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1.
公开(公告)号:US5817829A
公开(公告)日:1998-10-06
申请号:US727571
申请日:1996-10-23
申请人: Shigeaki Akiyama , Toshiaki Takeyama , Junichi Watanabe , Yasuyuki Nakajima , Hiroyuki Suzuki , Yoshiaki Yasumi , Takamasa Kikuchi , Hiroshi Ohya , Shigeru Sasabe , Masanori Nishioka , Takashi Furusato
发明人: Shigeaki Akiyama , Toshiaki Takeyama , Junichi Watanabe , Yasuyuki Nakajima , Hiroyuki Suzuki , Yoshiaki Yasumi , Takamasa Kikuchi , Hiroshi Ohya , Shigeru Sasabe , Masanori Nishioka , Takashi Furusato
IPC分类号: A01N43/56 , A01N43/78 , A01N47/24 , C07D231/14 , C07D231/16 , C07D277/20 , C07D277/56
CPC分类号: C07D277/56 , A01N43/56 , A01N43/78 , A01N47/24 , C07D231/14
摘要: The present invention provides a plant disease control agent containing as active ingredient one or more compounds of the formula �1! A--COOR.sup.1 �1! wherein R.sup.1 represents a hydrogen atom or a C.sub.1 -C.sub.4 alkyl group, and A represents a group of the formula (A-1) or (A-2) ##STR1## R.sup.2 represents a C.sub.1 -C.sub.4 alkyl group, R.sup.3 represents a C.sub.1 -C.sub.4 alkyl group, R.sup.4 represents a halogen atom or a C.sub.1 -C.sub.4 alkyl group, and R.sup.5 represents a C.sub.1 -C.sub.4 alkyl group. Further, the compound of A-1 in the formula �1! in which R.sup.3 is a halogen atom is also included in the present invention.
摘要翻译: PCT No.PCT / JP95 / 00808 Sec。 371日期:1996年10月23日 102(e)日期1996年10月23日PCT 1995年4月25日提交PCT公布。 公开号WO95 / 29161 日本公开日1995年11月2日本发明提供含有作为有效成分的一种或多种式[1] A-COOR1 [1]的化合物的植物病害防治剂,其中R1表示氢原子或C1-C4烷基,A 表示式(A-1)或(A-2)A-1或A-2的基团R 2表示C 1 -C 4烷基,R 3表示C 1 -C 4烷基,R 4表示 卤素原子或C1-C4烷基,R5表示C1-C4烷基。 此外,式(1)中R3为卤素原子的化合物A-1也包括在本发明中。
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公开(公告)号:US08022089B2
公开(公告)日:2011-09-20
申请号:US12509859
申请日:2009-07-27
IPC分类号: A61K31/42
CPC分类号: A61K31/421 , A01N43/80 , A61K9/0053 , C07C25/02 , C07C25/06 , C07C25/08 , C07C25/13 , C07C25/24 , C07C43/1742 , C07C43/1745 , C07C205/11 , C07C205/12 , C07C211/52 , C07C251/48 , C07C255/29 , C07C255/50 , C07C255/60 , C07C281/02 , C07C323/09 , C07D261/04 , C07D261/16 , C07D413/04 , C07D413/06 , C07D413/12 , C07D413/14 , C07D417/06 , C07D417/12 , C07F7/0812
摘要: An isoxazoline-substituted benzamide compound of formula (1) or a salt thereof: wherein A1, A2 and A3 independently of one another are carbon atom or nitrogen atom, G is benzene ring, etc., X is halogen atom, C1-C6haloalkyl, etc., Y is halogen atm, C1-C6alkyl, etc., R1 is C1-C12alkyl arbitrarily substituted with R16, C3-C12alkenyl, arbitrarily substituted with R16 is oxygen atom or sulfur atom, —N(R20)R19, etc., R2 is hydrogen atom, C1-C4alkoxy C1-C6alkyl, etc., R3 is C1-C6haloalkyl, etc., R16 is halogen atom, cyano, phenyl substituted with (Z)p1, D-1 to D-60, E-1 to E-49, etc., R19 is phenyl, phenyl substituted with (Z)p1, etc., R20 is hydrogen atom, C1-C6alkyl, etc., Z is halogen atom, nitro, C1-C4alkoxy, etc., D-1 to D-60 are 5- or 6-membered aromatic heterocyclic rings, E-1 to E-49 are 5- or 6-membered saturated heterocyclic rings, m is an integer of 0 to 5, n is an integer of 0 to 4, p1 is an integer of 1 to 5. The pesticide containing these compounds.
摘要翻译: 式(1)的异恶唑啉取代的苯甲酰胺化合物或其盐:其中A1,A2和A3彼此独立地为碳原子或氮原子,G为苯环等,X为卤素原子,C1-C6卤代烷基, 等等,Y是卤素原子,C 1 -C 6烷基等,R 1是被R 16任意取代的C 1 -C 12烷基,被R 16任意取代的C 3 -C 12烯基是氧原子或硫原子,-N(R 20)R 19等, R2是氢原子,C1-C4烷氧基C1-C6烷基等,R3是C1-C6卤代烷基等,R16是卤素原子,氰基,被(Z)p1,D-1到D-60,E-1 至E-49等,R19为苯基,被(Z)p1取代的苯基等,R20为氢原子,C1-C6烷基等,Z为卤素原子,硝基,C1-C4烷氧基等,D -1至D-60为5-或6-元芳族杂环,E-1至E-49为5-或6-元饱和杂环,m为0-5的整数,n为整数0 至4,p1为1〜5的整数。含有这些化合物的农药。
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公开(公告)号:US20070066617A1
公开(公告)日:2007-03-22
申请号:US11514921
申请日:2006-09-05
IPC分类号: A61K31/53 , A61K31/501 , A61K31/497 , A61K31/4439 , A61K31/42 , A61K31/427 , C07D417/14 , C07D413/14
CPC分类号: A61K31/421 , A01N43/80 , A61K9/0053 , C07C25/02 , C07C25/06 , C07C25/08 , C07C25/13 , C07C25/24 , C07C43/1742 , C07C43/1745 , C07C205/11 , C07C205/12 , C07C211/52 , C07C251/48 , C07C255/29 , C07C255/50 , C07C255/60 , C07C281/02 , C07C323/09 , C07D261/04 , C07D261/16 , C07D413/04 , C07D413/06 , C07D413/12 , C07D413/14 , C07D417/06 , C07D417/12 , C07F7/0812
摘要: An isoxazoline-substituted benzamide compound of formula (1) or a salt thereof: wherein A1, A2 and A3 independently of one another are carbon atom or nitrogen atom, G is benzene ring, etc., X is halogen atom, C1-C6haloalkyl, etc., Y is halogen atm, C1-C6alkyl, etc., R1 is C1-C12alkyl arbitrarily substituted with R16, C3-C2alkenyl, arbitrarily substituted with R16 is oxygen atom or sulfur atom, —N(R20)R19, etc., R2 is hydrogen atom, C1-C4alkoxy C1-C6alkyl, etc., R3 is C1-C6haloalkyl, etc., R16 is halogen atom, cyano, phenyl substituted with (Z)p1, D-1 to D-60, E-1 to E-49, etc., R19 is phenyl, phenyl substituted with (Z)p1, etc., R20 is hydrogen atom, C1-C6alkyl, etc., Z is halogen atom, nitro, C1-C4alkoxy, etc., D-1 to D-60 are 5- or 6-membered aromatic heterocyclic rings, E-1 to E-49 are 5- or 6-membered saturated heterocyclic rings, m is an integer of 0 to 5, n is an integer of 0 to 4, p1 is an integer of 1 to 5. The pesticide containing these compounds.
摘要翻译: 式(1)的异恶唑啉取代的苯甲酰胺化合物或其盐:其中A 1,A 2和A 3彼此独立地 是碳原子或氮原子,G是苯环等,X是卤素原子,C 1 -C 6卤代烷基等,Y是卤素原子,C C 1 -C 12烷基等,R 1是C 1 -C 12烷基, 被R 16任意取代的被R 16,C 3 -C 2 - 链烯基任意取代的亚烷基是 氧原子或硫原子,-N(R 20)R 19等,R 2是氢原子,C 1 C 3 -C 4烷氧基C 1 -C 6烷基等,R 3是C R 16卤代烷基等,R 16是卤素原子,氰基,被(Z) u> p1 u> SUB,D-1至D-60,E-1至E-49等,R 19是苯基,被(Z)取代的苯基等 R 20是氢原子,C 1 -C 6烷基, 烷基等,Z是卤素原子,硝基,C 1 -C 4烷氧基等,D-1至D-60是5-或 6元芳族杂环,E-1〜E-49为5〜6元饱和杂环,m为0〜5的整数,n为0〜4的整数,p1为1〜 5.含有这些化合物的农药。
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公开(公告)号:US20120172615A1
公开(公告)日:2012-07-05
申请号:US13350297
申请日:2012-01-13
IPC分类号: C07C255/50 , C07C43/176 , C07C33/48 , C07C205/12 , C07C43/225 , C07C25/24 , C07C323/07
CPC分类号: A61K31/421 , A01N43/80 , A61K9/0053 , C07C25/02 , C07C25/06 , C07C25/08 , C07C25/13 , C07C25/24 , C07C43/1742 , C07C43/1745 , C07C205/11 , C07C205/12 , C07C211/52 , C07C251/48 , C07C255/29 , C07C255/50 , C07C255/60 , C07C281/02 , C07C323/09 , C07D261/04 , C07D261/16 , C07D413/04 , C07D413/06 , C07D413/12 , C07D413/14 , C07D417/06 , C07D417/12 , C07F7/0812
摘要: A substituted alkenylbenzene compound of formula (4): wherein X1 is a halogen atom, —SF5, C1-C6haloalkyl, hydroxy C1-C6haloalkyl, C1-C6alkoxy C1-C6haloalkyl, C3-C8halocycloalkyl, C1-C6haloalkoxy, C1-C3haloalkoxy C1-C3haloalkoxy, C1-C6haloalkylthio, C1-C6haloalkylsulfinyl or C1-C6haloalkylsulfonyl; X3 is a hydrogen, halogen, cyano, nitro, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy or C1-C6alkylthio; X4 is a hydrogen, halogen, cyano, C1-C4alkyl, C1-C4alkoxy or C1-C4haloalkoxy; R3 is —C(R3a)(R3b)R3c, where R3a and R3b are a halogen, or R3a and R3b together form a 3- to 6-membered ring together with the carbon bonding them by forming a C2-C5haloalkylene chain, and R3c is a hydrogen, halogen, C1-C5alkyl, C1-C5haloalkyl, C1-C4haloalkoxy or C1-C4haloalkylthio, with a proviso that where X1 is a fluorine, chlorine or trifluoromethyl, and X2 and X3 are hydrogen, where X1 and X2 are fluorine and X3 is a hydrogen, or where X1 and X2 are trifluoromethyl and X3 is a hydrogen, R3c is a hydrogen, chlorine, bromine, iodine, C1-C5alkyl, C1-C5haloalkyl, C1-C4haloalkoxy or C1-C4haloalkylthio.
摘要翻译: 式(4)的取代烯基苯化合物:其中X 1是卤素原子,-SF 5,C 1 -C 6卤代烷基,羟基C 1 -C 6卤代烷基,C 1 -C 6烷氧基C 1 -C 6卤代烷基,C 3 -C 8卤代环烷基,C 1 -C 6卤代烷氧基,C 1 -C 3卤代烷氧基C 1 -C 3卤代烷氧基 ,C 1 -C 6卤代烷硫基,C 1 -C 6卤代烷基亚磺酰基或C 1 -C 6卤代烷基磺酰基; X 3是氢,卤素,氰基,硝基,C 1 -C 6烷基,C 1 -C 6卤代烷基,C 1 -C 6烷氧基或C 1 -C 6烷硫基; X 4是氢,卤素,氰基,C 1 -C 4烷基,C 1 -C 4烷氧基或C 1 -C 4卤代烷氧基; R3是-C(R3a)(R3b)R3c,其中R3a和R3b是卤素,或者R3a和R3b与通过形成C 2 -C 5卤代亚烷基链键合的碳一起形成3-至6-元环,并且R3c 是卤素,C 1 -C 5烷基,C 1 -C 5卤代烷基,C 1 -C 4卤代烷氧基或C 1 -C 4卤代烷硫基,条件是其中X 1是氟,氯或三氟甲基,X 2和X 3是氢,其中X 1和X 2是氟, X 3是氢,或者其中X 1和X 2是三氟甲基,X 3是氢,R 3c是氢,氯,溴,碘,C 1 -C 5烷基,C 1 -C 5卤代烷基,C 1 -C 4卤代烷氧基或C 1 -C 4卤代烷硫基。
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公开(公告)号:US08138213B2
公开(公告)日:2012-03-20
申请号:US13166294
申请日:2011-06-22
IPC分类号: A61K31/42 , C07D261/04
CPC分类号: A61K31/421 , A01N43/80 , A61K9/0053 , C07C25/02 , C07C25/06 , C07C25/08 , C07C25/13 , C07C25/24 , C07C43/1742 , C07C43/1745 , C07C205/11 , C07C205/12 , C07C211/52 , C07C251/48 , C07C255/29 , C07C255/50 , C07C255/60 , C07C281/02 , C07C323/09 , C07D261/04 , C07D261/16 , C07D413/04 , C07D413/06 , C07D413/12 , C07D413/14 , C07D417/06 , C07D417/12 , C07F7/0812
摘要: A 3,5-Bis (substituted aryl) substituted isoxazoline compound of formula (2) or a salt thereof: wherein A1 is a carbon atom or nitrogen atom; X1 is selected from the group consisting of a halogen atom, —SF5, C1-C6haloalkyl, hydroxy C1-C6haloalkyl, C1-C6alkoxy C1-C6haloalkyl, C1-C6haloalkoxy C1-C6haloalkyl, C3-C8halocycloalkyl, C1-C6haloalkoxy, C1-C3haloalkoxy C1-C3haloalkoxy, C1-C6haloalkylthio, C1-C6haloalkylsulfinyl and C1-C6haloalkylsulfonyl; X2 is selected from the group consisting of a halogen atom, cyano, nitro, C1-C6alkyl, C1-C6haloalkyl, —OR5, —OSO2R5 and —S(O)rR5; Y is selected from the group consisting of a halogen atom, cyano, nitro, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy, C1-C6alkylthio, C1-C6haloalkylthio, C1-C6alkylsulfonyl, C1-C6haloalkylsulfonyl, —NHR7 and —N(R7)R6; R is selected from the group consisting of a halogen atom, cyano, nitro, —NH2, halosulfonyloxy, C1-C6alkylsulfonyloxy, C1-C6haloalkylsulfonyloxy, phenylsulfonyloxy, phenylsulfonyloxy substituted with (Z)p1 and —C(O)Ra; m1 is an integer of 0 to 2; n is an integer of 0 or 1; p1 is an integer of 1 to 5; and r is an integer of 0 to 2.
摘要翻译: 式(2)的3,5-双(取代的芳基)取代的异恶唑啉化合物或其盐:其中A1是碳原子或氮原子; X1选自卤素原子,-SF 5,C 1 -C 6卤代烷基,羟基C 1 -C 6卤代烷基,C 1 -C 6烷氧基C 1 -C 6卤代烷基,C 1 -C 6卤代烷氧基C 1 -C 6卤代烷基,C 3 -C 8卤代环烷基,C 1 -C 6卤代烷氧基,C 1 -C 3卤代烷氧基C1 C 3卤代烷氧基,C 1 -C 6卤代烷硫基,C 1 -C 6卤代烷基亚磺酰基和C 1 -C 6卤代烷基磺酰基; X 2选自卤素原子,氰基,硝基,C 1 -C 6烷基,C 1 -C 6卤代烷基,-OR 5,-OSO 2 R 5和-S(O)r R 5; Y选自卤素原子,氰基,硝基,C 1 -C 4烷基,C 1 -C 4卤代烷基,C 1 -C 4烷氧基,C 1 -C 4卤代烷氧基,C 1 -C 6烷硫基,C 1 -C 6卤代烷硫基,C 1 -C 6烷基磺酰基,C 1 -C 6卤代烷基磺酰基,-NHR 7 和-N(R 7)R 6; R选自卤素原子,氰基,硝基,-NH 2,卤代磺酰氧基,C 1 -C 6烷基磺酰氧基,C 1 -C 6卤代烷基磺酰氧基,苯基磺酰氧基,被(Z)p1和-C(O)Ra取代的苯基磺酰氧基; m1为0〜2的整数; n为0或1的整数; p1为1〜5的整数, r为0〜2的整数。
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公开(公告)号:US07662972B2
公开(公告)日:2010-02-16
申请号:US11514921
申请日:2006-09-05
IPC分类号: C07D261/04 , A61K31/42
CPC分类号: A61K31/421 , A01N43/80 , A61K9/0053 , C07C25/02 , C07C25/06 , C07C25/08 , C07C25/13 , C07C25/24 , C07C43/1742 , C07C43/1745 , C07C205/11 , C07C205/12 , C07C211/52 , C07C251/48 , C07C255/29 , C07C255/50 , C07C255/60 , C07C281/02 , C07C323/09 , C07D261/04 , C07D261/16 , C07D413/04 , C07D413/06 , C07D413/12 , C07D413/14 , C07D417/06 , C07D417/12 , C07F7/0812
摘要: An isoxazoline-substituted benzamide compound of formula (1) or a salt thereof: wherein A1, A2 and A3 independently of one another are carbon atom or nitrogen atom, G is benzene ring, etc., X is halogen atom, C1-C6haloalkyl, etc., Y is halogen atom, C1-C6alkyl, etc., R1 is C1-C12alkyl arbitrarily substituted with R16, C3-C2alkenyl, arbitrarily substituted with R16 is oxygen atom or sulfur atom, —N(R20)R19, etc., R2 is hydrogen atom, C1-C4alkoxy C1-C6alkyl, etc., R3 is C1-C6haloalkyl, etc., R16 is halogen atom, cyano, phenyl substituted with (Z)p1, D-1 to D-60, E-1 to E-49, etc., R19 is phenyl, phenyl substituted with (Z)p1, etc., R20 is hydrogen atom, C1-C6alkyl, etc., Z is halogen atom, nitro, C1-C4alkoxy, etc., D-1 to D-60 are 5- or 6-membered aromatic heterocyclic rings, E-1 to E-49 are 5- or 6-membered saturated heterocyclic rings, m is an integer of 0 to 5, n is an integer of 0 to 4, p1 is an integer of 1 to 5. The pesticide containing these compounds.
摘要翻译: 式(1)的异恶唑啉取代的苯甲酰胺化合物或其盐:其中A1,A2和A3彼此独立地为碳原子或氮原子,G为苯环等,X为卤素原子,C1-C6卤代烷基, 等等,Y是卤素原子,C1-C6烷基等,R1是被R16任意取代的C 1 -C 12烷基,被R 16任意取代的C 3 -C 21烯基是氧原子或硫原子,-N(R 20)R 19等, R2是氢原子,C1-C4烷氧基C1-C6烷基等,R3是C1-C6卤代烷基等,R16是卤素原子,氰基,被(Z)p1,D-1到D-60,E-1 至E-49等,R19为苯基,被(Z)p1取代的苯基等,R20为氢原子,C1-C6烷基等,Z为卤素原子,硝基,C1-C4烷氧基等,D -1至D-60为5-或6-元芳族杂环,E-1至E-49为5-或6-元饱和杂环,m为0-5的整数,n为整数0 至4,p1为1〜5的整数。含有这些化合物的农药。
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公开(公告)号:US20200000777A1
公开(公告)日:2020-01-02
申请号:US16508818
申请日:2019-07-11
申请人: Takeshi MITA , Takamasa KIKUCHI , Takashi MIZUKOSHI , Manabu YAOSAKA , Mitsuaki KOMODA , Shinji TAKII
发明人: Takeshi MITA , Takamasa KIKUCHI , Takashi MIZUKOSHI , Manabu YAOSAKA , Mitsuaki KOMODA , Shinji TAKII
IPC分类号: A61K31/421 , C07C25/13 , C07C25/24 , C07C25/02 , C07C25/06 , C07C25/08 , A01N43/80 , C07C43/174 , C07C205/11 , C07C205/12 , C07C211/52 , C07C251/48 , C07C255/29 , C07C255/50 , C07C255/60 , C07C281/02 , C07C323/09 , C07D261/16 , C07D413/06 , C07D413/12 , C07D417/06 , C07D417/12 , C07F7/08 , C07D413/04 , C07D261/04 , C07D413/14 , A61K9/00
摘要: A substituted alkenylbenzene compound of formula (4): wherein X1 is selected from the group consisting of a halogen atom, —SF5, C1-C6haloalkyl, hydroxy C1-C6haloalkyl, C1-C6alkoxy C1-C6haloalkyl, C3-C8halocycloalkyl, C1-C6haloalkoxy, C1-C3haloalkoxy C1-C3haloalkoxy, C1-C6haloalkylthio, C1-C6haloalkylsulfinyl and C1-C6haloalkylsulfonyl; X3 is selected from the group consisting of a hydrogen atom, halogen atom, cyano, nitro, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy and C1-C6alkylthio; X4 is selected from the group consisting of a hydrogen atom, halogen atom, cyano, C1-C4alkyl, C1-C4alkoxy and C1-C4haloalkoxy; R3 is —C(R3a)(R3b)R3c, where R3a and R3b independently of each other are a halogen atom, or R3a and R3b together form 3- to 6-membered ring together with the carbon atom bonding them by forming a C2-C5haloalkylene chain, and R3c is selected from the group consisting of a hydrogen atom, halogen atom, C1-C5alkyl, C1-C5haloalkyl, C1-C4haloalkoxy and C1-C4haloalkylthio, with a proviso that in case where X1 is a fluorine atom, chlorine atom or trifluoromethyl, and both X2 and X3 are a hydrogen atom, in case where both X1 and X2 are fluorine atom and X3 is a hydrogen atom, and in case where both X1 and X2 are trifluoromethyl and X3 is a hydrogen atom, R3c is a hydrogen atom, chlorine atom, bromine atom, iodine atom, C1-C5alkyl, C1-C5haloalkyl, C1-C4haloalkoxy or C1-C4haloalkylthio.
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公开(公告)号:US20110251398A1
公开(公告)日:2011-10-13
申请号:US13166294
申请日:2011-06-22
IPC分类号: C07D261/04 , C07D413/10 , C07D413/14 , C07D413/04
CPC分类号: A61K31/421 , A01N43/80 , A61K9/0053 , C07C25/02 , C07C25/06 , C07C25/08 , C07C25/13 , C07C25/24 , C07C43/1742 , C07C43/1745 , C07C205/11 , C07C205/12 , C07C211/52 , C07C251/48 , C07C255/29 , C07C255/50 , C07C255/60 , C07C281/02 , C07C323/09 , C07D261/04 , C07D261/16 , C07D413/04 , C07D413/06 , C07D413/12 , C07D413/14 , C07D417/06 , C07D417/12 , C07F7/0812
摘要: A 3,5-Bis (substituted aryl) substituted isoxazoline compound of formula (2) or a salt thereof: wherein A1 is a carbon atom or nitrogen atom; X1 is selected from the group consisting of a halogen atom, —SF5, C1-C6haloalkyl, hydroxy C1-C6haloalkyl, C1-C6alkoxy C1-C6haloalkyl, C1-C6haloalkoxy C1-C6haloalkyl, C3-C8halocycloalkyl, C1-C6haloalkoxy, C1-C3haloalkoxy C1-C3haloalkoxy, C1-C6haloalkylthio, C1-C6haloalkylsulfinyl and C1-C6haloalkylsulfonyl; X2 is selected from the group consisting of a halogen atom, cyano, nitro, C1-C6alkyl, C1-C6haloalkyl, —OR5, —OSO2R5 and —S(O)rR5; Y is selected from the group consisting of a halogen atom, cyano, nitro, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy, C1-C6alkylthio, C1-C6haloalkylthio, C1-C6alkylsulfonyl, C1-C6haloalkylsulfonyl, —NHR7 and —N(R7)R6; R is selected from the group consisting of a halogen atom, cyano, nitro, —NH2, halosulfonyloxy, C1-C6alkylsulfonyloxy, C1-C6haloalkylsulfonyloxy, phenylsulfonyloxy, phenylsulfonyloxy substituted with (Z)p1 and —C(O)Ra; m1 is an integer of 0 to 2; n is an integer of 0 or 1; p1 is an integer of 1 to 5; and r is an integer of 0 to 2.
摘要翻译: 式(2)的3,5-双(取代的芳基)取代的异恶唑啉化合物或其盐:其中A1是碳原子或氮原子; X1选自卤素原子,-SF 5,C 1 -C 6卤代烷基,羟基C 1 -C 6卤代烷基,C 1 -C 6烷氧基C 1 -C 6卤代烷基,C 1 -C 6卤代烷氧基C 1 -C 6卤代烷基,C 3 -C 8卤代环烷基,C 1 -C 6卤代烷氧基,C 1 -C 3卤代烷氧基C1 C 3卤代烷氧基,C 1 -C 6卤代烷硫基,C 1 -C 6卤代烷基亚磺酰基和C 1 -C 6卤代烷基磺酰基; X 2选自卤素原子,氰基,硝基,C 1 -C 6烷基,C 1 -C 6卤代烷基,-OR 5,-OSO 2 R 5和-S(O)r R 5; Y选自卤素原子,氰基,硝基,C 1 -C 4烷基,C 1 -C 4卤代烷基,C 1 -C 4烷氧基,C 1 -C 4卤代烷氧基,C 1 -C 6烷硫基,C 1 -C 6卤代烷硫基,C 1 -C 6烷基磺酰基,C 1 -C 6卤代烷基磺酰基,-NHR 7 和-N(R 7)R 6; R选自卤素原子,氰基,硝基,-NH 2,卤代磺酰氧基,C 1 -C 6烷基磺酰氧基,C 1 -C 6卤代烷基磺酰氧基,苯基磺酰氧基,被(Z)p1和-C(O)Ra取代的苯基磺酰氧基; m1为0〜2的整数; n为0或1的整数; p1为1〜5的整数, r为0〜2的整数。
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公开(公告)号:US08492311B2
公开(公告)日:2013-07-23
申请号:US13350297
申请日:2012-01-13
IPC分类号: A01N43/80 , C07D261/04
CPC分类号: A61K31/421 , A01N43/80 , A61K9/0053 , C07C25/02 , C07C25/06 , C07C25/08 , C07C25/13 , C07C25/24 , C07C43/1742 , C07C43/1745 , C07C205/11 , C07C205/12 , C07C211/52 , C07C251/48 , C07C255/29 , C07C255/50 , C07C255/60 , C07C281/02 , C07C323/09 , C07D261/04 , C07D261/16 , C07D413/04 , C07D413/06 , C07D413/12 , C07D413/14 , C07D417/06 , C07D417/12 , C07F7/0812
摘要: A substituted alkenylbenzene compound of formula (4): wherein X1 is a halogen atom, —SF5, C1-C6haloalkyl, hydroxy C1-C6haloalkyl, C1-C6alkoxy C1-C6haloalkyl, C3-C8halocycloalkyl, C1-C6haloalkoxy, C1-C3haloalkoxy C1-C3haloalkoxy, C1-C6haloalkylthio, C1-C6haloalkylsulfinyl or C1-C6haloalkylsulfonyl; X3 is a hydrogen, halogen, cyano, nitro, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy or C1-C6alkylthio; X4 is a hydrogen, halogen, cyano, C1-C4alkyl, C1-C4alkoxy or C1-C4haloalkoxy; R3 is —C(R3a)(R3b)R3c, where R3a and R3b are a halogen, or R3a and R3b together form a 3- to 6-membered ring together with the carbon bonding them by forming a C2-C5haloalkylene chain, and R3c is a hydrogen, halogen, C1-C5alkyl, C1-C5haloalkyl, C1-C4haloalkoxy or C1-C4haloalkylthio, with a proviso that where X1 is a fluorine, chlorine or trifluoromethyl, and X2 and X3 are hydrogen, where X1 and X2 are fluorine and X3 is a hydrogen, or where X1 and X2 are trifluoromethyl and X3 is a hydrogen, R3c is a hydrogen, chlorine, bromine, iodine, C1-C5alkyl, C1-C5haloalkyl, C1-C4haloalkoxy or C1-C4haloalkylthio.
摘要翻译: 式(4)的取代烯基苯化合物:其中X 1是卤素原子,-SF 5,C 1 -C 6卤代烷基,羟基C 1 -C 6卤代烷基,C 1 -C 6烷氧基C 1 -C 6卤代烷基,C 3 -C 8卤代环烷基,C 1 -C 6卤代烷氧基,C 1 -C 3卤代烷氧基C 1 -C 3卤代烷氧基 ,C 1 -C 6卤代烷硫基,C 1 -C 6卤代烷基亚磺酰基或C 1 -C 6卤代烷基磺酰基; X 3是氢,卤素,氰基,硝基,C 1 -C 6烷基,C 1 -C 6卤代烷基,C 1 -C 6烷氧基或C 1 -C 6烷硫基; X 4是氢,卤素,氰基,C 1 -C 4烷基,C 1 -C 4烷氧基或C 1 -C 4卤代烷氧基; R3是-C(R3a)(R3b)R3c,其中R3a和R3b是卤素,或者R3a和R3b与通过形成C 2 -C 5卤代亚烷基链键合的碳一起形成3-至6-元环,并且R3c 是卤素,C 1 -C 5烷基,C 1 -C 5卤代烷基,C 1 -C 4卤代烷氧基或C 1 -C 4卤代烷硫基,条件是其中X 1是氟,氯或三氟甲基,X 2和X 3是氢,其中X 1和X 2是氟, X 3是氢,或者其中X 1和X 2是三氟甲基,X 3是氢,R 3c是氢,氯,溴,碘,C 1 -C 5烷基,C 1 -C 5卤代烷基,C 1 -C 4卤代烷氧基或C 1 -C 4卤代烷硫基。
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公开(公告)号:US20090312330A1
公开(公告)日:2009-12-17
申请号:US12509859
申请日:2009-07-27
IPC分类号: A61K31/53 , A61K31/501 , A61K31/497 , A61K31/427 , A61K31/4439 , A61K31/42
CPC分类号: A61K31/421 , A01N43/80 , A61K9/0053 , C07C25/02 , C07C25/06 , C07C25/08 , C07C25/13 , C07C25/24 , C07C43/1742 , C07C43/1745 , C07C205/11 , C07C205/12 , C07C211/52 , C07C251/48 , C07C255/29 , C07C255/50 , C07C255/60 , C07C281/02 , C07C323/09 , C07D261/04 , C07D261/16 , C07D413/04 , C07D413/06 , C07D413/12 , C07D413/14 , C07D417/06 , C07D417/12 , C07F7/0812
摘要: An isoxazoline-substituted benzamide compound of formula (1) or a salt thereof: wherein A1, A2 and A3 independently of one another are carbon atom or nitrogen atom, G is benzene ring, etc., X is halogen atom, C1-C6haloalkyl, etc., Y is halogen atm, C1-C6alkyl, etc., R1 is C1-C12alkyl arbitrarily substituted with R16, C3-C12alkenyl, arbitrarily substituted with R16 is oxygen atom or sulfur atom, —N(R20)R19, etc., R2 is hydrogen atom, C1-C4alkoxy C1-C6alkyl, etc., R3 is C1-C6haloalkyl, etc., R16 is halogen atom, cyano, phenyl substituted with (Z)p1, D-1 to D-60, E-1 to E-49, etc., R19 is phenyl, phenyl substituted with (Z)p1, etc., R20 is hydrogen atom, C1-C6alkyl, etc., Z is halogen atom, nitro, C1-C4alkoxy, etc., D-1 to D-60 are 5- or 6-membered aromatic heterocyclic rings, E-1 to E-49 are 5- or 6-membered saturated heterocyclic rings, m is an integer of 0 to 5, n is an integer of 0 to 4, p1 is an integer of 1 to 5. The pesticide containing these compounds.
摘要翻译: 式(1)的异恶唑啉取代的苯甲酰胺化合物或其盐:其中A1,A2和A3彼此独立地为碳原子或氮原子,G为苯环等,X为卤素原子,C1-C6卤代烷基, 等等,Y是卤素原子,C 1 -C 6烷基等,R 1是被R 16任意取代的C 1 -C 12烷基,被R 16任意取代的C 3 -C 12烯基是氧原子或硫原子,-N(R 20)R 19等, R2是氢原子,C1-C4烷氧基C1-C6烷基等,R3是C1-C6卤代烷基等,R16是卤素原子,氰基,被(Z)p1,D-1到D-60,E-1 至E-49等,R19为苯基,被(Z)p1取代的苯基等,R20为氢原子,C1-C6烷基等,Z为卤素原子,硝基,C1-C4烷氧基等,D -1至D-60为5-或6-元芳族杂环,E-1至E-49为5-或6-元饱和杂环,m为0-5的整数,n为整数0 至4,p1为1〜5的整数。含有这些化合物的农药。
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