N-ACRYLIMINO HETEROCYCLIC COMPOUNDS
    2.
    发明申请
    N-ACRYLIMINO HETEROCYCLIC COMPOUNDS 审中-公开
    N-丙烯酰胺杂环化合物

    公开(公告)号:US20160235069A1

    公开(公告)日:2016-08-18

    申请号:US15023176

    申请日:2014-09-19

    Applicant: BASF SE

    Abstract: The present invention relates to N-acrylimino compound of formula (I): wherein X is O or S, in particular O; Het is a 5- or 6-membered carbon-bound or nitrogen-bound heterocyclic ring, W1-W2-W3-W4 represents a carbon chain group connected to N and C═N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W1, W2, W3 and W4 each individually represent CRvRw, R1, R2 may be hydrogen, halogen, etc. R3 is selected from the group consisting of hydrogen, halogen, CN, C1-C6-alkyl, etc. R4 is selected from the group consisting of hydrogen, halogen, CN, C1-C10-alkyl, etc. R5 is selected from the group consisting of hydrogen CN, C1-C10-alkyl, C2-C10-alkenyl C3-C8-cycloalkyl, S(O)nNR9aR9b, O—NR9aR9b, NR9aR9b, NR9a NR9aR9b, NR9aC(═O)R7a, NR9aC(═S)R7a, NR9aC(═O)NR9aR9b, NR9aC(═S)NR9aR9b, C(═O)OR8, C(═O)NR9aR9b, C(═S)NR9aR9b, C(═O)R7a, C(═S)R7a, a moitey Q-phenyl, where the phenyl ring is optionally substituted with 1, 2, 3, 4 or 5 identical or different substituents R10, and a moiety Q-Het# where Het# represents a 3- to 10-membered saturated, partly saturated or unsaturated aromatic heterocyclic ring. The invention also relates to the use of the N-acrylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

    Abstract translation: 本发明涉及式(I)的N-丙烯酰亚氨基化合物:其中X是O或S,特别是O; Het是5或6元碳键或氮键合的杂环,W1-W2-W3-W4表示与N和C = N连接的碳链基团,因此形成饱和的,不饱和的或部分不饱和的 5或6元含氮杂环,其中W1,W2,W3和W4各自独立地表示CRvRw,R1,R2可以是氢,卤素等。R3选自氢,卤素,CN,C1-C6- 烷基等.R 4选自氢,卤素,CN,C 1 -C 10 - 烷基等。R 5选自氢CN,C 1 -C 10 - 烷基,C 2 -C 10 - 烯基C3- C 9 - 环烷基,S(O)n NR 9 a R 9 b,O-NR 9 a R 9 b,NR 9 a R 9 b,NR 9 a NR 9 a R 9 b,NR 9 a C(= O)R 7a,NR 9 a C(≡S)R 7a,NR 9 a C(≡O)NR 9 a R 9 b,NR 9 a C(≡S)NR 9 a R 9 b,C O)OR 8,C(= O)NR 9 a R 9 b,C(= S)NR 9 a R 9 b,C(= O)R 7a,C(= O)R 7a,其中苯环任选被1,2, 3,4或5个相同或不同的取代基R10,和其中Het#表示a的部分Q-Het# 3-至10-元饱和,部分饱和或不饱和的芳族杂环。 本发明还涉及N-丙烯酰胺杂环化合物,其立体异构体,其互变异构体及其盐的用途,用于对抗无脊椎动物害虫。 此外,本发明还涉及防治无脊椎害虫的方法,其包括施用这样的化合物。

    N-SUBSTITUTED IMINO HETEROCYCLIC COMPOUNDS
    3.
    发明申请
    N-SUBSTITUTED IMINO HETEROCYCLIC COMPOUNDS 审中-公开
    N-取代的IMINO杂环化合物

    公开(公告)号:US20160326153A1

    公开(公告)日:2016-11-10

    申请号:US15105239

    申请日:2014-12-17

    Applicant: BASF SE

    Abstract: The present invention relates to N-substituted imino compound of formula (I): wherein Y is a radical Y1, Y2, Y3, Y4 or Y5, where Y1 is O—C(═X)—R3; Y2 is S—C(═X)—R3; Y3 is N(R5)—C(═X)—R3; Y4 is N(R5)—S(═O)—R4; Y5 is N(R5)—S(═O)2—R4; and where X is O or S; Het is a 5 or 6 membered carbon-bound or nitrogen-bound heterocyclic ring, W1—W2—W3—W4 represents a carbon chain group connected to N and C═N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W1, W2, W3 and W4 each individually represent CRvRw; R1, R2 may be hydrogen, halogen, C1-C6-alkyl etc.; and where R3, R4 and R5 are as defined herein. The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

    Abstract translation: 本发明还涉及N-酰基亚氨基杂环化合物,其立体异构体,其互变异构体及其盐的用途,用于防治无脊椎动物害虫。 此外,本发明还涉及防治无脊椎害虫的方法,其包括施用这样的化合物。

    N-ACYLIMINO HETEROCYCLIC COMPOUNDS
    4.
    发明申请
    N-ACYLIMINO HETEROCYCLIC COMPOUNDS 有权
    N-乙酰氨基杂环化合物

    公开(公告)号:US20160297793A1

    公开(公告)日:2016-10-13

    申请号:US15038272

    申请日:2014-11-21

    Applicant: BASF SE

    Abstract: The present invention relates to N-acylimino compound of formula (I): wherein X is O or S, in particular O; Y is a single bond, O, S or NR5; Het is a 5 or 6 membered carbon-bound or nitrogen-bound heterocyclic ring, W1—W2—W3—W4 represents a carbon chain group connected to N and C═N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W1, W2, W3 and W4 each individually represent CRvRw; R1, R2 may be hydrogen, halogen, etc.; R3 may be hydrogen, CN, C1-C6-alkyl, etc.; R4 may be of hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, Q-phenyl, Q′-O-phenyl, Q′-S-phenyl, where the phenyl ring is optionally substituted with one or more, e.g. 1, 2, 3, 4 or 5 identical or different substituents R10, and the moieties Q-Het#, Q′-O-Het# and Q′-S-Het# where Het# represents a heterocyclic radical and where Q and Q′ are C1-C6-alkandiyl, C2-C6-alkendiyl, or C2-C6-alkyndiyl, and where Q may also be a single bond; R3 and R4 together may also may also a bivalent radical, selected from the group consisting of C2-C5-alkandiyl, C2-C5-alkendiyl, Q″-C1-C4-alkandiyl and Q″-C2-C4-alkendiyl, where Q″ is O or S. The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

    Abstract translation: 本发明还涉及N-酰基亚氨基杂环化合物,其立体异构体,其互变异构体及其盐的用途,用于防治无脊椎动物害虫。 此外,本发明还涉及防治无脊椎害虫的方法,其包括施用这样的化合物。

    N-Acylimino Heterocyclic Compounds
    5.
    发明申请
    N-Acylimino Heterocyclic Compounds 审中-公开
    N-酰基亚氨基杂环化合物

    公开(公告)号:US20160227777A1

    公开(公告)日:2016-08-11

    申请号:US15023128

    申请日:2014-09-18

    Applicant: BASF SE

    Abstract: The present invention relates to N-acylimino compound of formula (I): wherein X is O or S, in particular O; m is an integer selected from 0, 1, 2, 3, 4, 5 or 6; Het is a 5 or 6 membered carbon-bound or nitrogen-bound heterocyclic ring, W1-W2-W3-W4 represents a carbon chain group connected to N and C═N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W1, W2, W3 and W4 each individually represent CRvRw, R1, R2 may be hydrogen, halogen, etc. R3 may be hydrogen, halogen, CN, C1-C6-alkyl, etc. R4a, R4b if present, may be hydrogen, halogen, C1-C6-alkyl, etc. R5 may be hydrogen, halogen, C1-C6-alkyl, C1-C6-alkenyl, C1-C6-alkinyl, C3-C8-cycloalkyl, S(O)nNR9aR9b, NR9aR9b, C(═O)OR8, C(═O)NR9aR9b, C(═S)NR9aR9b, C(═O)R7a, C(═S)R7a, NR9a—C(═O)R7a, NR9a—C(═S)R7a, NR9a—S(O)nR8a, a moiety Q-phenyl, where the phenyl ring is optionally substituted with one or more, e.g. 1, 2, 3, 4 or 5 identical or different substituents R10, or a moiety Q-Het#, or R3 and R5 together may also form with the carbon atom they are bound to, a 3, 4, 5 or 6 membered saturated partially unsaturated carbocycle or heterocycle. The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

    Abstract translation: 本发明涉及式(I)的N-酰基亚胺基化合物:其中X是O或S,特别是O; m为选自0,1,2,3,4,5或6的整数; Het是5或6元碳键或氮键的杂环,W1-W2-W3-W4表示与N和C = N连接的碳链基团,从而形成饱和的,不饱和的或部分不饱和的5或 6元含氮杂环,其中W1,W2,W3和W4各自独立地表示CRvRw,R1,R2可以是氢,卤素等。R3可以是氢,卤素,CN,C1-C6-烷基等。R4a,R4b R 5可以是氢,卤素,C 1 -C 6 - 烷基,C 1 -C 6 - 烯基,C 1 -C 6 - 炔基,C 3 -C 8 - 环烷基,S( O(n)NR 9a R 9 b,C(= O)OR 8,C(= O)NR 9 a R 9 b,C(= S)NR 9 a R 9 b,C(= O) NR9a-C(= S)R7a,NR9a-S(O)nR8a,部分Q-苯基,其中苯环任选被一个或多个例如 1,2,3或4或5个相同或不同的取代基R10或部分Q-Het#,或R3和R5一起也可以与它们所键合的碳原子一起形成,3,4,5或6元饱和 部分不饱和碳环或杂环。 本发明还涉及N-酰基亚氨基杂环化合物,其立体异构体,其互变异构体及其盐的用途,用于防治无脊椎动物害虫。 此外,本发明还涉及防治无脊椎害虫的方法,其包括施用这样的化合物。

    Substituted Pyrimidinium Compounds and Derivatives for Combating Animal Pests
    7.
    发明申请
    Substituted Pyrimidinium Compounds and Derivatives for Combating Animal Pests 有权
    取代的嘧啶鎓化合物和衍生物用于防治动物害虫

    公开(公告)号:US20160122351A1

    公开(公告)日:2016-05-05

    申请号:US14898892

    申请日:2014-06-17

    Applicant: BASF SE

    CPC classification number: C07D471/16 A01N43/90 C07D471/14

    Abstract: Substituted pyrimidinium compounds of the general formula (I) and their uses for combating animal pestsThe present invention relates to substituted pyrimidinium compounds of formula (I), to the stereoisomers, salts, tautomers and N-oxides thereof and to compositions comprising such compounds. The invention also relates to methods and uses of these substituted pyrimidinium compounds and of compositions thereof, for combating and controlling animal pests. Furthermore the invention relates also to pesticidal methods of applying such substituted pyrimidinium compounds.The substituted pyrimidinium compounds of the present invention are defined by the following general formula (I): wherein X, Y, Z, R1, R2, A, A1 and A2 are defined as in the description.

    Abstract translation: 通式(I)的取代嘧啶化合物及其用于对抗动物害虫的用途本发明涉及式(I)的取代嘧啶鎓化合物,其立体异构体,盐,互变异构体和N-氧化物以及包含这些化合物的组合物。 本发明还涉及这些取代的嘧啶鎓化合物及其组合物用于对抗和控制动物害虫的方法和用途。 此外,本发明还涉及施用这种取代的嘧啶鎓化合物的杀虫方法。 本发明的取代的嘧啶鎓化合物由以下通式(I)定义:其中X,Y,Z,R 1,R 2,A,A 1和A 2如说明书中所定义。

    N-Acylimino Heterocyclic Compounds
    9.
    发明申请

    公开(公告)号:US20190142004A1

    公开(公告)日:2019-05-16

    申请号:US16245471

    申请日:2019-01-11

    Applicant: BASF SE

    Abstract: The present invention relates to N-acylimino compound of formula (I): wherein X is O or S, in particular O; m is an integer selected from 0, 1, 2, 3, 4, 5 or 6; Het is a 5 or 6 membered carbon-bound or nitrogen-bound heterocyclic ring, W1-W2-W3-W4 represents a carbon chain group connected to N and C═N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W1, W2, W3 and W4 each individually represent CRvRw, R1, R2 may be hydrogen, halogen, etc. R3 may be hydrogen, halogen, CN, C1-C6-alkyl, etc. R4a, R4b if present, may be hydrogen, halogen, C1-C6-alkyl, etc. R5 may be hydrogen, halogen, C1-C6-alkyl, C1-C6-alkenyl, C1-C6-alkinyl, C3-C8-cycloalkyl, S(O)nNR9aR9b, NR9aR9b, C(═O)OR8, C(═O)NR9aR9b, C(═S)NR9aR9b, C(═O)R7a, C(═S)R7a, NR9a—C(═O)R7a, NR9a—C(═S)R7a, NR9a—S(O)nR8a, a moitey Q-phenyl, where the phenyl ring is optionally substituted with one or more, e.g. 1, 2, 3, 4 or 5 identical or different substituents R10, or a moiety Q-Het#, or R3 and R5 together may also form with the carbon atom they are bound to, a 3, 4, 5 or 6 membered saturated partially unsaturated carbocycle or heterocycle. The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

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