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    Process for preparing N-substituted 1H-pyrazole-5-carboxylate compounds and derivatives thereof
    1.
    发明授权
    Process for preparing N-substituted 1H-pyrazole-5-carboxylate compounds and derivatives thereof 有权
    制备N-取代的1H-吡唑-5-羧酸酯化合物及其衍生物的方法

    公开(公告)号：US09556141B2

    公开(公告)日：2017-01-31

    申请号：US14359446

    申请日：2012-11-20

    Applicant: BASF SE

    Inventor： Maximilian Dochnahl ,  Karsten Koerber ,  Prashant Deshmukh ,  Florian Kaiser ,  Michael Rack ,  Timo Frassetto ,  Gemma Veitch

    IPC: C07D401/14 ,  C07D471/10 ,  C07D401/04

    CPC classification number: C07D401/04 ,  C07D471/10

    Abstract: The present invention relates to a process for preparing an N-substituted 1H-pyrazole-5-carboxylate compound of the formula (I-A) comprising the steps of i) deprotonating a compound of the formula (II) in which the variables R1, R2 and r are each as defined in the description and the claims, with a magnesium-organic base having a carbon bound magnesium; and ii) subjecting the product obtained in step (i) to a carbonylation by reacting it with a reagent selected from the group consisting carbon dioxide or a carbon dioxide equivalent, to obtain a compound of formula (I-A); and it relates to further conversions to yield a N-substituted 1H-pyrazole-5-carbonyl chloride compound of the formula (I)

    Abstract translation: 本发明涉及制备式（IA）的N-取代的1H-吡唑-5-羧酸酯化合物的方法，包括以下步骤：i）将式（II）的化合物去质子化，其中变量R1，R2和 r各自如说明书和权利要求中所定义，其中镁 - 有机碱具有碳结合的镁; 和ii）通过使步骤（i）中获得的产物与选自二氧化碳或二氧化碳当量的试剂反应来进行羰基化，得到式（I-A）化合物; 并且涉及进一步转化得到式（I）的N-取代的1H-吡唑-5-碳酰氯化合物，

    USE OF ANTHRANILAMIDE COMPOUNDS IN SOIL AND SEED TREATMENT APPLICATION METHODS
    2.
    发明申请
    USE OF ANTHRANILAMIDE COMPOUNDS IN SOIL AND SEED TREATMENT APPLICATION METHODS 审中-公开
    在土壤和种子处理中使用蒽醌化合物的应用方法

    公开(公告)号：US20150250172A1

    公开(公告)日：2015-09-10

    申请号：US14431974

    申请日：2013-09-27

    Applicant: BASF SE

    Inventor： Karsten Körber ,  Florian Kaiser ,  Prashant Deshmukh ,  Matthias Pohlman ,  Jean-Yves Wach ,  Deborah L. Culbertson ,  W. David Rogers ,  Michael David ,  Franz Josef Braun ,  Sarah Thompson

    IPC: A01N43/56 ,  C07D401/04

    CPC classification number: A01N43/56 ,  C07D401/04

    Abstract: The present invention relates to agricultural methods using anthranilamide compounds of formula (I) wherein R1, R2, R3, R4, R5, R6, R7 and k are as defined in the description; and their mixtures; for controlling and/or combating animal pests in soil application methods and seed treatment methods The anthranilamide compounds of formula (I) are highly suitable for controlling animal pests such as insects and/or spider mites and/or nematodes by treating the soil/growth substrate by drenching or drip application or dipping or soil injection.

    Abstract translation: 本发明涉及使用式（I）的邻氨基苯甲酰胺化合物的农业方法，其中R 1，R 2，R 3，R 4，R 5，R 6，R 7和k如说明书中所定义; 及其混合物; 用于在土壤施用方法和种子处理方法中控制和/或对抗动物害虫。式（I）的邻氨基苯甲酰胺化合物非常适合于通过处理土壤/生长底物来控制动物害虫如昆虫和/或蜘蛛螨和/或线虫 通过浸泡或滴灌施用或浸渍或土壤注射。

    Process for preparing N-substituted 1H-pyrazole-5-carboxylate compounds and derivatives thereof
    3.
    发明申请
    Process for preparing N-substituted 1H-pyrazole-5-carboxylate compounds and derivatives thereof 有权
    制备N-取代的1H-吡唑-5-羧酸酯化合物及其衍生物的方法

    公开(公告)号：US20150087843A1

    公开(公告)日：2015-03-26

    申请号：US14359446

    申请日：2012-11-20

    Applicant: BASF SE

    Inventor： Maximilian Dochnahl ,  Karsten Koerber ,  Prashant Deshmukh ,  Florian Kaiser ,  Michael Rack ,  Timo Frassetto ,  Gemma Veitch

    IPC: C07D401/04

    CPC classification number: C07D401/04 ,  C07D471/10

    Abstract: The present invention relates to a process for preparing an N-substituted 1H-pyrazole-5-carboxylate compound of the formula (I-A) comprising the steps of i) deprotonating a compound of the formula (II) in which the variables R1, R2 and r are each as defined in the description and the claims, with a magnesium-organic base having a carbon bound magnesium; and ii) subjecting the product obtained in step (i) to a carbonylation by reacting it with a reagent selected from the group consisting carbon dioxide or a carbon dioxide equivalent, to obtain a compound of formula (I-A); and it relates to further conversions to yield a N-substituted 1H-pyrazole-5-carbonyl chloride compound of the formula (I)

    Abstract translation: 本发明涉及制备式（IA）的N-取代的1H-吡唑-5-羧酸酯化合物的方法，包括以下步骤：i）将式（II）的化合物去质子化，其中变量R1，R2和 r各自如说明书和权利要求中所定义，其中镁 - 有机碱具有碳结合的镁; 和ii）通过使步骤（i）中获得的产物与选自二氧化碳或二氧化碳当量的试剂反应来进行羰基化，得到式（I-A）化合物; 并且涉及进一步转化得到式（I）的N-取代的1H-吡唑-5-碳酰氯化合物，

    PESTICIDALLY ACTIVE MIXTURES COMPRISING ANTHRANILAMIDE COMPOUNDS
    7.
    发明申请
    PESTICIDALLY ACTIVE MIXTURES COMPRISING ANTHRANILAMIDE COMPOUNDS 审中-公开
    包含蒽醌化合物的农药活性混合物

    公开(公告)号：US20150250175A1

    公开(公告)日：2015-09-10

    申请号：US14432505

    申请日：2013-09-27

    Applicant: BASF SE

    Inventor： Karsten Koerber ,  Jean-Yves Wach ,  Florian Kaiser ,  Matthias Pohlman ,  Prashant Deshmukh ,  Deborah L. Culbertson ,  W. David Rogers ,  Koshi Gunjima ,  Michael David ,  Franz Josef Braun ,  Juergen Langewald

    IPC: A01N43/56 ,  A01N47/40 ,  A01N43/22 ,  A01N43/40 ,  A01N53/00 ,  A01N43/36 ,  A01N43/90 ,  A01N47/06 ,  A01N47/44

    CPC classification number: A01N43/56 ,  A01N43/22 ,  A01N43/36 ,  A01N43/40 ,  A01N43/90 ,  A01N47/06 ,  A01N47/40 ,  A01N47/44 ,  A01N53/00 ,  A01N43/707 ,  A01N43/88 ,  A01N47/02 ,  A01N47/34 ,  A01N47/38 ,  A01N51/00 ,  A01N2300/00

    Abstract: The present invention relates to pesticidal mixtures comprising as active compounds 1) at least one pesticidally active anthranilamide compound of formula (I) wherein R1, R2, R3, R4, R5, R6, R7 and k are as defined in the description; and 2) at least one pesticidally active compound II selected from a group M comprising acteylcholine esterase inhibitors, GABA-gated chloride channel antagonists, sodium channel modulators, nicotinic acteylcholine receptor agonists/antagonists, allosteric nicotinic acetylcholine receptor activitaors, chloride channel activators, juvenile hormone mimics, homopteran feeding blockers, mit grow inhibitors, inhibitors of mitochondrial bATP synthase, uncouplers of the oxidative phosphorylation, inhibitors of the chitin biosynthesis, moulting disruptors, ecdyson receptor agonists, octamin receptor agonists, inhibitors of the MET, voltage-dependent sodium channel blockers, inhibitors of the lipid synthesis, ryanodine receptor modulators and other compounds as defined in the description, in synergistically effective amounts. The invention relates further to methods and use of these mixtures for combating and controlling insects, acarids or nematodes in and on plants, and for protecting such plants being infested with pests, especially also for protecting plant propagation material, such as seeds.

    Abstract translation: 本发明涉及包含作为活性化合物的杀虫混合物1）至少一种式（I）的杀虫活性邻氨基苯甲酰胺化合物，其中R 1，R 2，R 3，R 4，R 5，R 6，R 7和k如说明书中所定义; 和2）至少一种选自包括活性胆碱酯酶抑制剂，GABA门控氯化物通道拮抗剂，钠通道调节剂，烟碱型活性胆碱受体激动剂/拮抗剂，变构烟碱乙酰胆碱受体活化剂，氯化物通道激活剂，幼年激素的组M的杀虫活性化合物II 模拟物，同翅目喂养阻断剂，mit生长抑制剂，线粒体bATP合成酶抑制剂，氧化磷酸化的解偶联剂，甲壳素生物合成抑制剂，蜕皮破坏剂，蜕皮激素受体激动剂，八胺受体激动剂，MET抑制剂，电压依赖性钠通道阻滞剂 ，脂质合成抑制剂，兰诺定受体调节剂和如说明书中所定义的其它化合物，具有协同有效量。 本发明还涉及这些混合物用于对抗和控制植物内和植物上的昆虫，螨虫或线虫的方法和用途，以及用于保护被害虫侵染的植物，特别是用于保护植物繁殖材料如种子的方法和用途。

    N-Thio-anthranilamide compounds and their use as pesticides
    8.
    发明申请
    N-Thio-anthranilamide compounds and their use as pesticides 审中-公开
    N-硫代邻氨基苯甲酰胺化合物及其作为农药的用途

    公开(公告)号：US20140309109A1

    公开(公告)日：2014-10-16

    申请号：US14365785

    申请日：2012-12-20

    Applicant: BASF SE

    Inventor： Karsten Koerber ,  Florian Kaiser ,  Prashant Deshmukh ,  Deborah L. Culbertson ,  Paul Neese ,  Koshi Gunjima

    IPC: A01N43/56 ,  C07D401/04

    CPC classification number: A01N43/56 ,  C07D401/04

    Abstract: The present invention relates to N-thio-anthranilamide compounds of the formula (I), the stereoisomers, the salts, the tautomers and the N-oxides thereof, wherein R1 is hydrogen, C1-C6-alkyl or C3-C8-cycloalkyl; R2 is hydrogen, halogen or cyano; R3 is hydrogen, C1-C6-alkyl, C1-C6-haloalkyl, C2-C6-alkenyl or the like; R4 is halogen or C1-C6-haloalkyl; R5 is an optionally substituted C1-C10-alkyl, C3-C8-cycloalkyl, C2-C10-alkenyl, C2-C10-alkynyl, phenyl, heterocyclic ring or the like; L is an optionally substituted C1-C8-alkanediyl, C2-C8-alkenediyl, C2-C8-alkynediyl, C3-C8-cycloalkanediyl or the like; G is an optionally substituted C3-C8-cycloalkyl, phenyl, heterocyclic ring or the like; and k is 0 or 1. The present invention further relates to a method for combating or controlling invertebrate pests, to a method for protecting plant propagation material and/or the plants which grow therefrom, to plant propagation material comprising at least one compound according to the present invention, to a method for treating or protecting an animal from infestation or infection by parasites, to a process for the preparation of a composition for treating infested or infected animals and/or for protecting animals against infestation or infection by parasites, and to a compound according to the invention for use as a medicament.

    Abstract translation: 本发明涉及式（I）的N-硫代 - 邻氨基苯甲酰胺化合物，其立体异构体，盐，互变异构体和N-氧化物，其中R 1是氢，C 1 -C 6 - 烷基或C 3 -C 8 - 环烷基; R2是氢，卤素或氰基; R3是氢，C1-C6-烷基，C1-C6-卤代烷基，C2-C6-烯基等; R4是卤素或C1-C6-卤代烷基; R5是任选取代的C 1 -C 10 - 烷基，C 3 -C 8 - 环烷基，C 2 -C 10 - 烯基，C 2 -C 10 - 炔基，苯基，杂环等; L是任选取代的C 1 -C 8 - 烷二基，C 2 -C 8 - 亚烯基，C 2 -C 8 - 炔二基，C 3 -C 8 - 环烷二基等; G是任选取代的C 3 -C 8 - 环烷基，苯基，杂环等; 本发明还涉及一种防治无脊椎害虫的方法，一种保护植物繁殖材料和/或从其生长的植物的方法，包括至少一种根据本发明的化合物的植物繁殖材料 本发明涉及用于治疗或保护动物免受寄生虫感染或感染的方法，涉及制备用于治疗感染或感染的动物和/或用于保护动物免受寄生虫感染或感染的组合物的方法，以及 用作药物的根据本发明的化合物。

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