10 atoms of which one may be nitrogen and the rest carbon each ring system being optionally substituted, or Q is a dihalovinyl group or a group R.sup.6 --C.tbd.C-- where R.sup.6 is C.sub.1-4 alkyl, tri C.sub.1-4 alkylsilyl, halogen or hydrogen; R.sup.2, R.sup.3, R.sup.4 and R.sup.5 are the same or different with at least one being hydrogen and the others being independently selected from hydrogen, halo, C.sub.1-4 alkyl or C.sub.1-4 haloalkyl; and R.sup.1 is selected from hydrogen and C.sub.1-8 hydrocarbyl optionally substituted by dioxalanyl, halo, cyano, trifluoromethyl, trifluoromethylthio or C.sub.1-6 alkoxy and X.sup.1 is hydrogen, fluoro or chloro.
摘要翻译: 本发明公开了式(II)的杀虫活性化合物或其盐,其中Q是单环芳香环,或稠合双环体系,其中至少一个芳环含有9或10个原子 其中一个可以是氮,其余的碳各个环系被任选取代,或Q是二卤乙烯基或R6-C 3BOND-,其中R6是C1-4烷基,三C1-4烷基甲硅烷基,卤素或氢; R 2,R 3,R 4和R 5相同或不同,至少一个为氢,其余独立地选自氢,卤素,C 1-4烷基或C 1-4卤代烷基; 卤素,氰基,三氟甲基,三氟甲硫基或C 1-6烷氧基,且X 1为氢,氟或氯。
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公开(公告)号:US5605912A
公开(公告)日:1997-02-25
申请号:US321843
申请日:1994-10-14
IPC分类号: A01N37/18 , A01N43/08 , A01N43/40 , A01N43/46 , A01N43/54 , A01N43/56 , A01N43/78 , A01N43/80 , A01N43/82 , C07C235/22 , C07C235/24 , C07D211/06 , C07D213/30 , C07D213/75 , C07D213/81 , C07D231/38 , C07D231/40 , C07D239/26 , C07D239/42 , C07D261/14 , C07D263/48 , C07D277/20 , C07D277/44 , C07D277/46 , C07D285/12 , C07D285/135 , C07D295/18 , C07D295/32 , C07D307/33 , C07D417/12 , C07F9/24 , C07D405/08 , C07D405/12
CPC分类号: C07D213/75 , A01N37/18 , A01N43/08 , A01N43/40 , A01N43/46 , A01N43/54 , A01N43/56 , A01N43/78 , A01N43/80 , A01N43/82 , C07D231/38 , C07D239/42 , C07D261/14 , C07D277/46 , C07D285/135 , C07D295/32 , C07D307/33
摘要: A compound of the formula: ##STR1## where Q is phenyl or naphthyl optionally substituted by (a) C.sub.1-6 hydrocarbyl, C.sub.1-6 alkoxy or methylenedioxy, which in turn is optionally substituted by one to five halogen atoms; or(b) halo, cyano, nitro; or(c) a group S(O).sub.n R.sub.7 wherein n=0, 1, or 2 and R.sub.7 is C.sub.1-6 alkyl optionally substituted by halogen, or R.sub.7 is amino optionally substituted by one or two C.sub.1-6 alkyl groups; or a group NR.sub.8 R.sub.9 where R.sub.8 and R.sub.9 are independently selected from hydrogen, C.sub.1-6 alkyl or a group COR.sub.12 where R.sub.12 is C.sub.1-6 alkyl or C.sub.1-6 alkoxy;Q.sub.1 is a 1,2-cyclopropyl ring optionally substituted by a group selected from C.sub.1-13 alkyl, halo, C.sub.1-3 haloalkyl or C.sub.1-13 alkynyl or cyano;R.sub.2, R.sub.3, R.sub.4 and R.sub.5 are the same or different with at least one being hydrogen and the others being independently selected from the group consisting of hydrogen, halo, C.sub.1-4, alkyl or C.sub.1-4 haloalkyl;X.sub.1 is oxygen or sulfur;R.sub.1 is a saturated 6 membered heterocycle containing a nitrogen atom which is bound to NH through a nitrogen atom and their use as pesticides, inecticides and acaricides.
摘要翻译: 其中Q是任选被(a)C 1-6烃基,C 1-6烷氧基或亚甲二氧基取代的苯基或萘基的化合物,其又可任选地被一至五个卤素原子取代; 或(b)卤素,氰基,硝基; 或(c)S(O)n R 7基团,其中n = 0,1或2,R 7为任选被卤素取代的C 1-6烷基,或者R 7为任选被一个或两个C 1-6烷基取代的氨基; 或NR 8 R 9基团,其中R 8和R 9独立地选自氢,C 1-6烷基或COR 12基团,其中R 12是C 1-6烷基或C 1-6烷氧基; Q1是任选被选自C 1-13烷基,卤素,C 1-3卤代烷基或C 1-13炔基或氰基的基团取代的1,2-环丙基环; R 2,R 3,R 4和R 5相同或不同,至少一个为氢,其余独立地选自氢,卤素,C 1-4,烷基或C 1-4卤代烷基; X1是氧或硫; R1是含有氮原子的饱和6元杂环,氮原子通过氮原子与NH键合,它们用作杀虫剂,杀虫剂和杀螨剂。
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公开(公告)号:US5352822A
公开(公告)日:1994-10-04
申请号:US43817
申请日:1993-04-07
IPC分类号: A01N37/18 , A01N49/00 , C07C45/00 , C07C45/29 , C07C45/44 , C07C45/54 , C07C47/24 , C07C47/457 , C07C47/546 , C07C47/55 , C07C49/237 , C07C57/60 , C07C63/33 , C07C63/72 , C07C233/10 , C07C233/11 , C07C233/22 , C07C235/34 , C07C327/44 , C07D213/61 , C07D317/28 , C07F7/08 , C07F9/24
CPC分类号: C07F9/247 , A01N37/18 , A01N49/00 , C07C233/10 , C07C233/11 , C07C233/22 , C07C235/34 , C07C327/44 , C07C45/00 , C07C45/29 , C07C45/292 , C07C45/44 , C07C45/54 , C07C47/24 , C07C47/457 , C07C47/546 , C07C47/55 , C07C49/237 , C07C57/60 , C07C63/33 , C07C63/72 , C07D213/61 , C07D317/28 , C07F7/0818 , C07C2101/02
摘要: The present invention discloses pesticidally active compounds of formula (II) ##STR1## or a salt thereof, wherein Q is an monocyclic aromatic ring, or fused bicyclic ring system of which at least one ring is aromatic containing 9 or 10 atoms of which one may be nitrogen and the rest carbon each ring system being optionally substituted, or Q is a dihalovinyl group or a group R.sup.6 --C.tbd.C-- where R.sup.6 is C.sub.1-4 alkyl, tri C.sub.1-4 alkylsilyl, halogen or hydrogen; R.sup.2, R.sup.3 , R.sup.4 and R.sup.5 are the same or different with at least one being hydrogen and the others being independently selected from hydrogen, halo, C.sub.1-4 alkyl or C.sub.1-4 haloalkyl; and R.sup.1 is selected from hydrogen and C.sub.1-8 hydrocarbyl optionally substituted by dioxalanyl, halo, cyano, trifluoromethyl, trifluoromethylthio or C.sub.1-6 alkoxy and X.sup.1 is hydrogen, fluoro or chloro.
摘要翻译: 本发明公开了式(II)的杀虫活性化合物或其盐,其中Q是单环芳香环或稠合双环体系,其中至少一个环是芳族的,含有9或10个原子的 其中一个可以是氮,其余的碳各个环系被任选取代,或Q是二卤乙烯基或R6-C 3BOND-,其中R6是C1-4烷基,三C1-4烷基甲硅烷基,卤素或氢; R 2,R 3,R 4和R 5相同或不同,至少一个为氢,其余独立地选自氢,卤素,C 1-4烷基或C 1-4卤代烷基; 卤素,氰基,三氟甲基,三氟甲硫基或C 1-6烷氧基,且X 1为氢,氟或氯。
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公开(公告)号:US5202356A
公开(公告)日:1993-04-13
申请号:US729847
申请日:1991-07-12
IPC分类号: A01N37/18 , A01N49/00 , C07C45/00 , C07C45/29 , C07C45/44 , C07C45/54 , C07C47/24 , C07C47/457 , C07C47/546 , C07C47/55 , C07C49/237 , C07C57/60 , C07C63/33 , C07C63/72 , C07C233/10 , C07C233/11 , C07C233/22 , C07C235/34 , C07C327/44 , C07D213/61 , C07D317/28 , C07F7/08 , C07F9/24
CPC分类号: C07F9/247 , A01N37/18 , A01N49/00 , C07C233/10 , C07C233/11 , C07C233/22 , C07C235/34 , C07C327/44 , C07C45/00 , C07C45/29 , C07C45/292 , C07C45/44 , C07C45/54 , C07C47/24 , C07C47/457 , C07C47/546 , C07C47/55 , C07C49/237 , C07C57/60 , C07C63/33 , C07C63/72 , C07D213/61 , C07D317/28 , C07F7/0818 , C07C2101/02
摘要: The present Application discloses pesticidally active compounds of the formula (I):Q Q.sup.1 CR.sup.2 =CR.sup.3 CR.sup.4 =CR.sup.5 C (.dbd.X) NHR.sup.1or a salt thereof, wherein Q is an monocyclic aromatic ring. or fused bicyclic ring system of which at least one ring is aromatic containing 9 or 10 atoms of which one may be nitrogen and the rest carbon each optionally substituted, or Q is a dihalovinyl group or a group R.sup.6 --C.tbd.C-- where R.sup.6 is C.sub.1-4 alkyl, tri C.sub.1-4 alkylsilyl, halogen or hydrogen; Q.sup.1 is a 1,2-cyclopropyl ring optionally substituted by one or more groups selected from C.sub.1-3 alkyl. halo, C.sub.1-3 haloalkyl, alkynyl, or cyano; R.sup.2,R.sup.3, R.sup.4 and R.sup.5 are the same or different with at least one being hydrogen and the others being independently selected from hydrogen, halo. C.sub.1-4 alkyl or C.sub.1-4 haloalkyl; X is oxygen or sulphur; and R.sup.1 is selected from hydrogen and C.sub.1-8 hydrocarbyl optionally substituted by dioxalanyl, halo, cyano, trifluoromethyl, trifluoromethylthio or C.sub.1-6 alkoxy. their preparation, pesticidal compositions containing them and their use against pests.
摘要翻译: 本申请公开了式(I)的杀虫活性化合物:Q Q1 CR2 = CR3 CR4 = CR5C(= X)NHR1或其盐,其中Q是单环芳香环。 或稠合双环体系,其中至少一个芳环含有9或10个原子,其中一个可以是氮,其余的碳各自任选被取代,或Q是二卤代乙烯基或R6-C 3BOND-,其中R6是 C 1-4烷基,三C 1-4烷基甲硅烷基,卤素或氢; Q1是任选被一个或多个选自C 1-3烷基的基团取代的1,2-环丙基环。 卤素,C 1-3卤代烷基,炔基或氰基; R 2,R 3,R 4和R 5相同或不同,至少一个为氢,而其它独立地选自氢,卤素。 C 1-4烷基或C 1-4卤代烷基; X是氧或硫; 卤素,氰基,三氟甲基,三氟甲硫基或C 1-6烷氧基取代的C 1-8烃基。 它们的制备,含有它们的杀虫剂组合物及其对害虫的用途。
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公开(公告)号:US5114940A
公开(公告)日:1992-05-19
申请号:US355976
申请日:1989-05-22
IPC分类号: A01N43/42 , A01N43/54 , A01N43/58 , A01N43/60 , A01N43/78 , A01N49/00 , C07D215/14 , C07D215/20 , C07D215/22 , C07D215/227 , C07D215/233 , C07D215/26 , C07D215/28 , C07D215/36 , C07D215/54 , C07D217/16 , C07D217/22 , C07D217/24 , C07D237/28 , C07D237/30 , C07D239/88 , C07D239/95 , C07D241/44 , C07D277/68 , C07D405/12
CPC分类号: C07D215/227 , A01N43/42 , A01N49/00 , C07D215/14 , C07D215/20 , C07D215/22 , C07D215/233 , C07D215/26 , C07D215/28 , C07D215/36 , C07D215/54 , C07D217/24 , C07D237/28 , C07D237/30 , C07D239/95 , C07D241/44 , C07D277/68
摘要: Compound of the formula (I) are disclosedArQQ.sup.1 C(.dbd.X)NHR.sup.1 (I)or a salt thereof, wherein Ar is an optionally substituted polycyclic ring system containing n rings, where n is the integer 2 or 3, at least n-1 rings being aromatic and containing one to three ring nitrogen atoms and optionally containing one or more additional heteroatoms; Q is an alkyl chain containing 1 to 12 carbon atoms and optionally containing a sulphur or one or two oxygen atoms; Q.sup.1 is a group (C(R.sup.2).dbd.C(R.sup.3)).sub.a --(C(R.sup.4).dbd.C(R.sup.5)) wherein a is 0 or 1, R.sup.2, R.sup.3, R.sup.4 and R.sup.5 are the same or different, at least two being hydrogen and the other two being independently selected from hydrogen, halo, C.sub.1-4 haloalkyl; X is oxygen or sulphur; and R.sup.1 is selected from hydrogen and C.sub.1-8 hydrocarbyl optionally substituted by dioxalanyl, halo, cyano, trifluoromethyl, trifluoromethylthio or C.sub.1-6 alkoxy are described which have activity particularly against arthropod pests. Pesticidal formulations containing the compounds of the formula (1), their use in the control of pests and method for their preparation are also disclosed.
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公开(公告)号:US5459149A
公开(公告)日:1995-10-17
申请号:US309430
申请日:1994-09-20
IPC分类号: A01N37/18 , A01N37/22 , A01N37/24 , A01N37/46 , A01N43/42 , A01N47/20 , A01N49/00 , A01P7/02 , A01P7/04 , C07C233/10 , C07C233/11 , C07C233/15 , C07C233/29 , C07C233/33 , C07C233/44 , C07C233/55 , C07C235/28 , C07C255/20 , C07C255/60 , C07C271/64 , C07C309/88 , C07C323/41 , C07C327/44 , C07D215/22 , C07D215/227 , C07F7/10 , C07C235/00
CPC分类号: C07D215/227 , A01N37/22 , A01N37/24 , A01N37/46 , A01N43/42 , A01N47/20 , A01N49/00 , C07C233/11 , C07C233/15 , C07C233/29 , C07C233/33 , C07C233/44 , C07C233/55 , C07C255/60 , C07C271/64 , C07C309/88 , C07C323/41 , C07C327/44 , C07C2101/02 , C07C2102/08 , C07C2102/10
摘要: The present Application discloses pesticidally active compounds of formula (I):Q(CH.sub.2).sub.a (O).sub.b Q.sup.1 CR.sup.2 =CR.sup.3 CR.sup.4 =CR.sup.5 CXNR.sup.1 R.sup.xor a salt or propesticide thereof, wherein Q is an optionally substituted aromatic monocyclic or fused bicyclic ring system in which at least one ring is aromatic, or Q is a dihalovinyl group or a group R.sup.6 --C=C--where R.sup.6 is C.sub.1-4 alkyl, tri C.sub.1-4 alkylsilyl, halo or hydrogen; Q.sup.1 is a 1,2-cyclopropyl ring optionally substituted by one or more groups selected from C.sub.1-3 alkyl, halo, C.sub.1-3 haloalkyl, C.sub.2-3 alkynyl, or cyano; or Q.sup.1 is (CH.sub.2).sub.7 ; a=0 or 1; b=0 or 1; R.sup.2, R.sup.3, R.sup.4 and R.sup.5 are the same or different with at least one being hydrogen and the others being independently selected from hydrogen, halo, C.sub.1-4 alkyl or C.sub.1-4 haloalkyl; X is oxygen or sulphur;R.sup.1 is phenyl optionally substituted by 1-5 substituents chosen from: a) C.sub.1-4 alkyl, C.sub.1-4 alkoxy, phenoxy and methylenedioxy, each optionally substituted by 1 to 5 halo; b) halo, cyano, nitro, formyl, C.sub.1-5 acyl; c) C.sub.2-3 alkynyl, C.sub.2-3 alkenyl, each optionally substituted by 1 to 5 halo; d) a group S(O).sub.n R.sup.7 wherein n=0, 1, 2 and R.sup.7 is C.sub.1-4 alkyl, halo or NR.sup.8 R.sup.9 wherein R.sup.8 and R.sup.9 are independently selected from hydrogen, C.sub.1-4 alkyl and C.sub.1-4 acyl; and a group e) NR.sup.8 R.sup.9 where R.sup.8 and R.sup.9 are as defined above; R.sup.X is hydrogen or an optionally substituted C.sub.1-8 alkyl or benzyl group, their preparation, pesticidal compositions containing them and their use against pests.
摘要翻译: 本申请公开了式(I)的杀虫活性化合物:Q(CH2)a(O)bQ1 CR2 = CR3 CR4 = CR5 CXNR1Rx或其盐或农药,其中Q是任选取代的芳族单环或稠合双环体系 其中至少一个环是芳族的,或Q是二卤代乙烯基或基团R6-C = C-,其中R6是C1-4烷基,三C1-4烷基甲硅烷基,卤素或氢; Q1是任选被一个或多个选自C 1-3烷基,卤素,C 1-3卤代烷基,C 2-3炔基或氰基的基团取代的1,2-环丙基环; 或Q 1为(CH 2)7; a = 0或1; b = 0或1; R 2,R 3,R 4和R 5相同或不同,至少一个为氢,其余独立地选自氢,卤素,C 1-4烷基或C 1-4卤代烷基; X是氧或硫; R1是任选被1-5个选自下列的取代基取代的苯基:a)C 1-4烷基,C 1-4烷氧基,苯氧基和亚甲二氧基,各自任选被1至5个卤素取代; b)卤素,氰基,硝基,甲酰基,C 1-5酰基; c)C2-3炔基,C2-3烯基,各自任选被1至5个卤素取代; d)基团S(O)n R 7,其中n = 0,1,2且R 7是C 1-4烷基,卤素或NR 8 R 9,其中R 8和R 9独立地选自氢,C 1-4烷基和C 1-4酰基; 和基团e)NR 8 R 9,其中R 8和R 9如上所定义; RX是氢或任选取代的C 1-8烷基或苄基,它们的制备方法,含有它们的杀虫组合物及其对害虫的用途。
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公开(公告)号:US5547976A
公开(公告)日:1996-08-20
申请号:US290921
申请日:1994-08-23
IPC分类号: A61K31/40 , A61K31/44 , A61P31/12 , A61P31/22 , C07D403/14 , C07D487/14 , C07D491/147 , A61K31/395
CPC分类号: C07D403/14 , A61K31/40 , A61K31/44 , C07D487/14
摘要: The present invention relates to indolopyrolocarbazole derivatives, to their use in methods of treatment or prophylaxis of at least one viral infection or cardiovascular diseases; and pharmaceutical formulations containing such derivatives.
摘要翻译: PCT No.PCT / GB93 / 00571 Sec。 371日期:1994年8月23日 102(e)日期1994年8月23日PCT 1993年3月19日PCT公布。 公开号WO93 / 18766 日期:1993年9月30日本发明涉及吲哚并咔唑衍生物,用于治疗或预防至少一种病毒感染或心血管疾病的方法; 和含有这些衍生物的药物制剂。
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公开(公告)号:US5270343A
公开(公告)日:1993-12-14
申请号:US898135
申请日:1992-06-15
IPC分类号: A01N37/18 , A01N37/22 , A01N37/24 , A01N37/46 , A01N43/42 , A01N47/20 , A01N49/00 , A01P7/02 , A01P7/04 , C07C233/10 , C07C233/11 , C07C233/15 , C07C233/29 , C07C233/33 , C07C233/44 , C07C233/55 , C07C235/28 , C07C255/20 , C07C255/60 , C07C271/64 , C07C309/88 , C07C323/41 , C07C327/44 , C07D215/22 , C07D215/227 , C07F7/10 , C07C235/00
CPC分类号: C07D215/227 , A01N37/22 , A01N37/24 , A01N37/46 , A01N43/42 , A01N47/20 , A01N49/00 , C07C233/11 , C07C233/15 , C07C233/29 , C07C233/33 , C07C233/44 , C07C233/55 , C07C255/60 , C07C271/64 , C07C309/88 , C07C323/41 , C07C327/44 , C07C2101/02 , C07C2102/08 , C07C2102/10
摘要: The present Application discloses pesticidally active compounds of formula (I):Q(CH.sub.2).sub.a (O).sub.b Q.sup.1 CR.sup.2 .dbd.CR.sup.2 .dbd.CR.sup.3 CR.sup.4 .dbd.CR.sup.5 CXNR.sup.1 R.sup.xor a salt or propesticide thereof, wherein Q is an optionally substituted aromatic monocyclic or fused bicyclic ring system in which at least one ring is aromatic, or Q is a dihalovinyl group or a group R.sup.6 --C.tbd.C-- where R.sup.6 is C.sub.1-4 alkyl, tri C.sub.1-4 alkylsilyl, halo or hydrogen; Q.sup.1 is a 1,2-cyclopropyl ring optionally substituted by one or more groups selected from C.sub.1-3 alkyl, halo, C.sub.1-3 haloalkyl, C.sub.2-3 alkynyl, or cyano; or is (CH.sub.2).sub.7 ;a=0 or 1; b= 0 or 1;R.sup.2, R.sup.3, R.sup.4 and R.sup.5 are the same or different with at least one being hydrogen and the others being independently selected from hydrogen, halo, C.sub.1-4 alkyl or C.sub.1-4 haloalkyl;X is oxygen or sulphur;R.sup.1 is phenyl optionally substituted by 1-5 substituents chosen from:a) C.sub.1-4 alkyl, C.sub.1-4 alkoxy, phenoxy and methylenedioxy, each optionally substituted by 1 to 5 halo;b) halo, cyano, nitro, formyl, C.sub.1-5 acyl;c) C.sub.2-3 alkynyl, C.sub.2-3 alkenyl, each optionally substituted by 1 to 5 halo;d) a group S(O).sub.n R.sup.7 wherein n=0,1,2 and R.sup.7 is C.sub.1-4 alkyl, halo or NR.sup.8 R.sup.9 wherein R.sup.8 and R.sup.9 are independently selected from hydrogen, C.sub.1-4 alkyl and C.sub.1-4 acyl;and a group e) NR.sup.8 R.sup.9 where R.sup.8 and R.sup.9 are as defined above;R.sup.X is hydrogen or an optionally substituted C.sub.1-8 alkyl or benzyl group, their preparation, pesticidal compositions containing them and their use against pests.
摘要翻译: 本申请公开了式(I)的杀虫活性化合物:Q(CH2)a(O)bQ1CR2 = CR2 = CR3CR4 = CR5 CXNR1Rx或其盐或杀虫剂,其中Q是任选取代的芳族单环或稠合双环体系 其中至少一个环是芳族的,或Q是二卤代乙烯基或R6-C 3BONDC,其中R6是C1-4烷基,三C1-4烷基甲硅烷基,卤素或氢; Q1是任选被一个或多个选自C 1-3烷基,卤素,C 1-3卤代烷基,C 2-3炔基或氰基的基团取代的1,2-环丙基环; 或为(CH 2)7; a = 0或1; b = 0或1; R 2,R 3,R 4和R 5相同或不同,至少一个为氢,其余独立地选自氢,卤素,C 1-4烷基或C 1-4卤代烷基; X是氧或硫; R1是任选被1-5个选自下列的取代基取代的苯基:a)C 1-4烷基,C 1-4烷氧基,苯氧基和亚甲二氧基,各自任选被1至5个卤素取代; b)卤素,氰基,硝基,甲酰基,C 1-5酰基; c)C2-3炔基,C2-3烯基,各自任选被1至5个卤素取代; d)基团S(O)n R 7,其中n = 0,1,2,R 7为C 1-4烷基,卤素或NR 8 R 9,其中R 8和R 9独立地选自氢,C 1-4烷基和C 1-4酰基; 和基团e)NR 8 R 9,其中R 8和R 9如上所定义; RX是氢或任选取代的C 1-8烷基或苄基,它们的制备方法,含有它们的杀虫组合物及其对害虫的用途。
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