Ester of (triarylphosphoranylidene)carbamic acid having diuretic and
ability to lower plasma renin properties
    81.
    发明授权
    Ester of (triarylphosphoranylidene)carbamic acid having diuretic and ability to lower plasma renin properties 失效
    具有利尿作用的(三芳基亚正膦基)氨基甲酸酯和降低血浆肾素性质的能力

    公开(公告)号:US4767749A

    公开(公告)日:1988-08-30

    申请号:US888613

    申请日:1986-07-23

    CPC分类号: C07F9/5355

    摘要: Novel triarylphosphinimide derivatives having the formula ##STR1## wherein R.sub.1, R.sub.2 and R.sub.3 are each at the ortho or meta position, represent mono- or disubstituents and are selected from the group consisting of hydrogen, alkyl(C.sub.1 -C.sub.3), alkoxy(C.sub.1 -C.sub.3), trifluoromethyl and halogen; and R.sub.4 is selected from the group consisting of alkyl(C.sub.1 -C.sub.3), alkenyl(C.sub.2 -C.sub.3), alkynyl(C.sub.2 -C.sub.4), cycloalkyl(C.sub.3 -C.sub.5), cycloalkyl(C.sub.3 -C.sub.6)methyl, 4-oxopentyl, 3-tetrahydrofuranyl, 2,3-dihydro-1H-inden-1-yl, 1-alkyl(C.sub.1 -C.sub.3)cyclopentyl, trans-2-alkyl(C.sub.1 -C.sub.3)cyclopentyl, trans-2-alkoxy(C.sub.1 -C.sub.3)cyclopentyl, 1-cyclopropylethyl, 2-methylcyclopropylmethyl, dicyclopropylmethyl, 2-, 3- or 4-pyridinylmethyl, 2-cyclopenten-1-yl, tetrahydro-2H-pyran-4-yl and cis and trans-2-methoxycyclohexyl; with the proviso that when R.sub.4 is alkyl(C.sub.1 -C.sub.3), R.sub.1, R.sub.2 and R.sub.3 may not each be hydrogen ##STR2## wherein R.sub.1, R.sub.2 and R.sub.3 are each at the ortho or meta position and are selected from hydrogen and alkyl(C.sub.1 -C.sub.3), and X is an acid addition salt; processes for producing them, compositions containing them, and methods for using them in mammals to effect diuresis; to lower plasma renin levels and to increase cardiac contractility.

    摘要翻译: 具有式“IMAGE”的新型三芳基膦酰亚胺衍生物,其中R 1,R 2和R 3各自为邻或间位,代表单取代或未取代的,并且选自氢,烷基(C1-C3),烷氧基(C1- C3),三氟甲基和卤素; 并且R 4选自烷基(C 1 -C 3),烯基(C 2 -C 3),炔基(C 2 -C 4),环烷基(C 3 -C 5),环烷基(C 3 -C 6)甲基,4-氧代戊基, (C 1 -C 3)环戊基,反式-2-烷基(C 1 -C 3)环戊基,反式-2-烷氧基(C 1 -C 3)环戊基 ,1-环丙基甲基,2-甲基环丙基甲基,二环丙基甲基,2-,3-或4-吡啶基甲基,2-环戊烯-1-基,四氢-2H-吡喃-4-基和顺式和反式-2-甲氧基环己基; 条件是当R 4是烷基(C 1 -C 3)时,R 1,R 2和R 3可以不是氢。其中R 1,R 2和R 3各自在邻位或间位,并且选自氢和烷基(C1 -C 3),X是酸加成盐; 生产它们的方法,含有它们的组合物,以及在哺乳动物中使用它们以产生利尿的方法; 降低血浆肾素水平并增加心脏收缩力。

    Multi-ring fluorinated carbamates with textiles soil repellent activity
    87.
    发明授权
    Multi-ring fluorinated carbamates with textiles soil repellent activity 失效
    多环氟化氨基甲酸酯具有纺织品防污性能

    公开(公告)号:US4534770A

    公开(公告)日:1985-08-13

    申请号:US674398

    申请日:1984-11-23

    申请人: Michael G. Kelly

    发明人: Michael G. Kelly

    摘要: Multi-ring fluorinated carbamates are disclosed which have excellent anti-soiling properties, durability and resistance to laundering. The compounds are represented by the formula ##STR1## wherein R.sub.f is a fluorinated radical. Compositions containing at least 10% of such compounds are also disclosed, as well as polyester and nylon fibers having such compounds incorporated therein.

    摘要翻译: 公开了具有优异的防污性能,耐久性和耐洗涤性的多环氟化氨基甲酸酯。 化合物由式(Ⅰ)表示,其中Rf是氟化基团。 还公开了含有至少10%的这类化合物的组合物,以及掺入其中的这种化合物的聚酯和尼龙纤维。

    Liquid diphenylmethane diisocyanate compositions
    88.
    发明授权
    Liquid diphenylmethane diisocyanate compositions 失效
    液体二苯基甲烷二异氰酸酯组合物

    公开(公告)号:US4490300A

    公开(公告)日:1984-12-25

    申请号:US538054

    申请日:1983-09-30

    CPC分类号: C08G18/8019 C07C263/18

    摘要: The invention is directed to a process for the production of an isocyanate which is both stable and liquid at room temperature comprising reacting pure diphenylmethane diisocyanate or crude diphenylmethane diisocyanate with a diol of the formula, ##STR1## wherein R is a C.sub.2 to a C.sub.5 aliphatic radical, at a temperature of from 20.degree. to 110.degree. C., in a ratio such that the resultant product has an isocyanate group content of from 20 to 30%, by weight and to the products produced therefrom.

    摘要翻译: 本发明涉及一种在室温下稳定和液体的异氰酸酯的制备方法,包括使纯二苯基甲烷二异氰酸酯或粗二苯基甲烷二异氰酸酯与下式的二醇反应,其中R是C 2至C 5脂族 自由基,以20至110℃的温度,使得所得产物的异氰酸酯基含量为20-30重量%,以及由其制备的产物。

    Carbaminic acid esters with herbicidal properties
    90.
    发明授权
    Carbaminic acid esters with herbicidal properties 失效
    具有除草性质的氨基甲酸酯

    公开(公告)号:US4426222A

    公开(公告)日:1984-01-17

    申请号:US337003

    申请日:1982-01-04

    CPC分类号: A01N47/22

    摘要: Novel carbaminic acid phenyl esters of the general formula ##STR1## are described, in which R.sub.1 is C.sub.1 -C.sub.2 -alkoxy-C.sub.1 -C.sub.2 -alkyl, di-C.sub.1 -C.sub.2 -alkoxy-C.sub.1 -C.sub.2 -alkyl, cyano-C.sub.1 -C.sub.2 -alkyl, halogen-C.sub.1 -C.sub.2 -alkyl, phenyl-C.sub.1 -C.sub.2 -alkyl, 1,3-dioxolan-2-yl-methyl, 2-methyl-1,3-dioxolan-4-yl-methyl, 2,2-dimethyl-1,3-dioxolan-4-yl-methyl or aminocarbonylmethyl;R.sub.2 is phenyl optionally mono- or disubstituted by one or more substituents selected from the group consisting of halogen, methyl and methoxy; andR.sub.3 is C.sub.1 -C.sub.8 alkyl, C.sub.2 -C.sub.8 alkenyl, cyclopropyl or trichloromethyl, or R.sub.1 is methyl or ethyl, R.sub.2 is .alpha.-cyanobenzyl or 1-cyano-2-phenylethyl and R.sub.3 is ethyl.

    摘要翻译: 描述了通式为“IMAGE”的新型氨基甲酸苯酯,其中R 1为C 1 -C 2烷氧基-C 1 -C 2烷基,二-C 1 -C 2烷氧基-C 1 -C 2烷基,氰基-C 1 -C 2 - 烷基,卤素-C 1 -C 2 - 烷基,苯基-C 1 -C 2 - 烷基,1,3-二氧戊环-2-基 - 甲基,2-甲基-1,3-二氧戊环-4-基 - 甲基,2,2 - 二甲基-1,3-二氧戊环-4-基 - 甲基或氨基羰基甲基; R2是任选被一个或多个选自卤素,甲基和甲氧基的取代基单取代或二取代的苯基; 且R 3为C 1 -C 8烷基,C 2 -C 8烯基,环丙基或三氯甲基,或R 1为甲基或乙基,R 2为α-氰基苄基或1-氰基-2-苯基乙基,且R 3为乙基。