公开(公告)号：US11427564B2

公开(公告)日：2022-08-30

申请号：US16624636

申请日：2018-06-22

Applicant: Nippon Soda Co., Ltd.

Inventor： Keita Sakanishi ,  Hikaru Aoyama ,  Norifumi Sakiyama ,  Takao Iwasa ,  Daisuke Ushijima ,  Maki Matsui

IPC: C07D401/04 ,  C07D401/14 ,  C07D403/04 ,  C07D403/14 ,  A01N43/82

Abstract: A compound represented by a formula (I) or a salt thereof: wherein A1 represents CR1 or a nitrogen atom; A2 represents CR2 or a nitrogen atom; A3 represents CR3 or a nitrogen atom, provided that two or more of A1 to A3 do not represent nitrogen atoms at the same time; R1, R2 and R3 each independently represent a hydrogen atom or the like; B1 represents CH or a nitrogen atom; R4 represents a substituted or unsubstituted C1-6 alkyl group or the like; R5 represents a substituted or unsubstituted C1-6 alkylthio group or the like; and R6 represents a substituted or unsubstituted C1-6 alkyl group or the like.

公开(公告)号：US12037326B2

公开(公告)日：2024-07-16

申请号：US17500866

申请日：2021-10-13

Applicant: Nippon Soda Co., Ltd.

Inventor： Keita Sakanishi ,  Takao Iwasa ,  Hikaru Aoyama ,  Norifumi Sakiyama ,  Daisuke Ushijima ,  Maki Matsui ,  Tomomi Kobayashi

IPC: C07D401/14 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A61K31/506 ,  A61P31/10 ,  A61P31/14 ,  C07D233/64 ,  C07D401/04 ,  C07D403/04 ,  C07D403/10 ,  C07D403/14 ,  C07D413/10

CPC classification number: C07D403/14 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A61K31/506 ,  A61P31/10 ,  A61P31/14 ,  C07D233/64 ,  C07D401/04 ,  C07D401/14 ,  C07D403/04 ,  C07D403/10 ,  C07D413/10

Abstract: A compound represented by Formula (I), or a salt thereof:




wherein, R1 represents an unsubstituted or substituted C1-6 alkylthio group, or the like; A1 represents a nitrogen atom or CH; A2 represents a nitrogen atom or CR2; R2 and R3 each independently represents a hydrogen atom, an unsubstituted or substituted C6-10 aryl group, an unsubstituted or substituted 3- to 6-membered heterocyclyl group, or the like; B1 and B2 each independently represents a nitrogen atom or CR5, with the proviso that B1 and B2 do not represent CR5 at the same time, wherein R5 represents a hydrogen atom, an unsubstituted or substituted C1-6 alkyl group, or the like; R4 represents an unsubstituted or substituted C1-6 alkyl group, or the like, and R4 binds to any one of nitrogen atoms forming an imidazole ring or a triazole ring; and Ar represents an unsubstituted or substituted C6-10 aryl group or the like.

公开(公告)号：US12180178B2

公开(公告)日：2024-12-31

申请号：US17271531

申请日：2019-09-02

Applicant: NIPPON SODA CO., LTD.

Inventor： Keita Sakanishi ,  Hikaru Aoyama ,  Daisuke Ushijima ,  Takao Iwasa ,  Norifumi Sakiyama ,  Maki Matsui

IPC: C07D401/04 ,  A01N43/50 ,  A01N43/54 ,  A01N43/653 ,  C07D233/64 ,  C07D401/14

Abstract: A heteroaryl azole compound of the following formula (II): an N-oxide compound, stereoisomer, tautomer or hydrate thereof, or a salt of any of these compounds. In the formula (II), R1 represents a substituted or unsubstituted C1-6 alkylthio group or the like; B1 represents a nitrogen atom or CR2; R2 represents a hydrogen atom, a substituted or unsubstituted C1-6 alkyl group or the like; R3 represents a hydrogen atom, a substituted or unsubstituted C1-6 alkyl group or the like; R represents a substituted or unsubstituted C1-6 alkyl group or the like; A represents a carbon atom or a nitrogen atom; X represents a substituted or unsubstituted C1-6 alkyl group or the like; n represents a number of chemically acceptable X, and is an integer of 0 to 2; and X is the same or different when n is 2.

公开(公告)号：US12195442B2

公开(公告)日：2025-01-14

申请号：US17286888

申请日：2019-10-23

Applicant: Nippon Soda Co., Ltd.

Inventor： Keita Sakanishi ,  Norifumi Sakiyama ,  Hikaru Aoyama ,  Maki Matsui ,  Takao Iwasa ,  Tomomi Kobayashi ,  Daisuke Ushijima ,  Keita Azuma ,  Masanori Sumino ,  Yasuhiko Ashikari ,  Kotaro Shibayama ,  Riho Taguchi

IPC: C07D401/04 ,  A01N43/50

Abstract: An object of the present invention is to provide a (hetero)aryl imidazole compound that is excellent in pest control activity, particularly, insecticidal activity and/or acaricidal activity, is excellent in safety, and may be industrially advantageously synthesized. The (hetero)aryl imidazole compound of the present invention is a compound represented by the formula (I) an N-oxide compound, stereoisomer, tautomer or hydrate thereof or a salt of any of these compounds. In the formula (I), B1 represents a nitrogen atom or CH; X represents a substituted or unsubstituted C3-8 cycloalkyl group; R1 represents a substituted or unsubstituted C1-6 alkylthio group or a substituted or unsubstituted C1-6 alkylsulfonyl group; R2 represents a substituted or unsubstituted C1-6 alkyl group; and R represents a substituted or unsubstituted C2-6 alkenyl group.

公开(公告)号：US11180485B2

公开(公告)日：2021-11-23

申请号：US16329198

申请日：2017-09-13

Applicant: Nippon Soda Co., Ltd.

Inventor： Keita Sakanishi ,  Takao Iwasa ,  Hikaru Aoyama ,  Norifumi Sakiyama ,  Daisuke Ushijima ,  Maki Matsui ,  Tomomi Kobayashi

IPC: C07D403/14 ,  C07D401/14 ,  A01N43/54 ,  C07D403/04 ,  A01N43/653 ,  A61K31/506 ,  A01N43/50 ,  C07D233/64 ,  C07D401/04 ,  A61P31/10 ,  A01N43/56 ,  C07D403/10 ,  A61P31/14 ,  C07D413/10

Abstract: A compound represented by Formula (I), or a salt thereof: wherein, R1 represents an unsubstituted or substituted C1-6 alkylthio group, or the like; A1 represents a nitrogen atom or CH; A2 represents a nitrogen atom or CR2; R2 and R3 each independently represents a hydrogen atom, an unsubstituted or substituted C6-10 aryl group, an unsubstituted or substituted 3- to 6-membered heterocyclyl group, or the like; B1 and B2 each independently represents a nitrogen atom or CR5, with the proviso that B1 and B2 do not represent CR5 at the same time, wherein R5 represents a hydrogen atom, an unsubstituted or substituted C1-6 alkyl group, or the like; R4 represents an unsubstituted or substituted C1-6 alkyl group, or the like, and R4 binds to any one of nitrogen atoms forming an imidazole ring or a triazole ring; and Ar represents an unsubstituted or substituted C6-10 aryl group or the like.

公开(公告)号：US11078181B2

公开(公告)日：2021-08-03

申请号：US16469937

申请日：2017-12-14

Applicant: Nippon Soda Co., Ltd.

Inventor： Keita Sakanishi ,  Takao Iwasa ,  Norifumi Sakiyama ,  Hikaru Aoyama ,  Tomomi Kobayashi

IPC: C07D401/04 ,  C07D401/14 ,  A01N43/56 ,  A01N43/653

Abstract: A compound represented by the following Formula (I) or a salt thereof, as well as a formulation for controlling harmful organisms, and in particular, an insecticidal formulation, a miticidal formulation, a formulation for controlling ectoparasites or a formulation for controlling or killing endoparasites, which contains at least one compound selected from the compounds of Formula (I) and salts thereof as an active ingredient wherein, each of R1 and R2 independently represents a hydrogen atom, a substituted or unsubstituted C1-6 alkyl group, or the like, with the proviso that when R2 represents a hydrogen atom, R1 represents a substituted or unsubstituted C6-10 aryl group or a substituted or unsubstituted 3- to 6-membered heterocyclyl group; R3 represents a C1-6 alkylthio group or the like; each of R4 and R5 independently represents a hydrogen atom, a halogeno group or the like; and Ar represents a substituted or unsubstituted C6-10 aryl group, or a substituted or unsubstituted 5- to 6-membered heteroaryl group.