Heteroaryl compounds used as pharmaceuticals
    31.
    发明授权
    Heteroaryl compounds used as pharmaceuticals 失效
    用作药物的杂芳基化合物

    公开(公告)号:US5786372A

    公开(公告)日:1998-07-28

    申请号:US771093

    申请日:1996-12-20

    CPC分类号: C07D405/12

    摘要: Compounds of formula (I), or pharmaceutically acceptable salts thereof are provided: ##STR1## in which X.sub.1 --(CH.sub.2).sub.x --X.sub.2 forms a 5-7 membered ring wherein: X.sub.1 is O or S; X.sub.2 is O, S or NR wherein R is hydrogen; x is 1, 2 or 3; R.sub.1 is hydrogen, amino, halo, C.sub.1-6 alkyl, hydroxy or C.sub.1-6 alkoxy; R.sub.2 is hydrogen, halo, C.sub.1-6 alkyl, C.sub.1-6 alkoxy, nitro, amino or C.sub.1-6 alkylthio; R.sub.3 is hydrogen, halo, C.sub.1-6 alkyl, C.sub.1-6 alkoxy or amino; R.sub.4 and R.sub.5 are independently hydrogen or C.sub.1-6 alkyl; Y is NH; Z is of sub-formula (a): ##STR2## wherein --(CH.sub.2).sub.n.sup.1 is attached at carbon; and n.sup.1 is 0, 1, 2, 3 or 4; q is 0, 1, 2 or 3; R.sub.a is (CH.sub.2).sub.n.sup.2 --R.sub.7 wherein n.sup.2 is 2 or 3 and R.sub.7 is selected from cyano, hydroxyl, C.sub.1-6 alkoxy, phenoxy, C(O)C.sub.1-6 alkyl, COC.sub.6 H.sub.5, --CONR.sub.8 R.sub.9, NR.sub.8 COR.sub.9, SO.sub.2 NR.sub.8 R.sub.9 or NR.sub.8 SO.sub.2 R.sub.9 wherein R.sub.8 and R.sub.9 are hydrogen or C.sub.1-6 alkyl; and R.sub.6 is hydrogen or C.sub.1-6 alkyl. The present compounds exhibit 5-HT.sub.4 receptor antagonist activity.

    摘要翻译: 提供式(I)化合物或其药学上可接受的盐:其中X 1 - (CH 2)x -X 2形成5-7元环,其中:X 1是O或S; X 2是O,S或NR,其中R是氢; x为1,2或3; R 1是氢,氨基,卤素,C 1-6烷基,羟基或C 1-6烷氧基; R 2是氢,卤素,C 1-6烷基,C 1-6烷氧基,硝基,氨基或C 1-6烷硫基; R3是氢,卤素,C1-6烷基,C1-6烷氧基或氨基; R4和R5独立地是氢或C1-6烷基; Y是NH; Z是亚式(a):其中 - (CH 2)n1连接在碳上; n1为0,1,2,3或4; q为0,1,2或3; R a是(CH 2)n R 2,其中n 2是2或3,R 7选自氰基,羟基,C 1-6烷氧基,苯氧基,C(O)C 1-6烷基,COC 6 H 5,-CONR 8 R 9,NR 8 COR 9,SO 2 NR 8 R 9或NR 8 SO 2 R 9 R8和R9是氢或C1-6烷基; R6是氢或C1-6烷基。 本发明化合物显示5-HT 4受体拮抗剂活性。

    Conceptual map showing the windows of a complex task
    32.
    发明授权
    Conceptual map showing the windows of a complex task 失效
    显示复杂任务窗口的概念图

    公开(公告)号:US5594857A

    公开(公告)日:1997-01-14

    申请号:US610797

    申请日:1996-03-04

    CPC分类号: G06Q10/109 G06F3/0489

    摘要: A visual conceptual map is displayed on each window of a program for accomplishing a complex task. In the preferred embodiment, the conceptual map includes all of the program's action dialogs and the potential paths between the action dialogs. The action dialog corresponding to the current window, the action dialogs that can presently be selected from the current window, and the other action dialogs are visually distinguished from each other. In addition, the potential paths from the action dialog corresponding to the current window to the action dialogs that may presently be selected from the current window are visually distinguished from the other potential paths.

    摘要翻译: 在程序的每个窗口上显示视觉概念图,以完成复杂任务。 在优选实施例中,概念图包括所有程序的动作对话和动作对话之间的潜在路径。 对应于当前窗口的动作对话框,当前可以从当前窗口选择的动作对话框和其他动作对话框在视觉上彼此区分开。 此外,从当前窗口对应的动作对话框到目前可以从当前窗口中选择的动作对话框的潜在路径与其他潜在路径视觉区分开。

    Method and system for the display of scheduling information for users
within a single viewport
    33.
    发明授权
    Method and system for the display of scheduling information for users within a single viewport 失效
    用于在单个视口内显示用户的调度信息的方法和系统

    公开(公告)号:US5528745A

    公开(公告)日:1996-06-18

    申请号:US330483

    申请日:1994-10-28

    摘要: A method and system in a data processing system for providing an intuitive display of scheduling information for multiple users within a single viewport. Each user is associated with scheduled events which may be displayed along a time line within a viewport on a display within the data processing system. Selection regions are determined within the viewport. Selection regions may be associated with scheduled events, users, or user specified time periods along the time line. Scheduling information is associated with each selection region. While a user is continuously selecting one of the selection regions, the scheduling information associated with the selection region being selected by the user is temporarily displayed. Once the user ceases selecting the selection region, the scheduling information disappears.

    摘要翻译: 数据处理系统中的方法和系统,用于在单个视口内为多个用户提供直观显示调度信息。 每个用户与可以在数据处理系统内的显示器上的视口内的时间线上显示的调度事件相关联。 选择区域在视口内确定。 选择区域可以与时间线上的调度事件,用户或用户指定的时间段相关联。 调度信息与每个选择区域相关联。 当用户连续地选择选择区域之一时,临时显示与用户选择的选择区域相关联的调度信息。 一旦用户停止选择选择区域,调度信息就会消失。

    Metal oxide films
    34.
    发明授权
    Metal oxide films 失效
    金属氧化膜

    公开(公告)号:US4065600A

    公开(公告)日:1977-12-27

    申请号:US144541

    申请日:1971-05-18

    IPC分类号: C23C14/00 H01B1/00 H01B5/14

    CPC分类号: C23C14/0036 H01B1/00

    摘要: In a method of depositing a transparent electrically conductive metal oxide coating by reactive sputtering onto the surface of a substrate, the substrate is supported, in spaced relationship with a cathode which is to be sputtered, in a vacuum chamber containing an atmosphere comprising an inert gas and a controlled oxygen concentration at a selected total pressure. The substrate is heated prior to sputtering to a selected elevated temperature, and reactive sputtering is caused by applying a selected negative potential relative to the substrate. The oxygen in the atmosphere is provided and maintained at a selected concentration, and the heating of said substrate is controlled during sputtering to maintain the substrate temperature substantially constant at the selected temperature during substrate heating caused by sputtering. The selected values of the oxygen concentration substrate temperature, vacuum chamber pressure, and cathode potential are so chosen that the deposited coating is haze-free, and its specific electrical resistivity lies at or close to the minimum of the curve which is obtained by plotting specific electrical resistivity against oxygen concentration while maintaining the substrate temperature, vacuum chamber pressure and cathode potential all constant at the selected values. Glass articles with stable, transparent and haze-free coatings having acceptable resistance are produced by the method.

    摘要翻译: 在通过反应性溅射将透明导电金属氧化物涂层沉积到衬底的表面上的方法中,衬底与包含惰性气体的气氛的真空室以与溅射的阴极隔开的关系被支撑 以及在所选择的总压力下的受控氧浓度。 将衬底在溅射之前被加热到选定的升高温度,并且通过相对于衬底施加选择的负电位而引起反应性溅射。 提供并保持大气中的氧气并保持选定的浓度,并且在溅射期间控制所述衬底的加热,以在由溅射引起的衬底加热期间使衬底温度基本保持恒定。 选择的氧浓度衬底温度,真空室压力和阴极电位的值被选择为沉积的涂层是无雾的,并且其特定的电阻率位于或接近曲线的最小值,其通过绘制具体的 保持基板温度,真空室压力和阴极电位的电阻率相对于氧气浓度全部恒定在所选择的值。 通过该方法产生具有可接受电阻的具有稳定,透明和无雾度的涂层的玻璃制品。

    Metal oxide films
    35.
    发明授权
    Metal oxide films 失效
    金属氧化膜

    公开(公告)号:US4006070A

    公开(公告)日:1977-02-01

    申请号:US220899

    申请日:1972-01-26

    摘要: A substantially uniform, transparent, electrically conducting, metal oxide film (e.g. of indium/tin oxide) can be deposited on to a substrate such as glass of large lateral dimensions, e.g. a windscreen for an aircraft or a land vehicle, by low-pressure reactive sputtering from a cathode of the metal, using an atmosphere of oxygen and another gas or gases (preferably an inert gas) at reduced pressure, by providing access for the sputtering atmosphere to penetrate into the whole of the working space between the cathode and the substrate so as to maintain a substantial degree of uniformity in the oxygen concentration in the working space. Access for the atmosphere may be provided by means of passages extending through the cathode assembly, by dividing the cathode assembly into parallel strips separated by gaps, and the atmosphere may be supplied direct to the working space through such gaps. Relative movement is effected between the cathode assembly and the substrate, e.g. by reciprocating the parallel strips of the divided cathode in the direction perpendicular to their length.

    摘要翻译: 可以将基本上均匀的,透明的,导电的金属氧化物膜(例如铟/锡氧化物)沉积到衬底上,例如大的侧向尺寸的玻璃,例如 用于飞机或地面车辆的挡风玻璃,通过从金属阴极的低压反应溅射,使用氧气和另一种气体(优选惰性气体)在减压下,通过提供溅射气氛的通路 以渗透到阴极和基板之间的整个工作空间中,以便保持工作空间中的氧浓度的显着程度的均匀性。 可以通过延伸穿过阴极组件的通道,通过将阴极组件划分为由间隙分开的平行条带来提供气氛,并且气氛可以通过这些间隙直接供应到工作空间。 在阴极组件和衬底之间进行相对运动,例如, 通过使垂直于其长度的方向使分割阴极的平行条带往复运动。

    Anchor device
    37.
    发明授权

    公开(公告)号:US10779515B1

    公开(公告)日:2020-09-22

    申请号:US16007159

    申请日:2018-06-13

    摘要: The present invention is an anchor for an artificial structure for attracting fish within a body of water. The structure is comprised of a base and has a central attachment post, a central column configured to secure to the attachment post, and a protective plate.

    Method And Apparatus For Creating A Composite Video From Multiple Sources
    38.
    发明申请
    Method And Apparatus For Creating A Composite Video From Multiple Sources 审中-公开
    用于从多个源创建复合视频的方法和装置

    公开(公告)号:US20140086562A1

    公开(公告)日:2014-03-27

    申请号:US14095830

    申请日:2013-12-03

    IPC分类号: G11B27/02 G11B27/10 H04N5/76

    摘要: The present system provides a method for a group of people, related or otherwise, to record an event on separate recording devices. The video from those recording devices can then be synchronized with each other. After synchronization, a composite movie is automatically generated using extracts from all or some of the video recordings. The composite movie is returned to a mobile device from where it can be shared and broadcast or re-edited inside the device.

    摘要翻译: 本系统提供了一组相关或其他方式在单独的记录装置上记录事件的方法。 然后可以将来自那些记录设备的视频彼此同步。 同步后,使用全部或部分视频录像的摘录自动生成复合影片。 复合电影返回到移动设备,从该设备可以共享并在设备中进行广播或重新编辑。

    Method and particle analyzer for determining a broad particle size distribution
    39.
    发明授权
    Method and particle analyzer for determining a broad particle size distribution 有权
    用于确定宽粒度分布的方法和粒子分析仪

    公开(公告)号:US08681215B2

    公开(公告)日:2014-03-25

    申请号:US13097285

    申请日:2011-04-29

    IPC分类号: H04N7/18

    摘要: A method and a particle analyzer are provided for determining a particle size distribution of a liquid sample including particles of a lower size range, particles of an intermediate size range, and particles of an upper size range. A dark-field image frame is captured in which the particles of the lower size range and the particles of the intermediate size range are resolved, and a bright-field image frame is captured in which the particles of the intermediate size range and the particles of the upper size range are resolved. Absolute sizes of the particles of the intermediate size range and the particles of the upper size range are determined from the bright-field image frame. Calibrated sizes of the particles of the lower size range are determined from the dark-field image frame by using the particles of the intermediate size range as internal calibration standards.

    摘要翻译: 提供了一种方法和粒子分析器,用于确定包括较小尺寸范围的颗粒,中等尺寸范围的颗粒和大尺寸范围的颗粒的液体样品的粒度分布。 捕获暗场图像帧,其中分辨较小尺寸范围的颗粒和中等尺寸范围的颗粒,并且捕获亮场图像帧,其中中等尺寸范围的颗粒和颗粒的 上限范围解决。 从亮场图像帧确定中等尺寸范围的颗粒的绝对尺寸和较大尺寸范围的颗粒。 通过使用中等尺寸范围的颗粒作为内部校准标准,从暗视野图像帧确定较小尺寸范围的颗粒的校准尺寸。

    ABSOLUTE POSITION DETECTION
    40.
    发明申请
    ABSOLUTE POSITION DETECTION 审中-公开
    绝对位置检测

    公开(公告)号:US20140002642A1

    公开(公告)日:2014-01-02

    申请号:US13918704

    申请日:2013-06-14

    IPC分类号: G06T7/00

    摘要: A system for determining the absolute position of a first object with respect to a second object includes a scalar element attached to the first object and a measuring device attached to the second object. The scalar element comprises a series of coded regions. The coded region represents a number designating a position along an axis of the scalar element. The measuring device includes a two-dimensional optical sensor array configured to capture an image of a portion of the scalar element. The system also includes a processor configured to receive the image and determine an absolute position of the first object with respect to the second object based on at least one coded region of the series of coded regions.

    摘要翻译: 用于确定第一对象相对于第二对象的绝对位置的系统包括附接到第一对象的标量元素和附接到第二对象的测量装置。 标量元素包括一系列编码区域。 编码区域表示沿着标量元素的轴指定位置的数字。 测量装置包括被配置为捕获标量元件的一部分的图像的二维光学传感器阵列。 该系统还包括处理器,该处理器被配置为基于所述一系列编码区域的至少一个编码区域接收图像并确定第一对象相对于第二对象的绝对位置。