公开(公告)号：US20220033384A1

公开(公告)日：2022-02-03

申请号：US17500866

申请日：2021-10-13

Applicant: Nippon Soda Co., Ltd.

Inventor： Keita SAKANISHI ,  Takao IWASA ,  Hikaru AOYAMA ,  Norifumi SAKIYAMA ,  Daisuke USHIJIMA ,  Maki MATSUI ,  Tomomi KOBAYASHI

IPC: C07D403/14 ,  C07D401/14 ,  A01N43/50 ,  A01N43/54 ,  C07D233/64 ,  C07D403/04 ,  C07D401/04 ,  A61P31/10 ,  A01N43/56 ,  C07D403/10 ,  A61P31/14 ,  A01N43/653 ,  C07D413/10 ,  A61K31/506

Abstract: A compound represented by Formula (I), or a salt thereof: wherein, R1 represents an unsubstituted or substituted C1-6 alkylthio group, or the like; A1 represents a nitrogen atom or CH; A2 represents a nitrogen atom or CR2; R2 and R3 each independently represents a hydrogen atom, an unsubstituted or substituted C6-10 aryl group, an unsubstituted or substituted 3- to 6-membered heterocyclyl group, or the like; B1 and B2 each independently represents a nitrogen atom or CR5, with the proviso that B1 and B2 do not represent CR5 at the same time, wherein R5 represents a hydrogen atom, an unsubstituted or substituted C1-6 alkyl group, or the like; R4 represents an unsubstituted or substituted C1-6 alkyl group, or the like, and R4 binds to any one of nitrogen atoms forming an imidazole ring or a triazole ring; and Ar represents an unsubstituted or substituted C6-10 aryl group or the like.

公开(公告)号：US20210380556A1

公开(公告)日：2021-12-09

申请号：US17280655

申请日：2019-09-30

Applicant: Nippon Soda Co., Ltd.

Inventor： Keita SAKANISHI ,  Norifumi SAKIYAMA ,  Hikaru AOYAMA ,  Takao IWASA ,  Maki MATSUI ,  Tomomi KOBAYASHI ,  Daisuke USHIJIMA

IPC: C07D401/14 ,  A01N43/54 ,  A01N43/653 ,  A01N43/50 ,  C07D401/04 ,  A01N25/00 ,  A01N25/12

Abstract: An object of the present invention is to provide a heteroaryl azole compound that is excellent in pest control activity, particularly, insecticidal activity and/or miticidal activity, is excellent in safety, and may be industrially advantageously synthesized. The compound of the present invention is a compound represented by the formula (I), an N-oxide compound, stereoisomer, tautomer or hydrate thereof or a salt of any of these compounds. In the formula (I), A represents CH or a nitrogen atom; B1 represents CX1 or a nitrogen atom; X1, X2 and X3 each independently represent a hydrogen atom, a substituted or unsubstituted C1-6 alkyl group, a substituted or unsubstituted C2-6 alkenyl group, or the like; R1 represents a substituted or unsubstituted C1-6 alkylthio group, a substituted or unsubstituted C1-6 alkylsulfinyl group, or the like; R2 represents a substituted or unsubstituted C1-6 alkyl group; and R represents a substituted or unsubstituted C1-6 alkyl group.

公开(公告)号：US20240327377A1

公开(公告)日：2024-10-03

申请号：US18743634

申请日：2024-06-14

Applicant: NIPPON SODA CO., LTD.

Inventor： Keita SAKANISHI ,  Hikaru AOYAMA ,  Daisuke USHIJIMA ,  Takao IWASA ,  Norifumi SAKIYAMA ,  Maki MATSUI

IPC: C07D401/04 ,  A01N43/50 ,  A01N43/54 ,  A01N43/653 ,  C07D233/64 ,  C07D401/14

CPC classification number: C07D401/04 ,  A01N43/50 ,  A01N43/54 ,  A01N43/653 ,  C07D233/64 ,  C07D401/14

Abstract: An object of the present invention is to provide a heteroaryl azole compound that is excellent in pest control activity, particularly, insecticidal activity and/or miticidal activity, is excellent in safety, and may be industrially advantageously synthesized. The heteroaryl azole compound of the present invention is a compound of the following formula (II), an N-oxide compound, stereoisomer, tautomer or hydrate thereof, or a salt of any of these compounds. Here, in the formula (II), R1 represents a substituted or unsubstituted C1-6 alkylthio group or the like; B1 represents a nitrogen atom or CR2; R2 represents a hydrogen atom, a substituted or unsubstituted C1-6 alkyl group or the like; R3 represents a hydrogen atom, a substituted or unsubstituted C1-6 alkyl group or the like; R represents a substituted or unsubstituted C1-6 alkyl group or the like; A represents a carbon atom or a nitrogen atom; X represents a substituted or unsubstituted C1-6 alkyl group or the like; n represents a number of chemically acceptable X, and is an integer of 0 to 2; and X is the same or different when n is 2.

公开(公告)号：US20190185459A1

公开(公告)日：2019-06-20

申请号：US16329198

申请日：2017-09-13

Applicant: Nippon Soda Co., Ltd.

Inventor： Keita SAKANISHI ,  Takao IWASA ,  Hikaru AOYAMA ,  Norifumi SAKIYAMA ,  Daisuke USHIJIMA ,  Maki MATSUI ,  Tomomi KOBAYASHI

IPC: C07D403/14 ,  C07D233/64 ,  C07D403/04 ,  C07D401/14 ,  A01N43/50 ,  A01N43/54

CPC classification number: C07D403/14 ,  A01N25/04 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/78 ,  A61K31/4439 ,  A61K31/506 ,  A61P31/10 ,  A61P31/14 ,  C07D233/64 ,  C07D401/04 ,  C07D401/14 ,  C07D403/04 ,  C07D403/10 ,  C07D413/10

Abstract: A compound represented by Formula (I), or a salt thereof: wherein, R1 represents an unsubstituted or substituted C1-6 alkylthio group, or the like; A1 represents a nitrogen atom or CH; A2 represents a nitrogen atom or CR2; R2 and R3 each independently represents a hydrogen atom, an unsubstituted or substituted C6-10 aryl group, an unsubstituted or substituted 3- to 6-membered heterocyclyl group, or the like; B1 and B2 each independently represents a nitrogen atom or CR5, with the proviso that B1 and B2 do not represent CR5 at the same time, wherein R5 represents a hydrogen atom, an unsubstituted or substituted C1-6 alkyl group, or the like; R4 represents an unsubstituted or substituted C1-6 alkyl group, or the like, and R4 binds to any one of nitrogen atoms forming an imidazole ring or a triazole ring; and Ar represents an unsubstituted or substituted C6-10 aryl group or the like.

公开(公告)号：US20220061325A1

公开(公告)日：2022-03-03

申请号：US17432870

申请日：2020-02-25

Applicant: Nippon Soda Co., Ltd.

Inventor： Takashi KITAYAMA ,  Keita SAKANISHI ,  Koichi HIRATA ,  Maki MATSUI ,  Hikaru AOYAMA

IPC: A01N43/90 ,  A01P7/04 ,  A01P7/02 ,  C07D413/04 ,  C07D417/04 ,  C07D401/04 ,  C07D498/04 ,  C07D513/04 ,  C07D471/04 ,  A01N43/76 ,  A01N43/78

Abstract: An object of the present invention is to provide a pyridine N-oxide compound that is excellent in pest control activity, particularly, insecticidal activity and/or acaricidal activity, is excellent in safety, and may be industrially advantageously synthesized. The pyridine N-oxide compound of the present invention is a compound of the formula (II), a stereoisomer, tautomer or hydrate thereof or a salt of any of these compounds, wherein R1 represents a substituted or unsubstituted C1-6 alkylsulfonyl group; R2 represents a hydrogen atom, a substituted or unsubstituted C1-6 alkyl group, or the like; A1 represents an oxygen atom, a sulfur atom, or the like; A2 and A3 each independently represent a carbon atom or a nitrogen atom; X represents a substituted or unsubstituted C1-6 alkyl group, a substituted or unsubstituted C1-6 alkoxy group, or the like; and n represents an integer of 0 to 2.

公开(公告)号：US20210380554A1

公开(公告)日：2021-12-09

申请号：US17286888

申请日：2019-10-23

Applicant: Nippon Soda Co., Ltd.

Inventor： Keita SAKANISHI ,  Norifumi SAKIYAMA ,  Hikaru AOYAMA ,  Maki MATSUI ,  Takao IWASA ,  Tomomi KOBAYASHI ,  Daisuke USHIJIMA ,  Keita AZUMA ,  Masanori SUMINO ,  Yasuhiko ASHIKARI ,  Kotaro SHIBAYAMA ,  Riho TAGUCHI

IPC: C07D401/04 ,  A01N43/50

Abstract: An object of the present invention is to provide a (hetero)aryl imidazole compound that is excellent in pest control activity, particularly, insecticidal activity and/or acaricidal activity, is excellent in safety, and may be industrially advantageously synthesized. The (hetero)aryl imidazole compound of the present invention is a compound represented by the formula (I) an N-oxide compound, stereoisomer, tautomer or hydrate thereof or a salt of any of these compounds. In the formula (I), B1 represents a nitrogen atom or CH; X represents a substituted or unsubstituted C3-8 cycloalkyl group; R1 represents a substituted or unsubstituted C1-6 alkylthio group or a substituted or unsubstituted C1-6 alkylsulfonyl group; R2 represents a substituted or unsubstituted C1-6 alkyl group; and R represents a substituted or unsubstituted C2-6 alkenyl group.

公开(公告)号：US20210002263A1

公开(公告)日：2021-01-07

申请号：US16975907

申请日：2019-03-08

Applicant: Nippon Soda Co., Ltd.

Inventor： Keita SAKANISHI ,  Hikaru AOYAMA ,  Norifumi SAKIYAMA ,  Takao IWASA ,  Maki MATSUI ,  Tomomi KOBAYASHI ,  Takashi KITAYAMA

IPC: C07D403/14 ,  C07D413/14 ,  A01N43/76 ,  A01N43/90

Abstract: The present invention relates to a compound represented by the following Formula (I) or a salt thereof, which exhibits superior insecticidal activity, acaricidal activity, and/or nematicidal activity, which exhibits superior safety, and which can be advantageously synthesized industrially, and also relates to a formulation for controlling harmful organisms containing the same as an active ingredient. wherein, X represents a halogeno group, a substituted or unsubstituted C1-6 alkyl group, or the like; n is an integer ranging from 1 to 3; Z represents an oxygen atom, a sulfur atom, or NR; R represents a hydrogen atom or a substituted or unsubstituted C1-6 alkyl group; A represents a benzene ring or a 6-membered heteroaryl ring; Ra represents a substituted or unsubstituted C1-6 alkylsulfonyl group; and Rb represents a substituted or unsubstituted C1-6 alkyl group, and the like.

公开(公告)号：US20180160686A1

公开(公告)日：2018-06-14

申请号：US15735713

申请日：2016-06-17

Applicant: Nippon Soda Co., Ltd.

Inventor： Hikaru AOYAMA ,  Maki MATSUI ,  Keita SAKANISHI ,  Takao IWASA ,  Tomomi KOBAYASHI ,  Koichi HIRATA

IPC: A01N43/56 ,  A01N43/653 ,  A01N43/90 ,  A01N47/18 ,  C07D231/12 ,  C07D231/16 ,  C07D231/40 ,  C07D249/06 ,  C07D401/04 ,  C07D403/04

Abstract: The present invention provides a compound represented by formula (I), (in the formula, A1 and A2 each independently represents a carbon atom or a nitrogen atom; X1 represents an unsubstituted or substituted C1-6 alkyl group or the like; n represents an integer of 0 to 4; R1 represents an unsubstituted or substituted C1-6 alkylthio group or the like; B1 and B4 each independently represent a carbon atom, a nitrogen atom or the like; R2 and R3 each independently represent a hydrogen atom, a halogeno group or the like; Ar represents an unsubstituted or substituted C6-10 aryl group or the like) or a salt thereof, and a harmful organism control agent including thereof.

公开(公告)号：US20220000112A1

公开(公告)日：2022-01-06

申请号：US17476407

申请日：2021-09-15

Applicant: Nippon Soda Co., Ltd.

Inventor： Hikaru Aoyama ,  Maki MATSUI ,  Takao IWASA ,  Kazushige FUJII ,  Tomomi KOBAYASHI ,  Keita SAKANISHI

IPC: A01N43/50 ,  A61K31/4164 ,  A61K31/4439 ,  C07D233/64 ,  C07D401/04 ,  A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/74 ,  C07D401/14 ,  C07D403/04 ,  C07D405/04 ,  C07D409/04 ,  C07D417/14

Abstract: The present invention provides a compound represented by formula (I) or salt thereof (in the formula, A1 and A2 each independently represents a nitrogen atom or the like, B1, B2, B3 and B4 each independently represents a carbon atom or nitrogen atom, X1 represents an unsubstituted or substituted C1-6 alkyl group or the like, n represents a number of X1 and represents an integer of 0-4, R1 represents a halogeno group or the like, R2 represents an unsubstituted or substituted C1-6 alkyl group or the like, m represents a number of the oxide group bonding with the nitrogen atom which does not bond with R2 on the imidazole ring, and represents 0 or 1, R3 represents a hydrogen atom or the like, Ar represents an unsubstituted or substituted C6-10 aryl group.

公开(公告)号：US20210269415A1

公开(公告)日：2021-09-02

申请号：US17271531

申请日：2019-09-02

Applicant: NIPPON SODA CO., LTD.

Inventor： Keita SAKANISHI ,  Hikaru AOYAMA ,  Daisuke USHIJIMA ,  Takao IWASA ,  Norifumi SAKIYAMA ,  Maki MATSUI

IPC: C07D401/04 ,  C07D401/14 ,  A01N43/653 ,  A01N43/54 ,  A01N43/50 ,  C07D233/64

Abstract: A heteroaryl azole compound of the following formula (II): an N-oxide compound, stereoisomer, tautomer or hydrate thereof, or a salt of any of these compounds. In the formula (II), R1 represents a substituted or unsubstituted C1-6 alkylthio group or the like; B1 represents a nitrogen atom or CR2; R2 represents a hydrogen atom, a substituted or unsubstituted C1-6 alkyl group or the like; R3 represents a hydrogen atom, a substituted or unsubstituted C1-6 alkyl group or the like; R represents a substituted or unsubstituted C1-6 alkyl group or the like; A represents a carbon atom or a nitrogen atom; X represents a substituted or unsubstituted C1-6 alkyl group or the like; n represents a number of chemically acceptable X, and is an integer of 0 to 2; and X is the same or different when n is 2.