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    Fungicidal compositions and methods of use employing pyrimidine derivatives
    2.
    发明授权
    Fungicidal compositions and methods of use employing pyrimidine derivatives 失效
    杀真菌组合物和使用嘧啶衍生物的使用方法

    公开(公告)号：US5468747A

    公开(公告)日：1995-11-21

    申请号：US352858

    申请日：1994-12-02

    申请人： John M. Clough ,  Christopher R. A. Godfrey ,  Ian T. Streeting ,  Rex Cheetham

    发明人： John M. Clough ,  Christopher R. A. Godfrey ,  Ian T. Streeting ,  Rex Cheetham

    IPC分类号： A01N43/54 ,  C07D239/52 ,  C07D401/12 ,  A61K31/535 ,  A01N59/02 ,  A01N59/20

    CPC分类号： C07D401/12 ,  A01N43/54 ,  C07D239/52

    摘要： Compounds having the formula (I): ##STR1## in which any two of K, L and M are nitrogen and the other is CE; X and Y are independently hydrogen, halogen, C.sub.1-4 alkyl, C.sub.3-6 cycloalkyl, C.sub.2-4 alkenyl, C.sub.2-4 alkynyl, C.sub.2-4 alkynyloxy, phenyl, benzyloxy, cyano, isocyano, isothiocyanato, nitro, NR.sup.1 R.sup.2, NR.sup.1 OR.sup.2,N.sub.3, NHCOR.sup.1, NR.sup.1 CO.sub.2 R.sup.2, NHCONR.sup.1 R.sup.2, N.dbd.CHNR.sup.1 R.sup.2, NHSO.sub.2 R.sup.1, OR.sup.1, OCOR.sup.1, OSO.sub.2 R.sup.1, SR.sup.1, SOR.sup.1, SO.sub.2 R.sup.1, SO.sub.2 OR.sup.1, SO.sub.2 NR.sup.1 R.sup.2, COR.sup.1, CR.sup.1 .dbd.NOR.sup.2, CHR.sup.1 CO.sub.2 R.sup.2, CO.sub.2 R.sup.1, CONR.sup.1 R.sup.2, CSNR.sup.1 R.sup.2, CH.sub.3 O.sub.2 C.C:CH.OCH.sub.3, 1-(imidazol-1-yl)vinyl, a 5-membered heterocyclic ring containing one, two or three nitrogen heteroatoms, or a 5- or 6-membered heterocyclic ring containing one or two oxygen or sulphur hetero-atoms, optionally a nitrogen heteroatom and optionally one or two oxo or thioxo substituents; or X and Y, when ortho to one another, join to form a 5- or 6-membered aliphatic or aromatic ring optionally containing one or two oxygen, sulphur or nitrogen atoms or one, two or three nitrogen atoms; A, B, D, E, G, U and V are independently hydrogen, halogen, C.sub.1-4 alkyl C.sub.1-4 alkoxy, cyano, nitro or trifluoromethyl; and R.sup.1 and R.sup.2 are independently hydrogen, C.sub.1-4 alkyl, C.sub.2-4 alkenyl or phenyl; the aliphatic moieties of any of theforegoing being optionally substituted with one or more of halogen, cyano, OR.sup.1, SR.sup.1, NR.sup.1 R.sup.2, SiR.sup.1.sub.3 or OCOR.sup.1 and the phenyl moieties of any of the foregoing being optionally substituted with one or more of halogen, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, nitro or cyano. The compounds are useful as fungicides.

    摘要翻译： 具有式（I）的化合物：其中K，L和M中的任一个为氮，另一个为CE; X和Y独立地是氢，卤素，C 1-4烷基，C 3-6环烷基，C 2-4烯基，C 2-4炔基，C 2-4炔氧基，苯基，苄氧基，氰基，异氰基，异硫氰酸酯基，硝基，NR1R2，NR1OR2， N3，NHCOR1，NR1CO2R2，NHCONR1R2，N = CHNR1R2，NHSO2R1，OR1，OCOR1，OSO2R1，SR1，SOR1，SO2R1，SO2OR1，SO2NR1R2，COR1，CR1 = NOR2，CHR1CO2R2，CO2R1，CONR1R2，CSNR1R2，CH3O2C.C：CH。 OCH 3，1-（咪唑-1-基）乙烯基，含有一个，两个或三个氮杂原子的5元杂环，或含有一个或两个氧或硫杂原子的5或6元杂环，任选地 氮杂原子和任选的一个或两个氧代或硫代取代基; 或X和Y，当彼此邻接时，连接形成任选地含有一个或两个氧，硫或氮原子或一个，两个或三个氮原子的5-或6-元脂族或芳族环; A，B，D，E，G，U和V独立地为氢，卤素，C 1-4烷基C 1-4烷氧基，氰基，硝基或三氟甲基; 并且R 1和R 2独立地是氢，C 1-4烷基，C 2-4链烯基或苯基; 任何前述的脂族部分任选被一个或多个卤素，氰基，OR 1，SR 1，NR 1 R 2，SiR 13或OCOR 1取代，任何前述的苯基部分任选被一个或多个卤素，C 1-4 烷基，C 1-4烷氧基，硝基或氰基。 这些化合物可用作杀真菌剂。

    Pyrimidine derivatives useful as fungicides
    5.
    发明授权
    Pyrimidine derivatives useful as fungicides 失效
    吡咯烷酮衍生物有效用作杀真菌剂

    公开(公告)号：US5059605A

    公开(公告)日：1991-10-22

    申请号：US506790

    申请日：1990-04-10

    申请人： John M. Clough ,  Christopher R. A. Godfrey ,  Ian T. Streeting

    发明人： John M. Clough ,  Christopher R. A. Godfrey ,  Ian T. Streeting

    IPC分类号： A01N43/54 ,  C07D20060101 ,  C07D401/12 ,  C07D401/14 ,  C07D413/14 ,  C07D417/14

    CPC分类号： C07D401/12 ,  A01N43/54

    摘要： Fungicidal compounds having the formula (I): ##STR1## in which any two of K, L and M are nitrogen and the other is CE; X and Y are independently hydrogen, halogen, C.sub.1-4 alkyl, C.sub.3-6 cycloalkyl, C.sub.2-4 alkenyl, C.sub.2-4 alkynyl, C.sub.2-4 alkenyloxy, C.sub.2-4 alkynyloxy, phenyl, benzyloxy, cyano, isocyano, isothiocyanato, nitro, NR.sup.1 R.sup.2, NR.sup.1 OR.sup.2, N.sub.3, NHCOR.sup.1, NR.sup.1 CO.sub.2 R.sup.2, NHCONR.sup.1 R.sup.2, N.dbd.CHNR.sup.1 R.sup.2, NHSO.sub.2 R.sup.1, OR.sup.1, OCOR.sup.1, OSO.sub.2 R.sup.1, SR.sup.1, SOR.sup.1, SO.sub.2 R.sup.1, SO.sub.2 OR.sup.1, SO.sub.2 NR.sup.1 R.sup.2, COR.sup.1, CR.sup.1 .dbd.NOR.sup.2, CHR.sup.1 CO.sub.2 R.sup.2, CO.sub.2 R.sup.2, CO.sub.2 R.sup.1, CONR.sup.1 R.sup.2, CSNR.sup.1 R.sup.2, CH.sub.3 O.sub.2 C.C:CH.OCH.sub.3, 1-(imidazol-1-yl)vinyl, a 5-membered heterocyclic ring containing one, two or three nitrogen heteroatoms, or a 5- or 6-membered heterocyclic ring containing one or two oxygen or sulphur heteroatoms, optionally a nitrogen heteroatom and optionally one or two oxo or thioxo substituents; or X and Y, when ortho to one another, join to form a 5- or 6-membered aliphatic or aromatic ring optionally containing one or two oxygen, sulphur or nitrogen atoms or one, two or three nitrogen or sulphur atoms; A, B, E, G and U are independently hydrogen, halogen, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, cyano, nitro or trifluoromethyl; and R.sup.1 and R.sup.2 are independently hydrogen, C.sub.1-4 alkyl, C.sub.2-4 alkenyl or phenyl; the aliphatic moieties of any of the foregoing being optionally substituted with one or more of halogen, cyano, OR.sup.1, SR.sup.1, NR.sup.1 R.sup.2, SiR.sup.1.sub.3 or OCOR.sup.1 and the phenyl moieties of any of the foregoing being optionally substituted with one or more of halogen, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, nitro or cyano; and their pyridine N-oxides and N-alkyl pyridinium salts.

    Pyrimidine derivatives and their use as fungicidal agents
    6.
    发明授权
    Pyrimidine derivatives and their use as fungicidal agents 失效
    嘧啶衍生物及其作为杀真菌剂的用途

    公开(公告)号：US5229391A

    公开(公告)日：1993-07-20

    申请号：US739468

    申请日：1991-08-02

    申请人： John M. Clough ,  Christopher R. A. Godfrey ,  Ian T. Streeting

    发明人： John M. Clough ,  Christopher R. A. Godfrey ,  Ian T. Streeting

    IPC分类号： A01N43/54 ,  C07D401/12

    CPC分类号： C07D401/12 ,  A01N43/54

    摘要： Fungicidal compounds having the formula (I): ##STR1## in which any two of K, L and M are nitrogen and the other is CE; X and Y are independently hydrogen, halogen, C.sub.1-4 alkyl, C.sub.3-6 cycloalkyl, C.sub.2-4 alkenyl, C.sub.2-4 alkynyl, C.sub.2-4 alkenyloxy, C.sub.2-4 alkynyloxy, phenyl, benzyloxy, cyano, isocyano, isothiocyanato, nitro, NR.sup.1 R.sup.2, NR.sup.1 OR.sup.2, N.sub.3, NHCOR.sup.1, NR.sup.1 CO.sub.2 R.sup.2, NHCONR.sup.1 R.sup.2, N.dbd.CHNR.sup.1 R.sup.2, NHSO.sub.2 R.sup.1, OR.sup.1, OCOR.sup.1, OSO.sub.2 R.sup.1, SR.sup.1, SOR.sup.1, SO.sub.2 R.sup.1, SO.sub.2 OR.sup.1, SO.sub.2 NR.sup.1 R.sup.2, COR.sup.1, CR.sup.1 .dbd.NOR.sup.2, CHR.sup.1 CO.sub.2 R.sup.2, CO.sub.2 R.sup.1, CONR.sup.1 R.sup.2, CSNR.sup.1 R.sup.2, CH.sub.3 O.sub.2 C.C:CH.OCH.sub.3, 1-(imidazol-1-yl)vinyl, a 5-membered heterocyclic ring containing one, two or three nitrogen heteroatoms, or a 5- or 6-membered heterocyclic ring containing one or two oxygen or sulphur heteroatoms, optionally a nitrogen heteroatom and optionally one or two oxo or thioxo substituents; or X and Y, when ortho to one another, join to form a 5- or 6-membered aliphatic or aromatic ring optionally containing one or two oxygen, sulphur or nitrogen atoms or one, two or three nitrogen or sulphur atoms; A, B, E, G and U are independently hydrogen, halogen, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, cyano, nitro or trifluoromethyl; and R.sup.1 and R.sup.2 are independently hydrogen, C.sub.1-4 alkyl, C.sub.2-4 alkenyl or phenyl; the aliphatic moieties of any of the foregoing being optionally substituted with one or more of halogen, cyano, OR.sup.1, SR.sup.1, NR.sup.1 R.sup.2, SiR.sup.1.sub.3 or OCOR.sup.1 and the phenyl moieties of any of the foregoing being optionally substituted with one or more of halogen, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, nitro or cyano; and their pyridine N-oxides and N-alkyl pyridinium salts.

    摘要翻译： 具有式（I）的杀真菌化合物：其中K，L和M中的任一个为氮，另一个为CE; X和Y独立地是氢，卤素，C 1-4烷基，C 3-6环烷基，C 2-4烯基，C 2-4炔基，C 2-4链烯氧基，C 2-4炔氧基，苯基，苄氧基，氰基，异氰基，异硫氰酸根合，硝基 ，NR1R2，NR1OR2，N3，NHCOR1，NR1CO2R2，NHCONR1R2，N = CHNR1R2，NHSO2R1，OR1，OCOR1，OSO2R1，SR1，SOR1，SO2R1，SO2OR1，SO2NR1R2，COR1，CR1 = NOR2，CHR1CO2R2，CO2R1，CONR1R2，CSNR1R2，CH3O2C C：CH.OCH 3，1-（咪唑-1-基）乙烯基，含有一个，两个或三个氮杂原子的5元杂环，或含有一个或两个氧或硫的5-或6-元杂环 杂原子，任选的氮杂原子和任选的一个或两个氧代或硫代取代基; 或X和Y，当彼此邻接时，连接形成任选地含有一个或两个氧，硫或氮原子或一个，两个或三个氮或硫原子的5-或6-元脂族或芳族环; A，B，E，G和U独立地为氢，卤素，C 1-4烷基，C 1-4烷氧基，氰基，硝基或三氟甲基; 并且R 1和R 2独立地是氢，C 1-4烷基，C 2-4链烯基或苯基; 前述任何一个的脂肪族部分任选被一个或多个卤素，氰基，OR 1，SR 1，NR 1 R 2，SiR 13或OCOR 1取代，并且前述任何一个的苯基部分任选被一个或多个卤素， 4烷基，C 1-4烷氧基，硝基或氰基; 和它们的吡啶N-氧化物和N-烷基吡啶鎓盐。

    Fungicidal aromatic pyrimidinyl oxime ethers
    7.
    发明授权
    Fungicidal aromatic pyrimidinyl oxime ethers 失效
    杀真菌抗真菌药

    公开(公告)号：US5206245A

    公开(公告)日：1993-04-27

    申请号：US736168

    申请日：1991-07-26

    申请人： John M. Clough ,  Christopher R. A. Godfrey ,  Ian T. Streeting ,  Rex Cheetham ,  Paul J. de Fraine

    发明人： John M. Clough ,  Christopher R. A. Godfrey ,  Ian T. Streeting ,  Rex Cheetham ,  Paul J. de Fraine

    IPC分类号： A01N43/54 ,  C07D239/52 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12

    CPC分类号： C07D401/12 ,  A01N43/54 ,  C07D239/52 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/10 ,  C07D417/12

    摘要： Fungicidal compounds having the formula (I): ##STR1## in which any two of K, L and M are nitrogen and the other is CE; X and Y are independently hydrogen, halogen, C.sub.1-4 alkyl, C.sub.3-6 cycloalkyl, C.sub.2-4 alkenyl, C.sub.2-4 alkynyl, C.sub.2-4 alkynyloxy, phenyl, benzyloxy, cyano, isocyano, thiocyanato, isothiocyanato, nitro, NR.sup.1 R.sup.2, NR.sup.1 OR.sup.2, N.sub.3, NHCOR.sup.1, NR.sup.1 CO.sub.2 R.sup.2, NHCONR.sup.1 R.sup.2, N.dbd.CHNR.sup.1 R.sup.2, NHSO.sub.2 R.sup.1, OR.sup.1, OCOR.sup.1, OSO.sub.2 R.sup.1, SR.sup.1, SOR.sup.1, SO.sub.2 R.sup.1, SO.sub.2 OR.sup.1,SO.sub.2 NR.sup.1 R.sup.2, COR.sup.1, CR.sup.1 .dbd.NOR.sup.2, CHR.sup.1 CO.sub.2 R.sup.2, CO.sub.2 R.sup.1, CONR.sup.1 R.sup.2, CSNR.sup.1 R.sup.2, CH.sub.3 O.sub.2 C.C:CH.OCH.sub.3, 1-(imidazol-1-yl)vinyl, a 5-membered heterocyclic ring containing one, two or three nitrogen heteroatoms, or a 5- or 6-membered heterocyclic ring containing one or two oxygen or sulphur heteroatoms, optionally a nitrogen heteroatom and optionally one or two oxo or thioxo substituents; or X and Y, when ortho to one another, join to form a 5- or 6-membered aliphatic or aromatic ring optionally containing one or two oxygen, sulphur or nitrogen atoms or one, two or three nitrogen atoms; A, Q, D, E, G, U and V are independently hydrogen, halogen (especially fluorine and chlorine), C.sub.1-4 alkyl (especially methyl), C.sub.1-4 alkoxy (especially methoxy), cyano, nitro or trifluoromethyl; and R.sup.1 and R.sup.2 are independently hydrogen, C.sub.1-4 alkyl, C.sub.2-4 alkenyl or phenyl; the aliphatic moieties of any of the foregoing being optionally substituted with one of more of halogen, cyano, OR.sup.1, SR.sup.1, NR.sup.1 R.sup.2, SiR.sup.1.sub.3 or OCOR.sup.1 and the phenyl moieties of any of the foregoing being optionally substituted with one or more of halogen, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, nitro or cyano.

    Benzoxazole, benzothiazole and benzimidazole derivatives as fungicides
    9.
    发明授权
    Benzoxazole, benzothiazole and benzimidazole derivatives as fungicides 失效
    苯并恶唑，苯并噻唑和苯并咪唑衍生物作为杀真菌剂

    公开(公告)号：US5491156A

    公开(公告)日：1996-02-13

    申请号：US196265

    申请日：1994-02-16

    申请人： Ian T. Streeting, deceased ,  Paul A. Worthington

    发明人： Ian T. Streeting, deceased ,  Paul A. Worthington

    IPC分类号： A01N43/52 ,  A01N43/74 ,  A01N43/76 ,  A01N43/78 ,  C07D235/26 ,  C07D263/58 ,  C07D277/68

    CPC分类号： C07D277/68 ,  A01N43/52 ,  A01N43/74

    摘要： ##STR1## Fungicidal compounds having general formula (I) and stereoisomers thereof, in which A, B, C and D are independently H, halo, C
    1-4 alkyl, C
    2-4 alkenyl, C
    2-4 alkynyl, C
    1-4 alkylthio, cyano, nitro, C
    1-4 haloalkyl, phenoxyobenzyl or benzyloxy, the phenyl moieties of any of the foregoing being optionally substituted with one or more of halo, C
    1-4 alkyl, C
    1-4 alkoxy, nitro or cyano; X is oxygen, sulphur or NR, in which R is H or C
    1-4 alkyl; and W is CH
    3 O.CH=C.CO.CH
    3 or CH
    3 O.N=C.CONR
    1 R
    2 , in which R
    1 and R
    2 are independently H or methyl.

    摘要翻译： PCT No.PCT / GB92 / 01860 Sec。 371日期：1994年2月16日 102（e）日期1994年2月16日PCT提交1992年10月12日PCT公布。 出版物WO93 / 08180 （I）具有通式（I）及其立体异构体的杀真菌化合物，其中A，B，C和D独立地为H，卤素，C 1-4烷基，C 2-4烯基， C 2-4炔基，C 1-4烷硫基，氰基，硝基，C 1-4卤代烷基，苯氧基苄基或苄氧基，任何前述的苯基部分任选被一个或多个卤素，C 1-4烷基，C 1-4烷氧基 ，硝基或氰基; X是氧，硫或NR，其中R是H或C 1-4烷基; 并且W是CH 3 O，CH = C.CO.CH 3或CH 3 O.N = C.CONR1R2，其中R1和R2独立地为H或甲基。