公开(公告)号：US20180139962A1

公开(公告)日：2018-05-24

申请号：US15575064

申请日：2016-05-19

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Julie GEIST ,  Lionel NICOLAS ,  Philippe RINOLFI ,  Jan Peter SCHMIDT ,  Tomoki TSUCHIYA

IPC: A01N43/56 ,  C07D333/12 ,  C07D333/16 ,  C07D333/20 ,  C07D333/22 ,  C07D333/24 ,  C07D401/12 ,  C07D409/12 ,  C07D409/14

CPC classification number: A01N43/56 ,  C07D333/12 ,  C07D333/16 ,  C07D333/20 ,  C07D333/22 ,  C07D333/24 ,  C07D401/12 ,  C07D409/12 ,  C07D409/14

Abstract: The invention relates to fungicidal N-cycloalkyl-N-{[ortho-(1-substituted-cycloalkyl)heteroaryl]methyl}carboxamides and their thiocarbonyl derivatives of formula (I), their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions, and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

公开(公告)号：US20160326120A1

公开(公告)日：2016-11-10

申请号：US15101380

申请日：2014-12-04

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Julie GEIST ,  Lionel NICOLAS ,  Philippe RINOLFI ,  Jan-Peter SCHMIDT ,  Tomoki TSUCHIYA ,  Jean-Pierre VORS ,  Ulrike WACHENDORFF-NEUMANN

IPC: C07D231/12 ,  C07D249/06 ,  C07D307/38 ,  C07D263/32 ,  C07C211/27 ,  C07C217/48 ,  C07F7/08 ,  C07C255/46 ,  C07C47/54 ,  C07C47/55 ,  C07C47/575 ,  C07C22/04 ,  A01N43/56 ,  A01N43/647 ,  A01N43/10 ,  A01N43/76 ,  A01N33/04 ,  A01N55/00 ,  A01N37/34 ,  A01N35/04 ,  C07D307/54

CPC classification number: C07D231/12 ,  A01N33/04 ,  A01N35/04 ,  A01N37/34 ,  A01N43/10 ,  A01N43/56 ,  A01N43/647 ,  A01N43/76 ,  A01N55/00 ,  C07C22/04 ,  C07C47/54 ,  C07C47/55 ,  C07C47/575 ,  C07C211/27 ,  C07C217/48 ,  C07C255/46 ,  C07C2601/02 ,  C07D231/14 ,  C07D231/16 ,  C07D233/28 ,  C07D249/06 ,  C07D263/32 ,  C07D307/38 ,  C07D307/54 ,  C07F7/0803

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-{[2-(1-substitutedcycloalkyl)phenyl]methylene} carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

Abstract translation: 本发明涉及杀真菌N-环烷基-N - {[2-（1-取代环烷基）苯基]亚甲基]甲酰胺衍生物及其硫代羰基衍生物，其制备方法及其制备中间体化合物，它们用作杀真菌剂，特别是在 使用这些化合物或其组合物的杀真菌组合物和控制植物病原性真菌的方法。

公开(公告)号：US20170247345A1

公开(公告)日：2017-08-31

申请号：US15314446

申请日：2015-05-27

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Günter HÖMBERGER ,  Mark James FORD ,  Andreas HÜGEL ,  Tomoki TSUCHIYA

IPC: C07D261/04 ,  A01N43/80

CPC classification number: C07D261/04 ,  A01N43/80

Abstract: The present invention relates to a novel process for preparing dihydroisoxazole derivatives.

公开(公告)号：US20160316752A1

公开(公告)日：2016-11-03

申请号：US15100966

申请日：2014-12-04

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Julie GEIST ,  Lionel NICOLAS ,  Philippe RINOLFI ,  Jan-Peter SCHMIDT ,  Tomoki TSUCHIYA ,  Jean-Pierre VORS ,  Ulrike WACHENDORFF-NEUMANN

IPC: A01N43/56 ,  C07C47/575 ,  C07D231/16 ,  C07C47/546 ,  C07C47/55 ,  C07C25/18

CPC classification number: A01N43/56 ,  C07C25/18 ,  C07C47/546 ,  C07C47/55 ,  C07C47/575 ,  C07C2601/02 ,  C07D231/16

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-{[2-(1-substitutedcycloalkyl)phenyl]methylene} carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions

Abstract translation: 本发明涉及杀真菌N-环烷基-N - {[2-（1-取代环烷基）苯基]亚甲基}甲酰胺衍生物及其硫代羰基衍生物，其制备方法及其制备中间体化合物，它们用作杀真菌剂，特别是在 使用这些化合物或其组合物的杀真菌组合物和控制植物病原性真菌的方法

公开(公告)号：US20160262393A1

公开(公告)日：2016-09-15

申请号：US15029581

申请日：2014-10-15

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Pierre CRISTAU ,  Peter DAHMEN ,  Philippe DESBORDES ,  Tomoki TSUCHIYA ,  Ulrike WACHENDORFF-NEUMANN ,  Pierre-Yves COQUERON

IPC: A01N43/56 ,  A01N43/72 ,  A01N43/42 ,  A01N43/653

CPC classification number: A01N43/56 ,  A01N43/42 ,  A01N43/653 ,  A01N43/72

Abstract: The present invention relates to active compound combinations, in particular within a fungicide composition, which comprises (A) a N-cyclopropyl-N-[substituted-benzyl]-3-(difluoromethyl)-5-fluoro-1-methyl-1H-pyrazole-4-carboxamide or thiocarboxamide derivative and a further fungicidally active compound (B). Moreover, the invention relates to a method for curatively or preventively or eradicatively controlling the phytopathogenic fungi of plants or crops, to the use of a combination according to the invention for the treatment of seed, to a method for protecting a seed and not at least to the treated seed.

Abstract translation: 本发明涉及活性化合物组合物，特别是杀真菌剂组合物，其包含（A）N-环丙基-N- [取代 - 苄基] -3-（二氟甲基）-5-氟-1-甲基-1H- 吡唑-4-甲酰胺或硫代羧酰胺衍生物和另外的杀真菌活性化合物（B）。 此外，本发明涉及一种方法，用于根据或预防或根除地控制植物或作物的植物病原真菌，根据本发明的组合用于种子的处理，用于保护种子的方法，至少不是至少 对待处理的种子。

公开(公告)号：US20160244433A1

公开(公告)日：2016-08-25

申请号：US15028004

申请日：2014-10-07

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Philippe DESBORDES ,  Philippe RINOLFI ,  Tomoki TSUCHIYA

IPC: C07D403/06 ,  A01N61/00 ,  C07D405/14 ,  A01N43/56 ,  C07D401/06 ,  A01N43/36 ,  C07D405/06 ,  C07D417/06 ,  A01N43/78 ,  A01N43/647 ,  C07D409/06

CPC classification number: C07D403/06 ,  A01N43/36 ,  A01N43/56 ,  A01N43/647 ,  A01N43/78 ,  A01N61/00 ,  C07D207/06 ,  C07D211/12 ,  C07D401/06 ,  C07D405/04 ,  C07D405/06 ,  C07D405/14 ,  C07D409/06 ,  C07D417/06

Abstract: The present invention relates to fungicidal N-hetarylcarbonyl-2-(benzocycloalken-1-yl)piperidines or pyrrolidines of formula (I), and their thiocarbonyl derivatives, wherein A represents a carbo-linked, unsaturated or partially saturated, 5-membered heterocyclyl group that can be substituted by up to four groups R that can be the same or different; T represents 0 or S; n represents 1 or 2; m represents 1, 2 or 3; p represents 1, 2, 3 or 4, L1 and L2 independently represent CZ4Z5, NZ6, 0, S, S(O) or S(0)2; and R and Z1-Z6 are as defined in the claims; their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

Abstract translation: 本发明涉及式（I）的杀真菌N-叔丁基羰基-2-（苯并环烯烃-1-基）哌啶或吡咯烷及其硫代羰基衍生物，其中A表示碳连接的不饱和或部分饱和的5元杂环基 可以被最多四个可以相同或不同的R基团取代的基团; T表示0或S; n表示1或2; m表示1,2或3; p表示1,2,3或4，L1和L2独立地表示CZ4Z5，NZ6,0，S，S（O）或S（0）2; 并且R和Z1-Z6如权利要求中所定义; 它们的制备方法和用于其制备的中间体化合物，它们用作杀真菌剂，特别是以杀真菌剂的形式和用于使用这些化合物或其组合物控制植物病原性真菌的方法。

公开(公告)号：US20190029255A1

公开(公告)日：2019-01-31

申请号：US16054744

申请日：2018-08-03

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Julie GEIST ,  Lionel NICOLAS ,  Philippe RINOLFI ,  Jan-Peter SCHMIDT ,  Tomoki TSUCHIYA ,  Jean-Pierre VORS ,  Ulrike WACHENDORFF-NEUMANN

IPC: A01N43/56 ,  C07C47/575 ,  C07C47/55 ,  C07D231/16 ,  C07C25/18 ,  C07C47/546

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-{[2-(1-substituted cycloalkyl)phenyl]methylene} carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

公开(公告)号：US20160198713A1

公开(公告)日：2016-07-14

申请号：US14914230

申请日：2014-08-26

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Stefan HILLEBRAND ,  Matthias RIEDRICH ,  Sebastian HOFFMANN ,  Mark James FORD ,  Joachim TELSER ,  Mazen ES-SAYED ,  Guenter HOEMBERGER ,  Pierre WASNAIRE ,  Ulrike WACHENDORFF-NEUMANN ,  Tomoki TSUCHIYA ,  Valerie TOQUIN

IPC: A01N43/80 ,  A01N43/82 ,  A01N43/78 ,  C07D417/14

CPC classification number: A01N43/80 ,  A01N43/78 ,  A01N43/82 ,  C07D417/14

Abstract: Malonic ester derivatives of the formula (I) in which the symbols A1, A2, Y, R10, p, X, R2, G, Q, L2 and R1 are each as defined in the description, and salts, metal complexes and N-oxides of the compounds of the formula (I), and the use thereof for controlling phytopathogenic harmful fungi and processes for preparing compounds of the formula (I).

Abstract translation: 其中符号A1，A2，Y，R10，p，X，R2，G，Q，L2和R1各自如说明书中所定义的式（I）的丙二酸酯衍生物，以及盐，金属络合物和N- 式（I）化合物的氧化物及其用于控制​​植物病原性有害真菌的用途及其制备式（I）化合物的方法。

公开(公告)号：US20180146670A1

公开(公告)日：2018-05-31

申请号：US15575292

申请日：2016-05-19

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Julie GEIST ,  Lionel NICOLAS ,  Philippe RINOLFI ,  Jan Peter SCHMIDT ,  Tomoki TSUCHIYA

IPC: A01N43/56 ,  C07D409/12 ,  C07D401/12

CPC classification number: A01N43/56 ,  C07D401/12 ,  C07D409/12

Abstract: The invention relates to fungicidal N-cycloalkyl-N-{[ortho-(1-substituted-cycloalkyl)heteroaryl]methyl}carboxamides and their thiocarbonyl analogs of formula (I), their process of preparation, their use as fungicides, particularly in the form of fungicidal compositions, and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions. A represents a carbo-linked, unsaturated or partially saturated, optionally substituted 5-membered heterocyclyl group; T represents O or S; Z1 represents an optionally substituted C3-C7-cycloalkyl; p represents 1-5; B1 represents a carbo-linked, unsaturated, monocyclic or fused bicyclic 5-, 6-, 8-, 9-, 10-membered heterocyclyl ring, wherein the dotted line between the two adjacent carbons represents a single bond, a double bond or an aromatic bond.

公开(公告)号：US20160255836A1

公开(公告)日：2016-09-08

申请号：US15029220

申请日：2014-10-15

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Philippe DESBORDES ,  Philippe RINOLFI ,  Tomoki TSUCHIYA ,  Julie GEIST ,  Lionel NICOLAS

IPC: A01N43/56 ,  C07D403/14 ,  C07D405/14 ,  C07D417/14 ,  A01N43/54 ,  A01N43/647 ,  A01N43/10 ,  A01N43/36 ,  C07D401/14 ,  C07D409/14 ,  A01N43/78

CPC classification number: A01N43/56 ,  A01N43/10 ,  A01N43/36 ,  A01N43/54 ,  A01N43/647 ,  A01N43/78 ,  C07D333/18 ,  C07D333/38 ,  C07D401/14 ,  C07D403/14 ,  C07D405/14 ,  C07D409/14 ,  C07D417/14

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-(biheterocyclylmethylene)carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

Abstract translation: 本发明涉及杀真菌N-环烷基-N-（双杂环亚甲基）甲酰胺衍生物及其硫代羰基衍生物，其制备方法及其制备中间体化合物，其用作杀真菌剂，特别是杀真菌组合物和控制方法 使用这些化合物或其组合物的植物致病真菌。