Invention Grant
- Patent Title: Prodrugs of benzenesulfonamide-containing COX-2 inhibitors
- Patent Title (中): 含有苯磺酰胺的COX-2抑制剂的前药
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Application No.: US5610Application Date: 1998-01-12
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Publication No.: US5932598APublication Date: 1999-08-03
- Inventor: John J Talley , James W Malecha , Stephen Bertenshaw , Matthew J Graneto , Jeffery Carter , Jinglin Li , Srinivasan Nagarajan , David L Brown , Donald J Rogier, Jr. , Thomas D Penning , Ish K Khanna , Xiangdong Xu , Richard M Weier
- Applicant: John J Talley , James W Malecha , Stephen Bertenshaw , Matthew J Graneto , Jeffery Carter , Jinglin Li , Srinivasan Nagarajan , David L Brown , Donald J Rogier, Jr. , Thomas D Penning , Ish K Khanna , Xiangdong Xu , Richard M Weier
- Applicant Address: IL Skokie
- Assignee: G. D. Searle & Co.
- Current Assignee: G. D. Searle & Co.
- Current Assignee Address: IL Skokie
- Main IPC: C07D233/64
- IPC: C07D233/64 ; A61K31/00 ; A61K31/18 ; A61K31/34 ; A61K31/341 ; A61K31/365 ; A61K31/40 ; A61K31/415 ; A61K31/4162 ; A61K31/4164 ; A61K31/42 ; A61K31/421 ; A61K31/44 ; A61K31/4427 ; A61K31/4439 ; A61K31/635 ; A61P1/02 ; A61P1/04 ; A61P3/10 ; A61P5/16 ; A61P7/06 ; A61P9/10 ; A61P11/02 ; A61P11/06 ; A61P11/08 ; A61P13/12 ; A61P15/06 ; A61P17/02 ; A61P17/04 ; A61P17/06 ; A61P19/02 ; A61P19/08 ; A61P21/00 ; A61P21/04 ; A61P25/00 ; A61P25/04 ; A61P25/28 ; A61P27/02 ; A61P27/12 ; A61P29/00 ; A61P29/02 ; A61P31/12 ; A61P35/00 ; A61P37/00 ; A61P43/00 ; C07C311/16 ; C07C311/39 ; C07C311/51 ; C07D20060101 ; C07D207/32 ; C07D207/327 ; C07D207/33 ; C07D231/12 ; C07D233/54 ; C07D233/62 ; C07D261/08 ; C07D263/32 ; C07D307/46 ; C07D307/58 ; C07D401/04 ; C07D417/04 ; C07D495/04 ; A61K31/16 ; C07D207/00 ; C07D207/12 ; C07D211/72 ; C07D211/84 ; C07D223/04 ; C07D231/10 ; C07D403/02
Abstract:
Prodrugs of COX-2 inhibitors are described as being useful in treating inflammation and inflammation-related disorders.
Public/Granted literature
- USD355524S High heeled sneaker Public/Granted day:1995-02-21
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