公开(公告)号：US4067720A

公开(公告)日：1978-01-10

申请号：US679334

申请日：1976-04-22

申请人： Jacques Perronnet ,  Laurent Taliani ,  Andre Teche

发明人： Jacques Perronnet ,  Laurent Taliani ,  Andre Teche

IPC分类号： A01N47/38 ,  C07D285/08 ,  A01N9/12

CPC分类号： C07D285/08 ,  C07C329/00

摘要： Novel thiadiazoles of the formula ##STR1## wherein R is selected from the group consisting of alkoxy of 1 to 8 carbon atoms, cycloalkyloxy of 3 to 7 carbon atoms, alkylthio of 1 to 8 carbon atoms optionally substituted with carbalkoxy of 2 to 5 carbon atoms, alkenylthio of 2 to 4 carbon atoms, ##STR2## and benzyloxy, benzylthio, benzyl and phenyl, all aryl being optionally substituted with 1 to 2 members of the group consisting of chlorine, bromine, alkyl of 1 to 3 carbon atoms and alkoxy of 1 to 3 carbon atoms, Z and Z.sub.1 are alkyl of 1 to 4 carbon atoms and R.sub.1 is selected from the group consisting of alkyl of 1 to 6 carbon atoms optionally substituted with a member of the group consisting of chlorine, bromine and alkyloxy of 1 to 4 carbon atoms, phenyl optionally substituted with 1 to 2 members of the group consisting of bromine, chlorine, alkyl of 1 to 3 carbon atoms and alkoxy of 1 to 3 carbon atoms, alkenyl of 2 to 4 carbon atoms optionally substituted with at least one member of the group consisting of chlorine and alkoxy of 1 to 3 carbon atoms, ##STR3## and carbalkoxy of 2 to 6 carbon atoms and X is selected from the group consisting of alkyl of 1 to 4 carbon atoms and alkenyl of 2 to 4 carbon atoms, both optionally substituted with at least one chlorine having herbicidal properties and novel intermediates.

摘要翻译： 式中，R选自碳原子数1〜8的烷氧基，碳原子数为3〜7的环烷氧基，碳原子数为1〜8的烷硫基，碳原子数2〜5的烷氧基的烷硫基的新颖噻唑，式 2至4个碳原子的链烯基硫基，苄氧基，苄硫基，苄基和苯基，所有芳基任选被1至2个由氯，溴，1至3个碳原子的烷基和烷氧基 1至3个碳原子的烷基，Z和Z 1为具有1至4个碳原子的烷基，并且R 1选自1-6个碳原子的烷基，任选被下列成员所取代：氯，溴和烷氧基 1至4个碳原子的苯基，任选被1至2个由溴，氯，1至3个碳原子的烷基和1至3个碳原子的烷氧基组成的组中任意取代的苯基，任选被 至少有一个成员 e为碳原子数为1〜3的烷氧基和碳原子数2〜6的烷氧基，X选自碳原子数为1〜4的烷基和碳原子数2〜4的烯基， 两者都任选被至少一种具有除草性的氯取代和新的中间体。

公开(公告)号：US3932433A

公开(公告)日：1976-01-13

申请号：US536424

申请日：1974-12-26

申请人： Jacques Perronnet ,  Laurent Taliani

发明人： Jacques Perronnet ,  Laurent Taliani

IPC分类号： A01N57/16 ,  A01P7/02 ,  A01P7/04 ,  C07F9/6539 ,  C07F9/6541 ,  C07D277/60

CPC分类号： C07F9/6541 ,  A01N57/16

摘要： Thiazole derivatives of the formula ##SPC1##Wherein A is alkylene of 3 to 5 carbon atoms optionally substituted with a member of the group consisting of =0 and ##EQU1## wherein R' is alkyl of 1 to 5 carbon atoms and R is alkyl of 2 to 3 carbon atoms having insecticidal and/or acaricidal properties and their preparation.

摘要翻译： 式WHEREIN A的噻唑衍生物是任选被0和O并原-C-OR'的成员任意取代的3至5个碳原子的亚烷基，其中R'是1至5个碳原子的烷基，R是烷基 具有2至3个具有杀虫和/或杀螨性质的碳原子及其制备。

公开(公告)号：US3988444A

公开(公告)日：1976-10-26

申请号：US627217

申请日：1975-10-30

申请人： Jacques Perronnet ,  Laurent Taliani

发明人： Jacques Perronnet ,  Laurent Taliani

IPC分类号： A01N57/16 ,  C07F9/6541 ,  A01N9/36

CPC分类号： A01N57/16 ,  C07F9/6541

摘要： Novel thiazole derivatives of the formula ##EQU1## wherein A is alkylene of 3 to 5 carbon atoms optionally substituted with a member of the group consisting of =0 and ##EQU2## wherein R' is alkyl of 1 to 5 carbon atoms and R is alkyl of 2 to 3 carbon atoms having insecticidal and/or acaricidal properties and their preparation.

摘要翻译： 式C的新型噻唑衍生物--- NS A平行平行平行或I CC-OP角度或S其中A是3至5个碳原子的亚烷基，其任选被= 0和O的平行的 - C-OR'，其中R'为1至5个碳原子的烷基，R为具有杀虫和/或杀螨性质的2至3个碳原子的烷基及其制备。

公开(公告)号：US3931175A

公开(公告)日：1976-01-06

申请号：US484774

申请日：1974-07-01

申请人： Jacques Perronnet ,  Laurent Taliani

发明人： Jacques Perronnet ,  Laurent Taliani

IPC分类号： C07D471/04 ,  A01N57/16 ,  C07F9/62 ,  C07F9/6561 ,  C07D237/26

CPC分类号： A01N57/16 ,  C07F9/6561

摘要： Substituted imidazo(1,2b)pyridazinyl esters having the formula ##SPC1##Wherein R.sub.1 is hydrogen or halogen, Y is oxygen or sulfur, X is alkyl having 1 to 6 carbon atoms and Z is hydrogen or --COOR' wherein R, is alkyl having 1 to 6 carbon atoms; as well as the process of preparation, insecticidal compositions containing the same, and the method of using the insecticidal compositions. The products of the invention are useful in agriculture to combat and control insects.

摘要翻译： 具有下式的取代的咪唑并（1,2b）哒嗪基酯，其中R 1是氢或卤素，Y是氧或硫，X是具有1至6个碳原子的烷基，Z是氢或-COOR'，其中R 1是具有1至 6个碳原子; 以及制备方法，含有该杀虫组合物的杀虫组合物和使用杀虫组合物的方法。 本发明的产品在农业中可用于对抗和控制昆虫。

公开(公告)号：US4108993A

公开(公告)日：1978-08-22

申请号：US729763

申请日：1976-10-05

申请人： Claude Bonne ,  Jacques Perronnet ,  Andre Teche

发明人： Claude Bonne ,  Jacques Perronnet ,  Andre Teche

IPC分类号： A61K8/00 ,  A61K8/49 ,  A61K31/535 ,  A61Q5/00 ,  A61Q19/00 ,  C07C275/64 ,  C07D273/04 ,  A01N9/00 ,  A01N9/22

CPC分类号： C07D273/04 ,  C07C275/64 ,  C07C323/00

摘要： Antiandrogenic compositions comprising an effective amount of at least one compound of the formula ##STR1## wherein X and Y are individually selected from the group consisting of hydrogen, halogen, --CF.sub.3, --NO.sub.3 and alkylthio of 1 to 4 carbon atoms and R is selected from the group consisting of hydrogen, alkyl of 1 to 6 carbon atoms, phenyl, benzyl and hydroxymethyl and an inert pharmaceutical carrier and a method of inducing antiandrogenic activity in warm-blooded animals as well as novel oxadiazines of formula I with the proviso that when R is other than benzyl or hydroxymethyl at least one of X and Y is alkylthio of 1 to 4 carbon atoms.

公开(公告)号：US4137068A

公开(公告)日：1979-01-30

申请号：US667992

申请日：1976-03-18

申请人： Jacques Perronnet ,  Jean-Pierre Demoute ,  Pierre Girault ,  Andre Teche

发明人： Jacques Perronnet ,  Jean-Pierre Demoute ,  Pierre Girault ,  Andre Teche

IPC分类号： A01N47/34 ,  C07C67/00 ,  C07C313/00 ,  C07C313/08 ,  C07C313/34 ,  C07D263/04 ,  A01N9/12 ,  C07C119/20

CPC分类号： C07C313/34

摘要： Novel ureas of the formula ##STR1## wherein A and B are chlorine or A is chlorine or hydrogen and B is --CF.sub.3, R and R.sub.1 are individually alkyl of 1 to 3 carbon atoms and R.sub.2 is alkyl of 1 to 6 carbon atoms optionally substituted with a halogen having herbicidal properties, particularly useful in cultivated grass crops and their preparation and use.

摘要翻译： 其中A和B为氯或A为氯或氢且B为-CF 3，R和R 1分别为1至3个碳原子的烷基和R 2为任选的1至6个碳原子的烷基的新颖的脲 被具有除草性的卤素取代，特别适用于栽培草作物及其制备和用途。

公开(公告)号：US4069319A

公开(公告)日：1978-01-17

申请号：US721373

申请日：1976-09-08

申请人： Jacques Perronnet ,  Laurent Taliani

发明人： Jacques Perronnet ,  Laurent Taliani

IPC分类号： A01N57/16 ,  C07D285/08 ,  C07F9/6539 ,  A61K31/425

CPC分类号： C07D285/08 ,  A01N57/16 ,  C07F9/65397

摘要： Novel thiadiazoles of the formula ##STR1## wherein R is alkyl of 1 to 3 carbon atoms, W is selected from the group consisting of oxygen and sulfur, X is selected from the group consisting of --O--, --S-- and ##STR2## R" is selected from the group consisting of hydrogen and alkyl of 1 to 3 carbon atoms, n is 1, 2, 3 or 4 and R' is selected from the group consisting of hydrogen, --CN, alkoxy of 1 to 3 carbon atoms, alkoxycarbonyl of 2 to 4 carbon atoms, alkenyl of 2 to 4 carbon atoms, phenyl optionally substituted with one member of the group consisting of halogen, alkyl of 1 to 3 carbon atoms and alkoxy of 1 to 3 carbon atoms or substituted with two members of the group consisting of halogen, alkyl of 1 to 3 carbon atoms and alkoxy of 1 to 3 carbon atoms, having insecticidal and nematocidal activity.

摘要翻译： 式I的新型噻二唑其中R是1至3个碳原子的烷基，W选自氧和硫，X选自-O - ， - S-和

公开(公告)号：US4000267A

公开(公告)日：1976-12-28

申请号：US589466

申请日：1975-06-23

申请人： Jacques Perronnet ,  Laurent Taliani

发明人： Jacques Perronnet ,  Laurent Taliani

IPC分类号： C07F9/6561 ,  A01N9/36

CPC分类号： C07F9/6561

摘要： Novel insecticidal and acaridicidal compositions containing organo-phosphorus compounds of the formula ##STR1## wherein R is selected from the group consisting of methine and nitrogen, R.sup.1 is selected from the group consisting of hydrogen, alkyl of 1 to 3 carbon atoms and NO.sub.2, R.sub.2 is selected from the group consisting of hydrogen, straight or branched alkyl of 1 to 3 carbon atoms, chlorine, bromine, alkoxycarbonyl of 2 to 4 carbon atoms, phenyl and thioalkyl of 1 to 4 carbon atoms, R.sub.3 is branched or straight chain alkyl of 1 to 3 carbon atoms and R.sub.4 is selected from the group consisting of straight and branched chain alkyl of 1 to 3 carbon atoms, alkoxy of 1 to 3 carbon atoms and ##STR2## wherein R.sub.5 and R.sub.6 are individually selected from the group consisting of hydrogen and branched and straight chain alkyl of 1 to 3 carbon atoms.

公开(公告)号：US3983129A

公开(公告)日：1976-09-28

申请号：US540381

申请日：1975-01-13

申请人： Jacques Perronnet ,  Laurent Taliani ,  Pierre Girault ,  Andre Poittevin

发明人： Jacques Perronnet ,  Laurent Taliani ,  Pierre Girault ,  Andre Poittevin

IPC分类号： A01N57/16 ,  A01N57/24 ,  C07F9/6539 ,  C07D261/12

CPC分类号： C07F9/6539 ,  A01N57/16 ,  A01N57/24

摘要： Novel 3-phosphoryloxy-isothiazoles of the formula ##SPC1##Wherein R is selected from the group consisting of alkyl of 1 to 3 carbon atoms, alkoxy of 1 to 3 carbon atoms and ##EQU1## R' and R" being individually SELECTED FROM THE GROUP CONSISTING OF HYDROGEN AND ALKYL OF 1 TO 3 CARBON ATOMS, R.sub.1 is alkyl of 1 to 3 carbon atoms, R.sub.2 is selected from the group consisting of hydrogen, alkyl of 1 to 5 carbon atoms, aryl of 6 to 10 carbon atoms, aralkyl of 7 to 12 carbon atoms, cyano, carbalkoxy of 2 to 4 carbon atoms and NHR'", and R'" is selected from the group consisting of hydrogen and aryl of 6 to 10 carbon atoms, R.sub.3 is selected from the group consisting of cyano, alkylthio of 1 to 4 carbon atoms, alkylsulfinyl of 1 to 4 carbon atoms, alkylsulfonyl of 1 to 4 carbon atoms, carbamoyl, carbalkoxy of 2 to 4 carbon atoms and ##EQU2## A and B are individually selected from the group consisting of hydrogen and alkyl of 1 to 3 carbon atoms and X is selected from the group consisting of oxygen and sulfur which have excellent insecticidal properties.

摘要翻译： 新颖的3-磷酰氧基 - 异噻唑，式WHEREIN R选自1至3个碳原子的烷基，1至3个碳原子的烷氧基和R'-N ANGLE，R“R'和R”为 单独选自含1至3个碳原子的氢和烷基的基团，R 1为1至3个碳原子的烷基，R 2选自氢，1至5个碳原子的烷基，6至10个的芳基 碳原子数为7〜12的芳烷基，氰基，2〜4个碳原子的烷氧基和NHR“'，R”'选自氢和6〜10个碳原子的芳基，R3为 选自氰基，1至4个碳原子的烷硫基，1至4个碳原子的烷基亚磺酰基，1至4个碳原子的烷基磺酰基，2至4个碳原子的氨基甲酰基，烷氧基烷氧基和A--SO 2 ANGLE，BA和B 分别选自氢和1至3个碳原子的烷基，X选自由以下组成的组 的氧和硫具有优异的杀虫性能。

公开(公告)号：US4155996A

公开(公告)日：1979-05-22

申请号：US944809

申请日：1978-09-22

申请人： Jacques Perronnet ,  Laurent Taliani

发明人： Jacques Perronnet ,  Laurent Taliani

IPC分类号： C07F9/6553 ,  A01N9/36 ,  C07F9/09 ,  C07F9/165

CPC分类号： C07F9/655345

摘要： Novel 3-(phosphoryloxy) or (phosphonyloxy)-thiophenes of the formula ##STR1## wherein R is alkyl of 1 to 4 carbon atoms, R.sub.1 is selected from the group consisting of alkyl of 1 to 4 carbon atoms, alkoxy of 1 to 4 carbon atoms and ##STR2## wherein R' and R" are individually selected from the group consisting of hydrogen and alkyl of 1 to 4 carbon atoms, R.sub.2 is selected from the group consisting of cyano, alkoxy carbonyl of 2 to 4 carbon atoms and ##STR3## wherein Z is selected from the group consisting of phenyl and alkyl of 1 to 4 carbon atoms, R.sub.3 is selected from the group consisting of alkyl of 1 to 6 carbon atoms, alkoxy of 1 to 6 carbon atoms, alkylthio of 1 to 6 carbon atoms, phenyl, morpholino, piperidinyl and alkoxy carbonyl of 2 to 4 carbon atoms and X is selected from the group consisting of oxygen and sulfur having pesticidal properties and their preparation.

摘要翻译： 新颖的3-（磷酰氧基）或（膦酰基氧基） - 噻吩类化合物其中R是1至4个碳原子的烷基，R 1选自1至4个碳原子的烷基，1至 4个碳原子和其中R'和R“分别选自氢和1至4个碳原子的烷基，R 2选自氰基，2至4个碳原子的烷氧基羰基 和其中Z选自苯基和1至4个碳原子的烷基，R 3选自1至6个碳原子的烷基，1至6个碳原子的烷氧基，1至6个碳原子的烷硫基， 2个碳原子的苯基，吗啉代，哌啶基和烷氧基羰基，X选自具有杀虫特性的氧和硫及其制备。