公开(公告)号：US06686469B2

公开(公告)日：2004-02-03

申请号：US10011012

申请日：2001-11-05

Applicant: Martin Eberle ,  André Jeanguenat ,  Werner Zambach ,  Arthur Steiger ,  Saleem Farooq

Inventor： Martin Eberle ,  André Jeanguenat ,  Werner Zambach ,  Arthur Steiger ,  Saleem Farooq

IPC: C07D2412

CPC classification number: C07D239/26 ,  A01N43/54 ,  C07D239/28 ,  C07D239/34 ,  C07D239/36 ,  C07D239/42 ,  C07D239/54

Abstract: The invention relates to compounds of the general formula wherein R1 is unsubstituted or mono- to penta-substituted aryl, whereby the substituents are selected from the group consisting for instance of OH, Halogen, CN, C1-C6-alkyl, optionally substituted C3-C8-cycloalkyl and optionally substituted C3-C8-cycloalkenyl; A is for instance a single bond, C1-C12-alkylene or O; X1 and X2, independently of one another, are R10; X3 is H or R10; R10 is for instance halogen, CN, NO2, C1-C6-alkyl, C3-C8-cycloalkyl or C1-C6-haloalkyl; R21 and R22, independently of one another are for instance H, halogen, CN, NO2, OH, SH, C1-C6-alkyl, C3-C8-cycloalkyl, C1-C6-alkyl-C3-C8-cycloalkyl or C3-C8-cycloalkyl-C1-C6-alkyl; R23 and R24, independently of one another, are for instance H, C1-C6-alkyl, C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C6-alkyl, C1-C6-haloalkyl or C3-C8-halocycloalkyl; m is 1, 2, 3 or 4; and n is 0, 1 or 2; as well as the physiologically acceptable addition compounds, a method of producing these compounds and the usage of these compounds, pesticide compositions whose active ingredient is chosen from these compounds, each in free form or in agrochemically employable salt form, and a method of producing and using these compositions. The active ingredients, in free form or in agrochemically employable salt form, have advantageous pesticidal properties. The are especially suitable for the control of pests in agriculture and in storage, as well as in the care of domestic animals.

Abstract translation: 本发明涉及通式为化学式R 1的化合物是未取代的或一至五取代的芳基，其中取代基选自例如OH，卤素，CN，C 1 -C 6 - 烷基，任选取代的C 3 -C 8 - 环烷基和任选取代的C 3 -C 8 - 环烯基; A为例如单键，C 1 -C 12 - 亚烷基或O; X 1和X 2彼此独立地为R 10; X3为H或R10; R10为卤素，CN，NO2，C1-C6-烷基，C3-C8-环烷基或C1-C6-卤代烷基; R21和R22彼此独立地为例如H，卤素，CN ，NO 2，OH，SH，C 1 -C 6烷基，C 3 -C 8 - 环烷基，C 1 -C 6烷基-C 3 -C 8 - 环烷基或C 3 -C 8环烷基-C 1 -C 6烷基; R 23和R 24独立地为 另一个例子是H，C 1 -C 6烷基，C 3 -C 8环烷基，C 3 -C 8环烷基-C 1 -C 6烷基，C 1 -C 6卤代烷基或C 3 -C 8卤代环烷基; m是1,2,3 或4; 和n为0,1或2;以及生理上可接受的加成化合物，这些化合物的制备方法和这些化合物的用途，其活性成分选自这些化合物的农药组合物，各自为游离形式或农业化学可使用的盐 形式，以及生产和使用这些组合物的方法。 活性成分，游离形式或具有农业化学应用的盐形式，具有有利的杀虫特性。 特别适用于农业，仓储以及家畜照顾中的害虫控制。