摘要:
Pesticidal substituted pyridazinones of the formula ##STR1## in which R.sup.1 represents alkyl, halogenolkyl, alkoxyalkyl, alkylthioalkyl, (di)alkylaminoalkyl, alkenyl or halogenoalkenyl, or represents in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl or aralkyl,R.sup.2 represents halogen or alkyl,R.sup.3 and R.sup.4 independently of one another in each case represent hydrogen or alkyl,R.sup.5 and R.sup.6 represent hydrogen, carboxyl, in each case optionally substituted straight-chain or branched alkyl, alkenyl, alkoxycarbonyl, aryl or aralkyl, or, together with the carbon atom to which they are bonded, rpresent an optionally substituted saturated or unsaturaated carbocyle,R.sup.7, R.sup.8, R.sup.9, R.sup.10 and R.sup.11 independently of one another in each case represent hydrogen, halogen, alkyl, halogenoalkyl, alkoxy, halogenoalkoxy, alkylthio or halogenoalkylthio, andX represents oxygen or sulphur.Several intermediates therefor are also new.
摘要:
Combatting fungi and bacteria with aminomethylheterocyclic compounds of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkenyl, in each case optionally substituted tetrahydronaphthyl, decahydronaphthyl, cycloalkyl or cycloalkenyl, furthermore alkyl which is substituted by cycloalkyl, cycloalkenyl, cycloalkyloxy or cycloalkylthio, where the cyclic radicals may optionally be substituted, furthermore optionally substituted aryl, in addition alkyl which is substituted by aryl, aryloxy, arylthio, arylsulphinyl or arylsulphonyl, or alkenyl which is substituted by aryl, where the aryl radicals may in each case optionally be substituted;R.sup.2 represents hydrogen or methyl,R.sup.3 represents alkyl, alkenyl, alkinyl, alkoxyalkyl, hydroxyalkyl, hydroxyalkoxyalkyl, dialkoxyalkyl, or in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl, aralkyl, aralkenyl, furanylalkyl, tetrahydrofuranylalkyl, tetrahydropyranylalkyl, dioxolanylalkyl or dioxanylalkyl, andX represents oxygen, sulphur or a CH.sub.2 group,or acid addition salts thereof.Many of the compounds wherein R.sup.1 has a narrower meaning are new.
摘要翻译:用下式(Ⅰ)的氨基甲基杂环化合物与R1代表氢,烷基,烯基,各取代四氢萘基,十氢萘基,环烷基或环烯基,以及被环烷基,环烯基,环烷基 或环烷硫基,其中环状基团可任选被取代,此外任选取代的芳基,另外被芳基,芳氧基,芳硫基,芳基亚磺酰基或芳基磺酰基取代的烷基或被芳基取代的烯基,其中芳基可以在每种情况下 任选被取代; R 2表示氢或甲基,R 3表示烷基,烯基,炔基,烷氧基烷基,羟基烷基,羟基烷氧基烷基,二烷氧基烷基,或在每种情况下任选取代的环烷基,环烷基烷基,芳基,芳烷基,芳烯基,呋喃基烷基,四氢呋喃基烷基,四氢吡喃基烷基,二氧戊环烷基或二烷基烷基,X 代表氧,硫或CH2基,或其酸加成盐。 其中R1具有较窄含义的许多化合物是新的。
摘要:
Fungicidally active compounds of the formula ##STR1## in which X represents oxygen or sulphur,R represents cycloalkyl, or represents optionally substituted aryl, or represents the radical ##STR2## R.sup.1 and R.sup.2 each independently is hydrogen or an organic radical, or together with the nitrogen atom form a heterocyclic radical,R.sup.3 represents hydrogen, alkyl or optionally substituted aryl, andR.sup.4 represents alkyl or cycloalkyl, or represents optionally substituted aryl,but wherein R.sup.3 and R.sup.4 may not simultaneously represent methyl,and acid addition salts thereof, as well as intermediates therefor.
摘要:
Fungicidally active 2-aminomethyltetrahydrofurans of the formula ##STR1## in which R.sup.1 represents in each case optionally substituted aryl, heteroaryl, cycloalkyl, tetrahydronaphthyl or decahydronaphthyl;R.sup.2 represents hydrogen or methyl; andR.sup.3 and R.sup.4, independently of one another, in each case represent hydrogen, alkyl, alkenyl, alkinyl, alkoxyalkyl, dialkoxyalkyl, hydroxyalkyl, hydroxyalkoxyalkyl, dioxolanylalkyl, oxolanylalkyl, dioxanylalkyl, or in each case optionally substituted cycloalkylalkyl, cycloalkyl, aralkyl, aralkenyl or aryl, orR.sup.3 and R.sup.4, together with the nitrogen atom to which they are bound, represent an optionally substituted saturated heterocyclic ring which may optionally contain further heteroatoms,or acid-addition salts thereof.
摘要:
Novel fungicidally active decahydronaphth-2-yl-alkylamines of the formula ##STR1## in which A represents optionally substituted decahydronaphth-2-yl andR.sup.1 and R.sup.2 are identical or different and represent alkyl or alkenyl, orR.sup.1 and R.sup.2, together with the nitrogen atom to which they are bound, represent an optionally substituted, saturated heterocycle which may contain further hetero atoms,or a plant-tolerated acid-addition salts thereof.
摘要:
Fungicidally active novel .beta.-naphthylalkylamines of the formula ##STR1## in which Ar represents optionally substituted .beta.-naphthyl andR.sup.1 and R.sup.2, which can be identical or different, represent alkyl or alkenyl orR.sup.1 and R.sup.2, together with the nitrogen atom to which they are bonded, represent an optionally substituted saturated heterocyclic radical, which can contain further hetero-atoms,or plant-tolerated acid addition salts thereof.
摘要:
Substituted 4-piperidinomethyl-1,3-dioxolanes of the formula ##STR1## in which R.sup.1 is tetrahydronaphthyl, decahydronaphthyl, optionally substituted naphthyl, optionally substituted cycloalkyl or cycloalkenyl, optionally substituted phenyl, or alkyl which is substituted by in each case optionally substituted phenyl, phenoxy, phenylthio, cyclohexyl, cyclohexyloxy or cyclohexylthio,R.sup.2 is hydrogen or methyl,R.sup.3 is hydrogen or an acyl radicalor plant-tolerated addition products thereof with acids or metal salts, which possess fungicidal activity.
摘要:
Fungicidally active compounds of the formula ##STR1## in which X represents oxygen or sulphur,R represents cycloalkyl, or represents optionally substituted aryl, or represents the radical ##STR2## R.sup.1 and R.sup.2 each independently is hydrogen or an organic radical, or together with the nitrogen atom form a heterocyclic radical,R.sup.3 represents hydrogen, alkyl or optionally substituted aryl, andR.sup.4 represents alkyl or cycloalkyl, or represents optionally substituted aryl,but wherein R.sup.3 and R.sup.4 may not simultaneously represent methyl,and acid addition salts thereof, as well as intermediates therefor.
摘要:
Fungicidally active aminomethyl-isoxazolidines of the ##STR1## in which R.sup.1 represents optionally substituted alkyl, or represents optionally substituted cycloalkyl, or represents optionally substituted tetrahydronaphthyl, or represents optionally substituted decahydronaphthyl andR.sup.2 and R.sup.3 independently of one another each represent hydrogen, or represent in each case optionally substituted alkyl, alkenyl, cycloalkyl or aryl, or together with the nitrogen atom to which they are bonded represent an optionally substituted saturated heterocyclic radical, which can optionally contain further hetero atoms,and acid addition salts thereof. Some intermediates therefor are also new.
摘要:
Fungicidal saccharine salts of substituted hydroxypropylamines of the formula ##STR1## in which R.sup.1 is optionally substituted phenyl, phenoxy, phenylthio, phenylalkyl, phenoxyalkyl, or phenylthioalkyl, or optionally substituted cyclohexyl, cylohexyloxy, cyclohexylalkyl, cyclohexyloxyalkyl or cyclohexylthioalkyl,R.sup.2 is hydrogen or methyl,R.sup.3 is methyl or ethyl, andR.sup.4 and R.sup.5 each independently is alkyl or alkenyl, orR.sup.4 and R.sup.5, together with the nitrogen atom to which they are bonded, are an optionally substituted saturated heterocyclic radical which can optionally contain further hetero atoms.
摘要翻译:其中R 1为任选取代的苯基,苯氧基,苯硫基,苯基烷基,苯氧基烷基或苯硫基烷基,或任选取代的环己基,环己氧基,环己基烷基,环己氧基烷基或环己基硫代烷基,R 2为氢或甲基的取代羟基丙基胺的杀真菌糖精盐, R 3是甲基或乙基,R 4和R 5各自独立地是烷基或链烯基,或者R 4和R 5与它们所连接的氮原子一起是任选取代的饱和杂环基,其可以任选地含有另外的杂原子。