知搜-全球专利检索

  1. 登录
  2. 注册

搜索结果

61 条记录 (耗时 0.082 秒)

    Benzimidazole compounds and drugs containing the same
    1.
    发明授权
    Benzimidazole compounds and drugs containing the same 失效
    苯并咪唑化合物和含有相同的药物

    公开(公告)号：US06815455B1

    公开(公告)日：2004-11-09

    申请号：US10019249

    申请日：2002-06-05

    申请人： Kozo Aoki ,  Kazuhiro Aikawa ,  Masayuki Kawakami ,  Yongzhe Yan

    发明人： Kozo Aoki ,  Kazuhiro Aikawa ,  Masayuki Kawakami ,  Yongzhe Yan

    IPC分类号： A61K31454

    CPC分类号： C07D401/12

    摘要： A benzimidazole compound or a salt thereof which has an inhibitory action of foaming of macrophages and is useful as an active ingredient of a medicament for preventive and/or therapeutic treatment of arteriosclerosis, which is represented by the formula (I): wherein R1 represents a hydrogen atom, a halogen atom, a lower alkyl group, or a lower alkoxy group; R2 represents a hydrogen atom, an alkyl group, or an acyl group; R3 represents a functional group on the ring; A represents O or CH2 or CH that forms a double bond with an adjacent carbon atom; L represents a C4-C8 alkylene group or an ethyleneoxy linking group represented by (CH2CH2O)nCH2CH2 wherein n represents 1 or 2; X represents O, S or methylene group; and m represents 0 or 1.

    Benzimidazole compounds
    2.
    发明授权
    Benzimidazole compounds 失效
    苯并咪唑化合物

    公开(公告)号：US06787561B1

    公开(公告)日：2004-09-07

    申请号：US10019668

    申请日：2002-06-05

    申请人： Kozo Aoki ,  Kazuhiro Aikawa ,  Masayuki Kawakami ,  Yongzhe Yan

    发明人： Kozo Aoki ,  Kazuhiro Aikawa ,  Masayuki Kawakami ,  Yongzhe Yan

    IPC分类号： A61K314439

    CPC分类号： C07D401/12 ,  C07D235/28 ,  C07D403/12 ,  C07D413/12 ,  C07D417/12

    摘要： A benzimidazole compound or a salt thereof which has an inhibitory action of forming of macrophages and is useful as an active ingredient of an orally available medicament for preventive and/or therapeutic treatment of arteriosclerosis, which is represented by the formula (I): wherein, R1 represents one or more functional groups on the benzene ring selected from the group consisting of hydrogen atom, a halogen atom, a lower alkyl group and a lower alkoxy group; R2 represents hydrogen atom, an alkyl group or an acyl group; L represents a C4-C8 alkylene group or an ethyleneoxy linking group represented as (CH2CH2O)nCH2CH2 wherein n represents 1 or 2; X represents O or NH; Y represents S or a single bond; and Q represents a 5- or 6-membered heterocyclic group which may have a functional group on the ring.

    摘要翻译： 具有抑制巨噬细胞形成作用的苯并咪唑化合物或其盐，可用作由式（I）表示的用于预防和/或治疗动脉硬化的口服药物的活性成分：其中， R 1表示选自氢原子，卤素原子，低级烷基和低级烷氧基的苯环上的一个或多个官能团; R 2表示氢原子，烷基或酰基; L表示作为（CH 2 CH 2 O）n CH 2 CH 2表示的C 4 -C 8亚烷基或亚乙氧基连接基，其中n表示1或2; X表示O或NH; Y表示S或单键; Q表示在环上可具有官能团的5或6元杂环基。

    Silver halide color photographic light-sensitive material
    4.
    发明授权
    Silver halide color photographic light-sensitive material 失效
    卤化银彩色摄影感光材料

    公开(公告)号：US5260177A

    公开(公告)日：1993-11-09

    申请号：US884897

    申请日：1992-05-18

    申请人： Kozo Aoki ,  Michio Ono ,  Katsuyoshi Yamakawa ,  Shigeru Yamazaki ,  Kei Sakanoue ,  Hidetoshi Kobayashi

    发明人： Kozo Aoki ,  Michio Ono ,  Katsuyoshi Yamakawa ,  Shigeru Yamazaki ,  Kei Sakanoue ,  Hidetoshi Kobayashi

    IPC分类号： C07D213/75 ,  C07D213/76 ,  C07D471/04 ,  G03C7/38 ,  G03C7/388

    CPC分类号： C07D213/75 ,  C07D213/76 ,  C07D471/04 ,  G03C7/3815

    摘要： A silver halide color photographic light-sensitive material comprises a novel cyan dye-forming coupler or a combination of a specific cyan dye-forming coupler with an .alpha.-pivaloylacetoanilide type yellow dye-forming coupler or a pyrazoloazole type magenta dye-forming coupler, the specific cyan dye-forming coupler being contained in the silver halide emulsion layer in the form of an emulsion of lipophilic fine particles obtained by mixing the coupler with at least one water-insoluble and organic solvent-soluble homo- or co-polymer to form a dispersion. The silver halide color photographic light-sensitive material is excellent in the reproduction of yellow, magenta and cyan colors and has low fog of cyan. Thus, the light-sensitive material can provide color images excellent in the fastness of the cyan color images.The cyan dye-forming coupler is represented by general formula (II): ##STR1## wherein R.sub.1 represents an aliphatic group, an aromatic group or a heterocyclic group; R.sub.2 represents a group or atom which can be bonded with the heterocyclic ring; X represents a hydrogen atom or a group which can be eliminated; Y represents a divalent bonding group having at least one amido bond and/or ester bond; Z represents a dissociative group; A, B, C, D and E each represents a nitrogen atom or a carbon atom a which hydrogen atom is bonded, provided that one or two of them represent a nitrogen atom; and n represents 0, 1 or 2.

    摘要翻译： 卤化银彩色照相感光材料包括新型的青色染料形成成色剂或特定的形成青色染料的成色剂与α-对甲酰基乙酰苯胺型黄色染料形成成色剂或吡唑并唑型品红色染料形成成色剂的组合， 通过将成色剂与至少一种水不溶性和有机溶剂可溶性均聚物或共聚物混合而形成的亲脂性细颗粒乳液形式的卤化银乳剂层中所含有特定的青色成色剂， 分散。 卤化银彩色摄影感光材料在黄色，品红色和青色的再现方面是优异的，并且具有低的青色雾。 因此，感光材料可以提供在青色图像的牢度方面优异的彩色图像。 青色染料成色剂由通式（II）表示：其中R 1表示脂族基团，芳族基团或杂环基团; R2表示可以与杂环结合的基团或原子; X表示氢原子或可被除去的基团; Y表示具有至少一个酰胺键和/或酯键的二价键合基​​团; Z表示离解基团; A，B，C，D和E各自表示氮原子或氢原子键合的碳原子a，条件是它们中的一个或两个表示氮原子; n表示0,1或2。

    Silver halide color photographic material containing 5-pyrazolone magenta coupler and amine-type stain preventing agent
    5.
    发明授权
    Silver halide color photographic material containing 5-pyrazolone magenta coupler and amine-type stain preventing agent 失效
    含有5-吡唑啉酮品红成色剂和胺型防污剂的卤化银彩色照相材料

    公开(公告)号：US5096805A

    公开(公告)日：1992-03-17

    申请号：US683503

    申请日：1991-04-05

    申请人： Kozo Aoki ,  Masakazu Morigaki

    发明人： Kozo Aoki ,  Masakazu Morigaki

    IPC分类号： G03C7/26 ,  G03C7/30 ,  G03C7/305 ,  G03C7/32 ,  G03C7/384 ,  G03C7/392

    CPC分类号： G03C7/30529 ,  G03C7/3012 ,  G03C7/3225

    摘要： A silver halide color photographic material containing at least one silver halide emulsion and at least one kind of 5-pyrazolone couplers having the releasable group shown by following formula (I) at the coupling position and at least one kind of the compounds shown by following formula (II): ##STR1## wherein L.sub.1 and L.sub.2 each represents a methylene group or an ethylene group; l and m each represents 0 or 1; R.sub.1 represents a hydrogen atom, an alkyl group, an aryl group, or a heterocyclic group; R.sub.2 represents a group bonded to A by a carbon atom, an oxygen atom, a nitrogen atom or a sulfur atom; A represents a carbon atom or a sulfur atom; n represents 1 when A is a carbon atom, or 1 or 2 when A is a sulfur atom; B represents a carbon atom, an oxygen atom, a nitrogen atom, or a sulfur atom; and X represents an atomic group necessary for forming a ring; said R.sub.1 and R.sub.2 may combine with each other to form a ring; and when B is a carbon atom or a nitrogen atom, said B and R.sub.2 may combine with each other to form a ring; ##STR2## wherein R.sub.21 represents a hydrogen atom, a hydroxy group, or a substituted or unsubstituted alkyl, alkenyl, alkoxy, acyl, aryloxy, heterocyclic oxy or acyloxy group and R.sub.22 and R.sub.23 each represents a substituted or unsubstituted alkyl, alkenyl or heterocyclic group; said R.sub.21, R.sub.22 and R.sub.23 may form together a nitrogen-containing monocyclic or polycyclic heterocyclic ring and the sum of the carbon atom numbers of R.sub.21, R.sub.22, and R.sub.23 is at least 10.

    摘要翻译： 含有至少一种卤化银乳剂和至少一种在偶合位置具有下式（I）所示的可释放基团的5-吡唑啉酮成色剂的卤化银彩色照相材料和至少一种下式所示的化合物 （II）：其中L 1和L 2各自表示亚甲基或亚乙基; l和m各自表示0或1; R1表示氢原子，烷基，芳基或杂环基; R2表示通过碳原子，氧原子，氮原子或硫原子与A键合的基团; A表示碳原子或硫原子; 当A为碳原子时，n表示1，A为硫原子时为1或2。 B表示碳原子，氧原子，氮原子或硫原子; X表示形成环所需的原子团; 所述R1和R2可以相互结合形成环; 当B为碳原子或氮原子时，所述B和R2可以相互结合形成环; （II）其中R21表示氢原子，羟基或取代或未取代的烷基，烯基，烷氧基，酰基，芳氧基，杂环氧基或酰氧基，R22和R23各自表示取代或未取代的烷基，烯基 或杂环基; 所述R 21，R 22和R 23可以一起形成含氮单环或多环杂环，R 21，R 22和R 23的碳原子数之和至少为10。

    Color photographic light-sensitive material
    6.
    发明授权
    Color photographic light-sensitive material 失效
    彩色摄影感光材料

    公开(公告)号：US5084375A

    公开(公告)日：1992-01-28

    申请号：US918659

    申请日：1986-10-15

    申请人： Makoto Umemoto ,  Kozo Aoki

    发明人： Makoto Umemoto ,  Kozo Aoki

    IPC分类号： G03C7/32 ,  G03C7/34

    CPC分类号： G03C7/342

    摘要： A color photographic light-sensitive material comprising a support having provided thereon a silver halide emulsion layer containing at least one each of cyan color image forming couplers represented by the following general formulae (I) and (II): ##STR1## and at least one compound represented by the formulae (III) or (IV): ##STR2## wherein all the symbols are defined in the specification.

    摘要翻译： 一种彩色摄影感光材料，其包括在其上设置有包含由以下通式（I）和（II）表示的青色成像成色剂中的至少一种的卤化银乳剂层的载体： （II）和至少一种由式（III）或（IV）表示的化合物：其中所有符号在说明书中定义。

    Silver halide photographic material
    7.
    发明授权
    Silver halide photographic material 失效

    公开(公告)号：US5009989A

    公开(公告)日：1991-04-23

    申请号：US246585

    申请日：1988-09-19

    申请人： Kozo Aoki ,  Osamu Takahashi

    发明人： Kozo Aoki ,  Osamu Takahashi

    IPC分类号： G03C7/26 ,  G03C7/30 ,  G03C7/34 ,  G03C7/392

    CPC分类号： G03C7/39232 ,  G03C7/3005 ,  G03C7/34

    摘要： A silver halide photographic material which contains, on a support, a combination of at least one cyan dye-forming coupler represented by the following formula (I) and at least one compound selected from among those represented by the following formulae (II) and (III), whereby achieving enhancement of keeping quality of the developed cyan color dye: ##STR1## wherein R.sub.1 represents an aliphatic group, an aromatic group or a heterocyclic group; R.sub.2 representing an alkyl group containing from 2 to 15 carbon atoms; Z represents a hydrogen atom, or a group or an atom capable of splitting off upon coupling with a developing agent; L.sub.1 and L.sub.2 each represents a divalent to a tetravalent aliphatic group; R.sub.3 and R.sub.4 each represents an aliphatic group, an aromatic group, or a heterocyclic group; and n and m each represents an integer of from 2 to 4, and therein the n R.sub.3 's and m R.sub.4 's, respectively, may be the same or different, and when m represents 2, L.sub.2 excludes a cyclohexylene group.

    Silver halide color photographic material
    8.
    发明授权
    Silver halide color photographic material 失效
    卤化银彩色照相材料

    公开(公告)号：US4929538A

    公开(公告)日：1990-05-29

    申请号：US102511

    申请日：1987-09-29

    申请人： Masakazu Morigaki ,  Kozo Aoki

    发明人： Masakazu Morigaki ,  Kozo Aoki

    IPC分类号： G03C7/32 ,  G03C7/26 ,  G03C7/30

    CPC分类号： G03C7/3006

    摘要： A novel silver halide color photographic material is provided, containing at least one coupler represented by formula (C-I) and at least one compound represented by formula (A-I) or (A-II) ##STR1## wherein Q.sub.1 represents an atomic group containing at least one nitrogen atom required to form a 5- or more membered nitrogen-containing heterocyclic ring together with the carbon atoms to which it is bonded; Z.sub.1 represents a hydrogen atom or a coupling-off group; R.sub.Cl represents an acyl or sulfonyl group; and R.sub.C2 represents a hydrogen atom or a C.sub.1-8 aliphatic group, or the substituents for R.sub.Cl, R.sub.C2, Z.sub.1, or Q.sub.1 form a dimeric or polymeric coupler; ##STR2## wherein R represents a hydrogen atom, an aliphatic group, an aromatic group, a heterocyclic group, or a hydrolyzable protective group; R.sub.1, R.sub.2, R.sub.3, R.sub.4, and R.sub.5 each represents a hydrogen atom or a substituent; R' represents a hydrogen atom, an aliphatic group, an acyl group, a sulfonyl group, a sulfinyl group, an oxyradical group or a hydroxyl group; A represents a non-metallic atomic group required to form a 5-, 6- or 7-membered ring; and R.sub.6, R.sub.7, R.sub.8, and R.sub.9 each represents a hydrogen atom or an alkyl group, or the substituents represented by R and R.sub.1 or two or R.sub.1, R.sub.2, R.sub.3, R.sub.4, and R.sub.5 in formula (A-I) which are in an ortho-position relation are bonded to each other to form a 5-, 6-, or 7-membered ring, or the substituents represented by R.sub.6 and R.sub.7, R.sub.8 and R.sub.9, or R' and R.sub.6 in formula (A-II) are bonded to each other to form a 5-, 6-, or 7-membered ring.

    摘要翻译： 提供了一种新颖的卤化银彩色照相材料，其含有至少一种由式（C1）表示的成色剂和至少一种由式（AI）或（A-II）表示的化合物（C1），其中Q1表示原子团 含有与其键合的碳原子一起形成5-或更多元含氮杂环所需的至少一个氮原子; Z1表示氢原子或偶联离子基团; RCl表示酰基或磺酰基; 和RC2表示氢原子或C1-8脂族基团，或者RCl，RC2，Z1或Q1的取代基形成二聚或聚合成色剂; （A-I）（A-II）其中R表示氢原子，脂族基团，芳族基团，杂环基或可水解保护基团; R1，R2，R3，R4和R5各自表示氢原子或取代基; R'表示氢原子，脂族基团，酰基，磺酰基，亚磺酰基，氧自由基或羟基; A表示形成5-，6-或7-元环所需的非金属原子团; 或者R 1，R 2，R 3，R 4和R 5分别表示氢原子或烷基，或者R 1和R 2所代表的取代基或式 或者由式（A-II）中的R 6和R 7，R 8和R 9或R'和R 6表示的取代基相互键合， 彼此形成5-，6-或7-元环。

    Photographic method using bleaching solution containing ferric complex salts and an aromatic compound
    9.
    发明授权
    Photographic method using bleaching solution containing ferric complex salts and an aromatic compound 失效
    使用含有铁络合物盐和芳族化合物的漂白溶液的照相方法

    公开(公告)号：US4894320A

    公开(公告)日：1990-01-16

    申请号：US101319

    申请日：1987-09-25

    申请人： Shinji Ueda ,  Masakazu Morigaki ,  Kozo Aoki

    发明人： Shinji Ueda ,  Masakazu Morigaki ,  Kozo Aoki

    IPC分类号： G03C7/42

    CPC分类号： G03C7/42

    摘要： A method of processing an imagewise exposed silver halide color photographic material comprising developing the material with a color developing solution, and then processing the material with a solution having a bleaching ability, wherein the processing solution having a bleaching ability contains a ferric complex salt comprising, as a complexing agent, an aromatic compound having at least one group represented by the following general formula (I): ##STR1## wherein X represents a hydrogen atom or an organic or inorganic cation, A represents a single bond or a divalent linking group, and R represents a hydrogen atom, an aliphatic group, an aromatic group, a heterocyclic ring group, an acyl group, a sulfonyl group, A or --CH.sub.2 PO.sub.3 X.sub.2.

    摘要翻译： 一种处理成像曝光的卤化银彩色照相材料的方法，包括用彩色显影液显影该材料，然后用具有漂白能力的溶液处理该材料，其中具有漂白能力的处理溶液含有三价络合盐， 作为络合剂，具有至少一个由以下通式（I）表示的基团的芳族化合物：其中X表示氢原子或有机或无机阳离子，A表示单键或二价 R表示氢原子，脂肪族基团，芳香族基团，杂环基团，酰基，磺酰基，A或-CH 2 PO 3 X 2。