Derivatives of 4,4-difluorobut-3-enylsulfinic acid and their use as pesticides
    36.
    发明授权
    Derivatives of 4,4-difluorobut-3-enylsulfinic acid and their use as pesticides 失效
    4,4-二氟丁-3-烯基亚磺酸的衍生物及其作为农药的用途

    公开(公告)号:US06274632B1

    公开(公告)日:2001-08-14

    申请号:US09380912

    申请日:1999-09-10

    申请人: Roger Salmon

    发明人: Roger Salmon

    IPC分类号: A61K31535

    摘要: The invention relates to compounds of the formula (I): CF2═CX—CH2—CH2—S(O)—R wherein X represents hydrogen, halogen or lower alkyl, and R represents a group OR1 or NR2R3 wherein R1, R2 and R3 are as defined in the description. The compounds are useful for controlling insect and like pests of agriculture.

    摘要翻译: 本发明涉及式(I)化合物:CF2 = CX-CH2-CH2-S(O)-R,其中X表示氢,卤素或低级烷基,R表示OR1或NR2R3基团,其中R1,R2和R3 如说明书中所定义。 这些化合物可用于控制昆虫和农业害虫。

    Bicyclic amines
    37.
    发明授权
    Bicyclic amines 有权
    双环胺

    公开(公告)号:US06207676B1

    公开(公告)日:2001-03-27

    申请号:US09207195

    申请日:1998-12-08

    IPC分类号: A61K31439

    摘要: A compound of formula (I): wherein R1 represents a group of formula (A) where each of W, X, Y and Z and Z represents either a group CR or the nitrogen atom, provided that not more than two of W, X, Y and Z represent the nitrogen atom and where each R present is independently selected from hydrogen and halogen atoms and cyano, amino, hydrazino, acylamino, hydroxy, alkyl, hydroxyalkyl, alkoxy, haloalkyl, haloalkoxy, alkenyl, alkenyloxy, alkoxyalkenyl, alkynyl, carboxylic acyl, alkoxycarbonyl, aryl and heterocyclyl groups, said groups comprising up to 6 carbon atoms, and wherein R2 represents hydrogen or cyano or a group selected from alkyl, aryl, heteroaryl, aralkyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, alkoxycarbonyl, alkanesulfonyl, arenesulfonyl, alkanyloxycarbonyl, aralkyloxycarbonyl, aryloxycarbonyl, heterocyclylalkyl, carbamyl or dithiocarboxyl groups, said groups comprising from 1 to 15 carbon atoms, said groups being optionally substituted with one or more substituents selected from, halogen, cyano, carboxyl, carboxylic acyl, carbamyl, alkoxycarbonyl, alkoxy, alkylenedioxy, hydroxy, nitro, haloalkyl, alkyl, amino, acylamino, imidate and phosphonato groups; and acid addition salts and quaternary ammonium salts and N-oxide derived therefrom. The compounds are useful as insecticides.

    摘要翻译: 式(I)的化合物:其中R 1表示式(A)的基团,其中W,X,Y和Z和Z各自表示基团CR或氮原子,条件是不大于2个W,X ,Y和Z代表氮原子,其中每个R独立地选自氢和卤素原子和氰基,氨基,肼基,酰氨基,羟基,烷基,羟基烷基,烷氧基,卤代烷基,卤代烷氧基,烯基,烯氧基,烷氧基烯基,炔基, 羧基酰基,烷氧基羰基,芳基和杂环基,所述基团包含至多6个碳原子,并且其中R 2表示氢或氰基或选自烷基,芳基,杂芳基,芳烷基,杂芳基烷基,烯基,芳烯基,炔基,烷氧基羰基,链烷磺酰基 ,芳基磺酰基,烷氧基羰基,芳烷氧基羰基,芳氧基羰基,杂环基烷基,氨基甲酰基或二硫代羧基,​​所述基团包含1至15个碳原子,所述基团任选被一个或多个取代基se 由卤素,氰基,羧基,羧基酰基,氨基甲酰基,烷氧基羰基,烷氧基,亚烷基二氧基,羟基,硝基,卤代烷基,烷基,氨基,酰氨基,亚氨酸酯和膦酸酯基组成。 和酸加成盐和季铵盐和由其衍生的N-氧化物。 这些化合物可用作杀虫剂。

    Bicyclic amine derivatives
    38.
    发明授权
    Bicyclic amine derivatives 失效
    双环胺衍生物

    公开(公告)号:US06174894B1

    公开(公告)日:2001-01-16

    申请号:US09357749

    申请日:1999-07-21

    IPC分类号: A61K31435

    摘要: The present invention provides a compound of Formula (I): wherein Ar is optionally substituted phenyl wherein the substutuents, if present, are selected from halogen atoms, cyano, alkyl, alkenyl, alkynyl, alkoxy, haloalkyl, haloalkenyl, alkylthio and alkyl amino groups; R represents hydrogen or cyano or a group selected from alkyl, aryl, heteroaryl, aralkyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, alkoxycarbonyl, alkanesulfonyl, arenesulfonyl, alkenyloxycarbonyl, aralkyloxycarbonyl, aryloxycarbonyl, heterocyclylalkyl, carbamyl, dithiocarboxyl or XR3 (where X represents oxygen or a group NR4); R3 and R4 are, independently, hydrogen, alkyl, aryl, heteroaryl, aralkyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, heterocyclylalkyl, alkoxycarbonyl or carboxylic acyl each of which may be optionally substituted; R1 represents hydrogen, hydroxy, alkyl, alkoxy, amino, nitro, isocyanato, acylamino, hydroxyalkyl, optionally substituted heteroaryl, alkoxyalkyl, haloalkyl, halohydroxyalkyl, aralkyloxyalkyl, acyloxyalkyl, amidoximido, sulfonyloxyalkyl, aminoalkyl, alkoxycarbonylamino, acylaminoalkyl, cyanoalkyl, imino, formyl, acyl or carboxylic acid or an ester or amide thereof, or alkenyl or alkynyl either of which is optionally substituted; or an acid addition salt, quaternary ammonium salt or N-oxide derived therefrom; an insecticidal, acaricidal or nematicidal composition comprising a compound of formula (I) and a suitable carrier or diluent therefor; and a method of combating and controlling insect, acarine or nematode pests at a locus which comprises treating the pests or the locus of the pests with an effective amount of a compound of formula (I) or a composition as hereinbefore described.

    摘要翻译: 本发明提供式(I)的化合物:其中Ar是任选取代的苯基,其中如果存在这些取代基,则选自卤素原子,氰基,烷基,烯基,炔基,烷氧基,卤代烷基,卤代烯基,烷硫基和烷基氨基 ; R表示氢或氰基或选自烷基,芳基,杂芳基,芳烷基,杂芳基烷基,烯基,芳烯基,炔基,烷氧基羰基,链烷磺酰基,芳烃磺酰基,烯氧基羰基,芳烷氧基羰基,芳氧基羰基,杂环基烷基,氨基甲酰基,二硫代羧基或XR3(其中X表示氧 或NR4组); R 3和R 4独立地是氢,烷基,芳基,杂芳基,芳烷基,杂芳基烷基,烯基,芳烯基,炔基,杂环基烷基,烷氧基羰基或羧酰基,各自可以任选被取代; R 1表示氢,羟基,烷基,烷氧基,氨基,硝基,异氰酸酯基,酰氨基,羟基烷基,任选取代的杂芳基,烷氧基烷基,卤代烷基,卤代羟烷基,芳烷氧基烷基,酰氧基烷基,酰氨基亚氨基,磺酰氧基烷基,氨基烷基,烷氧基羰基氨基,酰氨基烷基,氰基烷基,亚氨基,甲酰基, 酰基或羧酸或其酯或酰胺,或任选被取代的链烯基或炔基; 或由其衍生的酸加成盐,季铵盐或N-氧化物; 杀虫杀螨或杀线虫组合物,其包含式(I)化合物及其合适的载体或稀释剂; 以及一种防治昆虫,螨虫或线虫害虫的场所的方法,包括用有效量的式(I)化合物或上述组合物处理害虫或害虫的场所。

    Bicyclic amine derivatives
    39.
    发明授权
    Bicyclic amine derivatives 失效
    双环胺衍生物

    公开(公告)号:US6093726A

    公开(公告)日:2000-07-25

    申请号:US969639

    申请日:1997-11-13

    摘要: A compound of formula (I): ##STR1## wherein Ar is optionally substituted phenyl or optionally substituted 5-or 6-membered heterocyclic ring containing from 1 to 3 heteroatoms individually selected from nitrogen, oxygen and sulfur atoms, and at least one unsaturation (double bond) between adjacent atoms in the ring, said heterocyclic ring being optionally fused to a benzene ring; or an acid addition salt, quaternary ammonium salt or N-oxide derived therefrom, an insecticidal, acaricidal or nematicidal composition comprising a compound of formula (I) and a suitable carrier or diluent therefor, a method of combating and controlling insect, acarine or nematode pests at a locus which comprises treating the pests or the locus of the pests with an effective amount of a compound of formula (I) or a composition as hereinbefore described.

    摘要翻译: 式(I)的化合物:其中Ar是任选取代的苯基或含有1至3个选自氮,氧和硫原子的杂原子的任选取代的5或6元杂环,和至少一个不饱和键(双键) 在环中的相邻原子之间,所述杂环任选地与苯环稠合; 或由其衍生的酸加成盐,季铵盐或N-氧化物,包含式(I)化合物及其合适的载体或稀释剂的杀虫,杀螨或杀线虫组合物,防治昆虫,螨虫或线虫的方法 包括用有效量的式(I)化合物或上述组合物处理害虫或害虫的场所的场所的害虫。