摘要:
Organic compounds of the class vinyl substituted phthalans are preared chemically from the corresponding vinyl isobenzofurylium compounds. The novel compounds are useful for their antidepressant activity.
摘要:
THIS INVENTION DESCRIBES NEW SUBSTITUTED INDOLE COMPOUNDS. INTERMEDIATE 3-HALODICARBONYL INDOLES ARE ALSO DESCRIBED. THE PREPARATION OF THE FINAL PRODUCTS FROM THE 3-HALODICARBONYL INDOLES WHEREIN THE 3-POSITION CONTAINS A DISUBSTITUTED B-AMINOETHYL GROUP IS DESCRIBED. THE COMPOUNDS HAVE UTILITY AS CENTRAL NERVOUS SYSTEM DEPRESSANTS, ANALGESICS, ANTI-INFLAMMATORY AGENTS, AND DIURETIC AGENTS.
摘要:
THE PREPARATION OF 4A,7,8,9A-TETRAHYDRO-9A-HYDROXYCARBAZOLE-3,4-(4H,6H)-DIONES BY REACTION OF A 2-TRIFLUOROMETHYL-1,4-BENZOQUINONE WITH AN AMINO OR LOWER ALKYLAMINO-2-CYCLOHEXEN-1-ONE, IS DESCRIBED. THE COMPOUNDS ARE PHYSIOLOGICALLY ACTIVE ON THE CENTRAL NERVOUS SYSTEM AND ARE USEFUL AS TRANQUILIZERS.
摘要:
THE PREPARATION OF SUBSTITUTED AMINO ALKYLENETETRAHYDROCARBAZOLES BY REACTING A 2,3-DIHYDROCARBAZOLONE WITH PARAFORMALDEHYDE AND AN AMINE AND SUBSEQUENTIALLY SUBJECTING THE REACTION PRODUCT TO REDUCTION, IS DESCRIBED. THE PRODUCTS ARE USEFUL FOR THEIR CENTRAL NERVOUS SYSTEM ACTIVITY AS TRANQUILIZERS.
摘要:
PREPARATION OF SUBSTITUTED TETRAHYDROCARBAZOLECARBOXYLIC DERIVATIVES, ARE DESCRIBED. THEY ARE USEFUL FOR THEIR CENTRAL NERVOUS SYSTEM ACTIVITY, AS ANTICONVULSANTS.
摘要:
THE PREPARATION OF 11-SUBSTITUTED 2-TRIFLUOROMETHOXYDIEBENZ(B,F)(1,4)OXAPZEPINES; 11-SUBSTITUTED 2-TRIFLUOROMETHOXY-DIBENZ(B,F)(1,4)THIAZEPINES AND 11-SUBSTITUTED 2-TRIFLUOROMETHOXY DIBENZ (B,F)(1,4) DIAZEPINES, BY RING CLOSURE OF SUITABLE INTERMEDIATES, IS DESCRIBED. THE NOVEL COMPOUNDS ARE USEFUL AS ANTI-DEPRESSANTS, ANTI-INFLAMMATORY AND ANTI-PYRETIC AGENTS.