公开(公告)号：US4999440A

公开(公告)日：1991-03-12

申请号：US395233

申请日：1989-08-17

Applicant: Graham Holmwood ,  Udo Kraatz ,  Karl H. Buchel ,  Wilhelm Brandes ,  Stefan Dutzmann ,  Paul Reinecke

Inventor： Graham Holmwood ,  Udo Kraatz ,  Karl H. Buchel ,  Wilhelm Brandes ,  Stefan Dutzmann ,  Paul Reinecke

IPC: A01N43/653 ,  C07C15/44 ,  C07C25/24 ,  C07D249/08 ,  C07D303/06 ,  C07D303/08 ,  C07D303/22 ,  C07D303/34 ,  C07D303/36 ,  C07D521/00

CPC classification number: C07D249/08 ,  A01N43/653 ,  C07C15/44 ,  C07C25/24 ,  C07D231/12 ,  C07D233/56 ,  C07D303/08

Abstract: Fungicidal hydroxyalkyl-triazdyl derivatives of the formula ##STR1## in which R represents a radical of the formula --CH.sub.2 --CH(CH.sub.3).sub.2, --(CH.sub.2).sub.4 --CH.sub.3, --(CH.sub.2).sub.5 --CH.sub.3, --(CH.sub.2).sub.6 --CH.sub.3, ##STR2## Z represents halogen, alkyl with 1 to 4 carbon atoms, halogenoalkyl with 1 or 2 carbon atoms and 1 to 5 halogen atoms, halogenoalkoxy with 1 or 2 carbon atoms and 1 to 5 halogen atoms, halogenoalkylthio with 1 or 2 carbon atoms and 1 to 5 halogen atoms, phenyl or alkoximinimethyl with 1 to 4 carbon atoms in the alkoxy group andm represents the numbers 0, 1, 2 or 3,and addition products thereof with acids and metal salts. Intermediates of the formulas ##STR3## are also new.

公开(公告)号：US4952595A

公开(公告)日：1990-08-28

申请号：US249480

申请日：1988-09-26

Applicant: Graham Holmwood ,  Joachim Weissmuller ,  Wilhelm Brandes ,  Paul Reinecke

Inventor： Graham Holmwood ,  Joachim Weissmuller ,  Wilhelm Brandes ,  Paul Reinecke

IPC: A01N37/18 ,  A01N37/20 ,  A01N43/40 ,  A01N43/60 ,  A01N47/38 ,  C07D213/82 ,  C07D233/60 ,  C07D233/61 ,  C07D233/90 ,  C07D239/28 ,  C07D241/24 ,  C07D249/08 ,  C07D521/00

CPC classification number: C07D213/82 ,  A01N43/40 ,  A01N43/60 ,  A01N47/38 ,  C07D231/12 ,  C07D233/56 ,  C07D233/90 ,  C07D239/28 ,  C07D249/08

Abstract: Novel heterocyclic amide derivatives of the formula ##STR1## in which R.sup.1 represents alkyl, or represents alkenyl which has more than 2 carbon atoms and is optionally substituted by halogen, or represents alkinyl which has more than 2 carbon atoms and is optionally substituted by halogen, or represents alkoxyalkyl or alkylthioalkyl;R.sup.2 represents optionally substituted naphtyl, or represents optionally substituted tetrahydronaphthyl, or represents optionally substituted indanyl;A represents an alkylene bridge, or also an alkenylene bridge if X denotes a direct bond;X represents oxygen, sulphur or a direct bond;Y represents oxygen or sulphur;B represents imidazol-1-yl, pyridin-3-yl, pyrazin-2-yl, pyrimidin-5-yl, 1,2,4-triazol-1-yl or 1-methyl-imidazol-5-yl;and their acid addition salts and metal salt complexes, are outstandingly active as fungicides.

公开(公告)号：US4929738A

公开(公告)日：1990-05-29

申请号：US350064

申请日：1989-05-10

Applicant: Klaus Jelich ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

Inventor： Klaus Jelich ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

IPC: A01N43/56 ,  A01N43/74 ,  A01N43/80 ,  A01N43/82 ,  A01N43/824 ,  C07D231/46 ,  C07D231/48 ,  C07D261/08 ,  C07D333/28 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D409/14 ,  C07D413/12 ,  C07D417/12 ,  C07D417/14 ,  C07D307/16 ,  C07D307/46 ,  C07D333/24

CPC classification number: C07D401/12 ,  A01N43/56 ,  A01N43/74 ,  A01N43/80 ,  A01N43/82 ,  C07D231/48 ,  C07D261/08 ,  C07D333/28 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12

Abstract: Microbicidal substituted pyrazolin-5-ones of the formula ##STR1## in which R.sup.1 and R.sup.2 independently of one another each represent hydrogen, alkyl, alkenyl, alkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkoxycarbonyl, hydroxycarbonylalkyl, alkoxycarbonylalkyl, aminocarbonylalkyl, alkylaminocarbonylalkyl or dialkylaminocarbonylalkyl, or represent in each case optionally substituted oxiranylalkyl, aralkyl, heterocyclyl or aryl andHet represents an optionally substituted heterocyclic radial.Intermediates therefor of the formula ##STR2## in which R is alkyl, are also new.

公开(公告)号：US4921529A

公开(公告)日：1990-05-01

申请号：US18658

申请日：1987-02-25

Applicant: Reinhard Lantzsch ,  Brandes Wilhelm ,  Gerd Hansller ,  Paul Reinecke ,  Klaus Lurssen

Inventor： Reinhard Lantzsch ,  Brandes Wilhelm ,  Gerd Hansller ,  Paul Reinecke ,  Klaus Lurssen

IPC: A01N43/653 ,  C07C45/45 ,  C07C45/62 ,  C07C49/255 ,  C07D249/08 ,  C07D303/22 ,  C07D521/00

CPC classification number: C07D303/22 ,  A01N43/653 ,  C07C45/455 ,  C07C45/62 ,  C07C49/255 ,  C07D231/12 ,  C07D233/56 ,  C07D249/08

Abstract: New 2-hydroxyethyl-azole derivatives of the formula ##STR1## in which R represents optionally substituted phenyl,X represents hydrogen or halogen andY represents hydrogen or halogen, and acid addition salts and metal salt complexes thereof,as well as the use of the novel compounds as fungicides and plant growth regulants.New intermediates for the synthesis of the novel 2-hydroxyethyl-azole derivatives.

Abstract translation: 新的式（I）的2-羟乙基 - 唑衍生物，其中R表示任选取代的苯基，X表示氢或卤素，Y表示氢或卤素，以及其酸加成盐和金属盐络合物，以及 使用新型化合物作为杀真菌剂和植物生长调节剂。 用于合成新型2-羟乙基 - 唑衍生物的新中间体。

公开(公告)号：US4897410A

公开(公告)日：1990-01-30

申请号：US281128

申请日：1988-12-07

Applicant: Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke ,  Hans Scheinpflug ,  Graham Holmwood

Inventor： Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke ,  Hans Scheinpflug ,  Graham Holmwood

IPC: A01N47/04 ,  A01N35/08 ,  A01N37/00 ,  A01N43/653 ,  A01N43/66 ,  A01N43/78 ,  A01N43/80 ,  A01N43/84 ,  A01N43/90 ,  A01N47/02 ,  A01N47/14 ,  A01N47/18 ,  A01N47/30 ,  A01N47/32 ,  A01N47/38 ,  A01N47/44 ,  A01N55/02 ,  A01N57/14 ,  A01N59/02

CPC classification number: A01N47/14 ,  A01N43/653 ,  A01N43/66 ,  A01N47/02 ,  A01N47/32 ,  A01N59/02

Abstract: Synergistic fungicidal compositions comprising(i) a substituted 1-hydroxyethyl-triazole of the formula ##STR1## in which R.sup.1, R.sup.2, X, Y and A have various meanings, or addition products thereof with acids or metal salts, and(ii) at least one of(A) wettable sulphur,(B) a polyhalogenoalkylthio derivative,(C) a quanidine derivative,(D) an aromatic acid lactone,(E) a dithiocarbamate,(F) a benzimidazole derivative,(G) an imidazole or triazole derivative,(H) a phosphoric acid ester,(I) a tetrahydroquinoline derivative,(J) an S, N-heterocyclic compound,(K) a urea derivative,(L) a sulphonamide derivative,(M) a polyhydroxyether derivative,(N) a triazine derivative,(O) a copper-hydroxy quinoline complex,(P) an N-formula derivative,(Q) a morpholine derivative,(R) a quinoxaline derivative, and(S) a dicarboxamide derivative.

公开(公告)号：US4888349A

公开(公告)日：1989-12-19

申请号：US22454

申请日：1987-03-06

Applicant: Wilhelm Brandes ,  Helmut Kaspers ,  Paul Reinecke ,  Hans Scheinpflug ,  Wolfgang Kramer

Inventor： Wilhelm Brandes ,  Helmut Kaspers ,  Paul Reinecke ,  Hans Scheinpflug ,  Wolfgang Kramer

IPC: A01N43/50 ,  A01N43/52 ,  A01N43/64 ,  A01N43/653 ,  A01N43/707 ,  A01N43/828 ,  A01N43/90 ,  A01N47/02 ,  A01N47/08 ,  A01N47/16 ,  A01N47/32 ,  A01N59/20

CPC classification number: A01N47/08 ,  A01N43/653 ,  A01N43/707 ,  A01N43/90 ,  A01N47/02 ,  A01N47/16 ,  A01N59/20

Abstract: This invention involves methods and composition for treating fungi comprising a fungicidally effective amount of a mixture of (I) a 1,2,4-triazole derivative of a phenoxyether-ketone or phenoxyether-alkanol selected from the group consisting of ##STR1## and (II) the compound of the formula ##STR2## the weight ratio of I:II ranging from 0.02-50:1.

Abstract translation: 本发明涉及用于治疗真菌的方法和组合物，其包含杀真菌有效量的（I）苯氧基醚 - 酮或苯氧基醚 - 链烷醇的1,2,4-三唑衍生物的混合物，所述苯氧基醚 - 酮或苯氧基醚 - 烷醇选自由下列组成的组：IMA图像 和（II）式（I）化合物，其重量比I：II为0.02-50:1。

公开(公告)号：US4878939A

公开(公告)日：1989-11-07

申请号：US258108

申请日：1988-10-13

Applicant: Gerhard Jager ,  Manfred Jautelat ,  Wolfgang Kramer ,  Karl H. Buchel ,  Paul Reinecke ,  Wilhelm Brandes ,  Gerd Hanssler ,  Klaus Lurssen

Inventor： Gerhard Jager ,  Manfred Jautelat ,  Wolfgang Kramer ,  Karl H. Buchel ,  Paul Reinecke ,  Wilhelm Brandes ,  Gerd Hanssler ,  Klaus Lurssen

IPC: C07C43/225 ,  A01N43/50 ,  A01N43/653 ,  C07C41/00 ,  C07C45/00 ,  C07C49/167 ,  C07C49/175 ,  C07C67/00 ,  C07D233/60 ,  C07D249/08 ,  C07D521/00

CPC classification number: C07D231/12 ,  A01N43/50 ,  A01N43/653 ,  C07D233/56 ,  C07D249/08

Abstract: Azolyl ether ketones and alcohols of the formula ##STR1## in which R.sup.1 and R.sup.2 each independently represents alkyl with more than one carbon atom, orR.sup.1 represents dichloromethyl, trichloromethyl, chlorovinyl or dichlorovinyl, andR.sup.2 represents alkyl,R.sup.3 represents alkyl,A represents the keto group or a CH(OH) grouping,Z represents a nitrogen atom or the CH group,X represents oxygen or sulphur andAr represents optionally substituted phenyl,or addition products thereof with acids and metal salts, are active against fungi and in regulating the growth of plants. New intermediates therefor are also shown.

Abstract translation: 其中R 1和R 2各自独立地表示具有多于一个碳原子的烷基，或者R 1表示二氯甲基，三氯甲基，氯乙烯基或二氯乙烯基，并且R 2表示烷基，R 3表示烷基， 酮基或CH（OH）基，Z表示氮原子或CH基，X表示氧或硫，Ar表示任选取代的苯基，或其与酸和金属盐的加成产物对真菌有活性， 植物生长。 还显示了其新的中间体。

公开(公告)号：US4875928A

公开(公告)日：1989-10-24

申请号：US792089

申请日：1985-10-28

Applicant: Erik Regel ,  Klaus Bockmann ,  Karl H. Buchel ,  Klaus Lurssen ,  Wilhelm Brandes ,  Jorg Konze ,  Paul Reinecke

Inventor： Erik Regel ,  Klaus Bockmann ,  Karl H. Buchel ,  Klaus Lurssen ,  Wilhelm Brandes ,  Jorg Konze ,  Paul Reinecke

IPC: A01N43/50 ,  A01N43/653 ,  C07D233/60 ,  C07D249/08 ,  C07D333/00 ,  C07D403/06 ,  C07D405/06 ,  C07D409/06 ,  C07D521/00

CPC classification number: C07D231/12 ,  A01N43/50 ,  A01N43/653 ,  C07D233/56 ,  C07D249/08 ,  Y02P60/246

Abstract: Substituted azolylcyclopropyl-azolylmethyl-carbinol derivatives of the formula ##STR1## in which Ar is optionally substituted aryl or optionally substituted heteroaryl,R is hydrogen, alkyl, alkenyl, alkinyl, trialkylsilyl, optionally substituted phenylalkyl or an acyl radical, andX and Y each independently is a nitrogen atom or a CH group,and addition products thereof with acids and metal salts are effective in regulating plant growth and combating fungi. New intermediates are described, some of which are themselves active.

Abstract translation: 其中Ar是任选取代的芳基或任选取代的杂芳基，R是氢，烷基，烯基，炔基，三烷基甲硅烷基，任选取代的苯基烷基或酰基，以及X和Y各自独立地取代的具有式“IMAGE”的唑基环丙基 - 甲基 - 甲醇衍生物 独立地是氮原子或CH基团，其与酸和金属盐的加成产物在调节植物生长和对抗真菌中是有效的。 描述了新的中间体，其中一些本身是活性的。

公开(公告)号：US4864029A

公开(公告)日：1989-09-05

申请号：US192799

申请日：1988-05-11

Applicant: Klaus Jelich ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

Inventor： Klaus Jelich ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

IPC: A01N43/56 ,  A01N43/74 ,  A01N43/80 ,  A01N43/82 ,  A01N43/824 ,  C07D231/46 ,  C07D231/48 ,  C07D261/08 ,  C07D333/28 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D409/14 ,  C07D413/12 ,  C07D417/12 ,  C07D417/14

CPC classification number: C07D401/12 ,  A01N43/56 ,  A01N43/74 ,  A01N43/80 ,  A01N43/82 ,  C07D231/48 ,  C07D261/08 ,  C07D333/28 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12

Abstract: Microbicidal substituted pyrazolin-5-ones of the formula ##STR1## in which R.sup.1 and R.sup.2 independently of one another each represent hydrogen, alkyl, alkenyl, alkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkoxycarbonyl, hydroxycarbonylalkyl, alkoxycarbonylalkyl, aminocarbonylalkyl, alkyllaminocarbonylalkyl or dialkylaminocarbonylalkyl, or represent in each case optionally substituted oxiranylalkyl, aralkyl, heterocyclyl or aryl andHet represents an optionally substituted heterocyclic radical.Intermediates therefor of the formula ##STR2## in which R is alkyl, are also new.

Abstract translation: 其中R1和R2彼此独立地表示氢，烷基，烯基，炔基，氰基烷基，羟基烷基，烷氧基烷基，烷硫基烷基，烷氧基羰基，羟基羰基烷基，烷氧基羰基烷基，氨基羰基烷基，烷基氨基羰基烷基或氨基羰基烷基， 二烷基氨基羰基烷基，或在每种情况下表示任选取代的环氧烷基烷基，芳烷基，杂环基或芳基，Het表示任选取代的杂环基。 其中R为烷基的式“IMAGE”的中间体也是新的。

公开(公告)号：US4845117A

公开(公告)日：1989-07-04

申请号：US204463

申请日：1988-06-09

Applicant: Stefan Dutzmann ,  Paul Reinecke ,  Hans Scheinpflug

Inventor： Stefan Dutzmann ,  Paul Reinecke ,  Hans Scheinpflug

IPC: A01N43/653

CPC classification number: A01N43/653

Abstract: The known compound 1-(4-chlorophenyl)-4,4-dimethyl-3-(1,2,4-triazol-1-yl-methyl)-pentan-3-ol of the formula ##STR1## in particularly suitable for combating Pseudocercosporella herpotrichoides.

Abstract translation: 将式（I）的已知化合物1-（4-氯苯基）-4,4-二甲基-3-（1,2,4-三唑-1-基 - 甲基） - 戊-3-醇在 特别适用于对抗假丝酵母（Pseudocercosporella herpotrichoides）。