公开(公告)号：US4310677A

公开(公告)日：1982-01-12

申请号：US217453

申请日：1980-12-17

申请人： Gernot Reissenweber ,  Dietrich Mangold

发明人： Gernot Reissenweber ,  Dietrich Mangold

IPC分类号： C07C229/56 ,  C07C227/22 ,  C07C229/58 ,  C07C229/64 ,  C07C79/46 ,  C07C101/54

CPC分类号： C07C227/22

摘要： Alkyl anthranilates are prepared by reacting an isatin with an alkanol and hydrogen peroxide in the presence of an alkali metal alkanolate.The alkyl anthranilates obtainable by the process of the invention are valuable starting materials for the preparation of pesticides, dyes and drugs.

摘要翻译： 烷基邻氨基苯甲酸酯通过在碱金属链烷醇酯存在下使靛红与链烷醇和过氧化氢反应来制备。 通过本发明方法可获得的烷基邻氨基苯甲酸酯是制备农药，染料和药物的有价值的原料。

公开(公告)号：US4202987A

公开(公告)日：1980-05-13

申请号：US966424

申请日：1978-12-04

申请人： Jurgen Habermeier ,  Roland Moser ,  Wolfgang Seiz

发明人： Jurgen Habermeier ,  Roland Moser ,  Wolfgang Seiz

IPC分类号： C08G18/00 ,  C07C67/00 ,  C07C239/00 ,  C07C275/10 ,  C08G18/10 ,  C08G18/38 ,  C08G18/65 ,  C08G59/40 ,  C07C101/54 ,  C08G59/54

CPC分类号： C08G59/4021 ,  C07C275/10 ,  C08G18/10 ,  C08G18/3829

摘要： Novel bis-anthranilates are obtained by reacting 1 mol of a N,N'-bis-(hydroxyalkyl)-urea with 2 mols of isatoic anhydride. The novel bis-anthranilates are valuable chain extenders for polyurethanes and valuable crosslinking agents for polyurea and epoxide resins.

摘要翻译： 通过使1摩尔N，N'-双 - （羟基烷基） - 脲与2摩尔的丙酮酸酐反应获得新的双 - 邻氨基苯甲酸酯。 新型双 - 邻氨基苯甲酸酯是聚氨酯和聚脲和环氧树脂的有价值交联剂的有价值的增链剂。

公开(公告)号：US4160100A

公开(公告)日：1979-07-03

申请号：US669567

申请日：1976-03-23

申请人： John H. Sellstedt ,  Charles J. Guinosso ,  Albert J. Begany

发明人： John H. Sellstedt ,  Charles J. Guinosso ,  Albert J. Begany

IPC分类号： C07C245/08 ,  C07D257/04 ,  C07C101/54

CPC分类号： C07D257/04 ,  C07C245/08

摘要： Anti-allergic agents of aromatic and heterocyclic oxamic acid derivation present the following formula: ##STR1## in which A is a member selected from the group consisting of 2-thiazolyl, 2-pyridyl, 2-pyridyl-N-oxide, 6-(lower)alkyl-2-pyridyl, 3-cyano-2-pyridyl, 3-pyridyl, 4-pyridyl, 2-pyrimidinyl, 2-pyrazinyl, .alpha.-naphthyl, .beta.-naphthyl, phenyl, 2,6-di-chlorophenyl, and substituted phenyl moieties containing from one to three substituents in any of the 2,3,4 and 5 positions of the phenyl ring, independently selected from the group consisting of lower alkyl, lower alkylthio, lower alkylsulfinyl, lower alkoxy, hydroxy(lower)alkoxy, 2-(lower alkoxy oxalyloxy) ethoxy, benzyloxy, N-mono-and di-lower alkylamino(lower)alkoxy, halo, sulfamyl, polyhalo(lower)alkyl, carbamyl, N-lower alkylcarbamyl, nitro, mono-and di-lower alkylamino, phenylazo, carboxy, lower alkylcarbonyl, cyano, carb(lower)alkoxy, phenoxy(lower)alkoxy, lower alkoxyoxalamido and lower alkoxyoxalamidophenoxy radicals;B, when taken alone, is a member selected from the group consisting of --OH, lower alkoxy, --NH.sub.2, --NHOH, cyclohexyloxy and phenoxy; andY is a member selected from the group consisting of oxygen and when taken with B and the carbon atom to which they are attached, forms the moiety ##STR2##

公开(公告)号：US4104049A

公开(公告)日：1978-08-01

申请号：US734478

申请日：1976-10-20

申请人： Fritz Maurer ,  Hans-Jochem Riebel ,  Rolf Schroder ,  Klaus Lurssen

发明人： Fritz Maurer ,  Hans-Jochem Riebel ,  Rolf Schroder ,  Klaus Lurssen

IPC分类号： A01N35/04 ,  A01N20060101 ,  A01N37/44 ,  C07C20060101 ,  C07C67/00 ,  C07C69/76 ,  C07C227/00 ,  C07C227/18 ,  C07C229/60 ,  C07C231/00 ,  C07C231/12 ,  C07C233/12 ,  C07C237/30 ,  C07C255/30 ,  C07C255/53 ,  C07C255/58 ,  A01N5/00 ,  A01N9/20 ,  C07C101/54 ,  C07C121/78

CPC分类号： C07C255/00

摘要： Chlorine-substituted vinylaminobenzoic acid compounds of the formula ##STR1## in which R is hydroxyl, alkoxy of from 1 to 4 carbon atoms or monoalkylamino of from 1 to 3 carbon atoms,R.sup.1, r.sup.4 and R.sup.5 are individually selected from hydrogen and chlorine, provided that at least one of R.sup.1, R.sup.4 and R.sup.5 is chlorine,R.sup.2 is alkylcarbonyl of from 1 to 4 carbon atoms in the alkyl moiety or carbalkoxy of from 1 to 4 carbon atoms in the alkoxy moiety; andR.sup.3 is cyano, alkylcarbonyl of from 1 to 4 carbon atoms in the alkyl moiety or carbalkoxy of from 1 to 4 carbon atoms in the alkoxy moietyExhibit outstanding plate growth regulating effects, e.g., the inhibition of vegetative plant growth.

摘要翻译： 式中：R为羟基的氯取代的乙烯基氨基苯甲酸化合物，1至4个碳原子的烷氧基或1至3个碳原子的单烷基氨基，R1，R4和R5分别选自氢和氯， R1，R4和R5中的至少一个是氯，R2是烷基部分中具有1至4个碳原子的烷基羰基或烷氧基部分中具有1至4个碳原子的烷氧基; 并且R3是氰基，在烷基部分中具有1至4个碳原子的烷基羰基或在烷氧基部分中具有1至4个碳原子的烷氧基。参考实施例：植物生长调节效应，E.G.，植物生长发育的抑制。

公开(公告)号：US3974201A

公开(公告)日：1976-08-10

申请号：US339374

申请日：1973-03-08

申请人： Harmannus Boelens

发明人： Harmannus Boelens

IPC分类号： A23L27/29 ,  C11B9/00 ,  C07C101/54

CPC分类号： C11B9/0061 ,  A23L27/29

摘要： A perfumed material containing methyl-N-(2-methylpentylidene) anthranilate prepared by incorporating methyl-N-(2-methylpentylidene) anthranilate into mixtures usual for such purpose to impart a citrus like note thereto.

摘要翻译： 含有甲基-N-（2-甲基戊叉基）邻氨基苯甲酸酯的加香物质，其通过将甲基-N-（2-甲基戊基）邻氨基苯甲酸酯掺入通常用于赋予柑橘类似注释的混合物的混合物中。

公开(公告)号：US3910985A

公开(公告)日：1975-10-07

申请号：US48864374

申请日：1974-07-15

申请人： SHELL OIL CO

发明人： MONTIJN PAULUS P ,  MULDER ALBERTUS J

IPC分类号： C07C101/54

摘要： Nitrobenzenes are converted to the corresponding 4-nitroanilines by treatment with hydrogen and hydrogen fluoride in the presence of one or more of certain hydrogenation catalysts, liquid hydrogen fluoride and one or more of certain fluorine-containing acids.

摘要翻译： 在一种或多种某些氢化催化剂，液体氟化氢和一种或多种某些含氟酸的存在下，用氢气和氟化氢处理，将硝基苯转化为相应的4-硝基苯胺。

公开(公告)号：US3852333A

公开(公告)日：1974-12-03

申请号：US67742267

申请日：1967-10-23

申请人： PARKE DAVIS & CO

发明人： FISHER J

IPC分类号： C07D317/46 ,  C07C101/54

CPC分类号： C07D317/46

摘要： The Alpha -monoglycerides of N-( Alpha , Alpha , Alpha trifluoro-m-tolyl)anthranilic acid, N-(2,3-xylyl)anthranilic acid, and N-(2,6-dichloro-m-tolyl)anthranilic acid, useful as pharmacological agents having anti-inflammatory activity, and their production by (a) reacting one of the named anthranilic acids or a carboxylate salt thereof with a 3-halo-1,2propanediol; and (b) reacting a (1,3-dioxolan-4-yl)methyl ester of one of the named anthranilic acids with a strong acid, whereby the dioxolane ring is cleaved.

摘要翻译： N-（α，α，α-三氟 - 间甲苯基）邻氨基苯甲酸，N-（2,3-二甲苯基）邻氨基苯甲酸和N-（2,6-二氯 - 间甲苯基）邻氨基苯甲酸的α-单酸甘油酯 酸，可用作具有抗炎活性的药理学试剂，以及它们的生产通过（a）使命名的邻氨基苯甲酸或其羧酸盐与3-卤代-1,2-丙二醇反应; 和（b）使命名的邻氨基苯甲酸之一的（1,3-二氧戊环-4-基）甲酯与强酸反应，由此二氧戊环被切割。

公开(公告)号：US3819680A

公开(公告)日：1974-06-25

申请号：US4153470

申请日：1970-05-28

申请人： GAF CORP

发明人： WELCH E ,  YAMASHITA K ,  GRAHAM D

IPC分类号： C07C205/57 ,  C07C205/58 ,  C07C101/54 ,  C07C101/58

CPC分类号： C07C205/57 ,  C07C201/08 ,  C07C201/16 ,  C07C205/58 ,  C07C227/04 ,  C07C229/60

摘要： MONONITRO DERIVATIVES OF BENZOIC ACID, AND MONO- AND DICHLORO-BENZOIC ACID, ARE PRODUCED ECONOMICALLY AND IN GOOD YIELD BY NITRATION OF BENZOIC ACID OR CHLORO- OR DICHLORO-BENZOIC ACID ESTERS, PREFERABLY A LOWER ALKYL ESTER, WITH A MIXTURE OF NITRIC ACID AND SULFURIC ACID, OR OLEUM CONTAINING UP TO THE THEORETICAL OF SULFUR TRIOXIDE REQUIRED TO COMBINE WITH THE WATER FORMED IN NITRATION, AT A TEMPERATURE OF ABOUT 10* C, TO ABOUT 80* C. THE THUS PRODUCED MONONITRO ESTERS MAY BE HYDROLYZED TO THE CORRESPONDING MONONITRO-ACID.

公开(公告)号：US3590039A

公开(公告)日：1971-06-29

申请号：US3590039D

申请日：1968-12-09

申请人： GEIGY CHEM CORP

发明人： SALLMANN ALFRED ,  PFISTER RUDOLF

IPC分类号： A61K31/245 ,  D04B1/26 ,  C07C101/54

CPC分类号： A61K31/245 ,  D04B1/26 ,  Y10S514/825

摘要： N-(A,A,A,A'',A''-HEXAFLUORO-3,5-XYLYL)-ANTHRANILIC ACID AND PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF WITH A BASE ARE ACTIVE INGREDIENTS IN PHARMACEUTICAL COMPOSITIONS USEFUL FOR THE TREATMENT OF INFLAMMATORY DISEASES.

公开(公告)号：US3574723A

公开(公告)日：1971-04-13

申请号：US3574723D

申请日：1968-03-20

申请人： UNIVERSAL OIL PROD CO

发明人： LOUVAR JAMES J

IPC分类号： C07C51/00 ,  C07C63/04 ,  C07C101/54 ,  C07C101/56

CPC分类号： C07C51/00 ,  Y02P20/582 ,  C07C63/36 ,  C07C63/04

摘要： AROMATIC ACTING COMPOUNDS MAY BE CARBOXYLATED BY TREATING THE COMPOUND WITH A CARBOXYLIC ACID IN THE PRESENCE OF A CATALYST COMPRISING A PHOSPHORUS-CONTAINING ACID, A MINERAL ACID OR A FRIEDEL-CRAFTS METAL HALIDE TO FORM THE DESIRED CARBOXYLATED COMPOUNDS.