Pesticidal chromen-6-yl-methyl-oxy-and-thiapyrizinones
    11.
    发明授权
    Pesticidal chromen-6-yl-methyl-oxy-and-thiapyrizinones 失效
    杀虫铬-6-甲基 - 氧 - 和 - 硫杂环酮

    公开(公告)号:US5141939A

    公开(公告)日:1992-08-25

    申请号:US686084

    申请日:1991-04-09

    摘要: Pesticidal substituted pyridazinones of the formula ##STR1## in which R.sup.1 represents alkyl, halogenolkyl, alkoxyalkyl, alkylthioalkyl, (di)alkylaminoalkyl, alkenyl or halogenoalkenyl, or represents in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl or aralkyl,R.sup.2 represents halogen or alkyl,R.sup.3 and R.sup.4 independently of one another in each case represent hydrogen or alkyl,R.sup.5 and R.sup.6 represent hydrogen, carboxyl, in each case optionally substituted straight-chain or branched alkyl, alkenyl, alkoxycarbonyl, aryl or aralkyl, or, together with the carbon atom to which they are bonded, rpresent an optionally substituted saturated or unsaturaated carbocyle,R.sup.7, R.sup.8, R.sup.9, R.sup.10 and R.sup.11 independently of one another in each case represent hydrogen, halogen, alkyl, halogenoalkyl, alkoxy, halogenoalkoxy, alkylthio or halogenoalkylthio, andX represents oxygen or sulphur.Several intermediates therefor are also new.

    摘要翻译: R 1表示烷基,卤代烷基,烷氧基烷基,烷基硫代烷基,(二)烷基氨基烷基,烯基或卤代烯基的农药取代的哒嗪酮,或者表示任意取代的环烷基,环烷基烷基,芳基或芳烷基,R 2表示 卤素或烷基,R 3和R 4彼此独立地表示氢或烷基,R 5和R 6表示氢,羧基,在每种情况下均为任选取代的直链或支链烷基,烯基,烷氧基羰基,芳基或芳烷基,或一起 与它们所键合的碳原子相互独立地表示任选取代的饱和或不饱和碳环,R7,R8,R9,R10和R11彼此独立地表示氢,卤素,烷基,卤代烷基,烷氧基,卤代烷氧基,烷硫基或 卤代烷硫基,X表示氧或硫。 其中的几个也是新的。

    Pesticides based on substituted aminomethyl heterocyclic compounds
    12.
    发明授权
    Pesticides based on substituted aminomethyl heterocyclic compounds 失效
    基于取代氨基甲基杂环化合物的农药

    公开(公告)号:US5128368A

    公开(公告)日:1992-07-07

    申请号:US595143

    申请日:1990-10-10

    摘要: Combatting fungi and bacteria with aminomethylheterocyclic compounds of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkenyl, in each case optionally substituted tetrahydronaphthyl, decahydronaphthyl, cycloalkyl or cycloalkenyl, furthermore alkyl which is substituted by cycloalkyl, cycloalkenyl, cycloalkyloxy or cycloalkylthio, where the cyclic radicals may optionally be substituted, furthermore optionally substituted aryl, in addition alkyl which is substituted by aryl, aryloxy, arylthio, arylsulphinyl or arylsulphonyl, or alkenyl which is substituted by aryl, where the aryl radicals may in each case optionally be substituted;R.sup.2 represents hydrogen or methyl,R.sup.3 represents alkyl, alkenyl, alkinyl, alkoxyalkyl, hydroxyalkyl, hydroxyalkoxyalkyl, dialkoxyalkyl, or in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl, aralkyl, aralkenyl, furanylalkyl, tetrahydrofuranylalkyl, tetrahydropyranylalkyl, dioxolanylalkyl or dioxanylalkyl, andX represents oxygen, sulphur or a CH.sub.2 group,or acid addition salts thereof.Many of the compounds wherein R.sup.1 has a narrower meaning are new.

    摘要翻译: 用下式(Ⅰ)的氨基甲基杂环化合物与R1代表氢,烷基,烯基,各取代四氢萘基,十氢萘基,环烷基或环烯基,以及被环烷基,环烯基,环烷基 或环烷硫基,其中环状基团可任选被取代,此外任选取代的芳基,另外被芳基,芳氧基,芳硫基,芳基亚磺酰基或芳基磺酰基取代的烷基或被芳基取代的烯基,其中芳基可以在每种情况下 任选被取代; R 2表示氢或甲基,R 3表示烷基,烯基,炔基,烷氧基烷基,羟基烷基,羟基烷氧基烷基,二烷氧基烷基,或在每种情况下任选取代的环烷基,环烷基烷基,芳基,芳烷基,芳烯基,呋喃基烷基,四氢呋喃基烷基,四氢吡喃基烷基,二氧戊环烷基或二烷基烷基,X 代表氧,硫或CH2基,或其酸加成盐。 其中R1具有较窄含义的许多化合物是新的。

    2-aminomethyltetrahydrofurans, fungicidal compositions and use
    14.
    发明授权
    2-aminomethyltetrahydrofurans, fungicidal compositions and use 失效
    2-氨基甲基四氢呋喃,杀真菌剂和用途

    公开(公告)号:US4904656A

    公开(公告)日:1990-02-27

    申请号:US148395

    申请日:1988-01-25

    摘要: Fungicidally active 2-aminomethyltetrahydrofurans of the formula ##STR1## in which R.sup.1 represents in each case optionally substituted aryl, heteroaryl, cycloalkyl, tetrahydronaphthyl or decahydronaphthyl;R.sup.2 represents hydrogen or methyl; andR.sup.3 and R.sup.4, independently of one another, in each case represent hydrogen, alkyl, alkenyl, alkinyl, alkoxyalkyl, dialkoxyalkyl, hydroxyalkyl, hydroxyalkoxyalkyl, dioxolanylalkyl, oxolanylalkyl, dioxanylalkyl, or in each case optionally substituted cycloalkylalkyl, cycloalkyl, aralkyl, aralkenyl or aryl, orR.sup.3 and R.sup.4, together with the nitrogen atom to which they are bound, represent an optionally substituted saturated heterocyclic ring which may optionally contain further heteroatoms,or acid-addition salts thereof.

    摘要翻译: 式(I)的杀真菌活性2-氨基甲基四氢呋喃,其中R 1在每种情况下表示任选取代的芳基,杂芳基,环烷基,四氢萘基或十氢萘基; R2代表氢或甲基; 在各种情况下,R 3和R 4彼此独立地表示氢,烷基,烯基,炔基,烷氧基烷基,二烷氧基烷基,羟基烷基,羟基烷氧基烷基,二氧戊环烷基,氧代烷基烷基,二烷基烷基,或在各种情况下任选取代的环烷基烷基,环烷基,芳烷基, 芳基或R 3和R 4与它们所连接的氮原子一起代表任选取代的饱和杂环,其可任选地含有其它杂原子,或其酸加成盐。

    Pesticidal aminomethylheterocyclic compounds
    18.
    发明授权
    Pesticidal aminomethylheterocyclic compounds 失效
    杀虫氨基甲基杂环化合物

    公开(公告)号:US5177103A

    公开(公告)日:1993-01-05

    申请号:US616155

    申请日:1990-11-20

    摘要: Fungicidally active compounds of the formula ##STR1## in which X represents oxygen or sulphur,R represents cycloalkyl, or represents optionally substituted aryl, or represents the radical ##STR2## R.sup.1 and R.sup.2 each independently is hydrogen or an organic radical, or together with the nitrogen atom form a heterocyclic radical,R.sup.3 represents hydrogen, alkyl or optionally substituted aryl, andR.sup.4 represents alkyl or cycloalkyl, or represents optionally substituted aryl,but wherein R.sup.3 and R.sup.4 may not simultaneously represent methyl,and acid addition salts thereof, as well as intermediates therefor.

    摘要翻译: 式(I)的杀真菌活性化合物,其中X表示氧或硫,R表示环烷基,或表示任选取代的芳基,或表示基团R 1和R 2各自独立地为氢或有机基团,或 与氮原子一起形成杂环基,R 3表示氢,烷基或任选取代的芳基,R 4表示烷基或环烷基,或表示任选取代的芳基,但其中R 3和R 4可不同时表示甲基,及其酸加成盐, 以及其中间体。