-
1.发明授权公开(公告)号：US08835633B2
公开(公告)日：2014-09-16
申请号：US13427767
申请日：2012-03-22
申请人： Sergio Cesco-Cancian , Jeffrey S. Grimm , Neelakandha S. Mani , Christopher M. Mapes , David C. Palmer , Daniel J. Pippel , Tong Xiao , Diego Broggini , Susanne Lochner
发明人： Sergio Cesco-Cancian , Jeffrey S. Grimm , Neelakandha S. Mani , Christopher M. Mapes , David C. Palmer , Daniel J. Pippel , Tong Xiao , Diego Broggini , Susanne Lochner
IPC分类号： C07D401/14 , C07D403/04
CPC分类号： C07D403/04
摘要： The present invention is directed to benzoimidazol-2-yl pyrimidine derivatives useful as histamine H4 receptor modulators and processes for the preparation of such compounds.
摘要翻译： 本发明涉及可用作组胺H 4受体调节剂的苯并咪唑-2-基嘧啶衍生物及其制备方法。
-
2.发明授权Process for the preparation of piperazinyl and diazepanyl benzamide derivatives 有权制备哌嗪基和二氮杂环庚烷基苯甲酰胺衍生物的方法公开(公告)号：US08680273B2
公开(公告)日：2014-03-25
申请号：US12987370
申请日：2011-01-10
申请人： Anusuya Choudhury , Jeffrey S. Grimm , Kirk L. Sorgi , David Palmer , Jing Liu
发明人： Anusuya Choudhury , Jeffrey S. Grimm , Kirk L. Sorgi , David Palmer , Jing Liu
IPC分类号： C07D241/04
CPC分类号： C07D413/10 , C07D241/04 , C07D401/10 , C07D403/10 , Y02P20/55
摘要： The present invention is directed to a novel process for the preparation of piperazinyl and diazepanyl benzamide derivatives, useful for the treatment of disorders and conditions mediated by a histamine receptor, preferably the H3 receptor.
摘要翻译： 本发明涉及用于制备哌嗪基和二氮杂环庚烷基苯甲酰胺衍生物的新方法，其可用于治疗由组胺受体介导的病症和病症，优选H3受体。
-
3.发明申请公开(公告)号：US20120184740A1
公开(公告)日：2012-07-19
申请号：US13427798
申请日：2012-03-22
申请人： Sergio Cesco-Cancian , Jeffrey S. Grimm , Neelakandha S. Mani , Christopher M. Mapes , David C. Palmer , Daniel J. Pippel , Tong Xiao , Diego Broggini , Susanne Lochner
发明人： Sergio Cesco-Cancian , Jeffrey S. Grimm , Neelakandha S. Mani , Christopher M. Mapes , David C. Palmer , Daniel J. Pippel , Tong Xiao , Diego Broggini , Susanne Lochner
IPC分类号： C07D401/14
CPC分类号： C07D403/04
摘要： The present invention is directed to benzoimidazol-2-yl pyrimidine derivatives useful as histamine H4 receptor modulators and processes for the preparation of such compounds.
摘要翻译： 本发明涉及可用作组胺H 4受体调节剂的苯并咪唑-2-基嘧啶衍生物及其制备方法。
-
4.发明申请PROCESS FOR THE PREPARATION OF PIPERAZINYL AND DIAZEPANYL BENZAMIDE DERIVATIVES 有权制备哌嗪和二氮茚衍生物衍生物的方法公开(公告)号：US20110105752A1
公开(公告)日：2011-05-05
申请号：US12987370
申请日：2011-01-10
申请人： Anusuya Choudhury , Jeffrey S. Grimm , Kirk L. Sorgi , David Palmer , Jing Liu
发明人： Anusuya Choudhury , Jeffrey S. Grimm , Kirk L. Sorgi , David Palmer , Jing Liu
IPC分类号： C07D241/04
CPC分类号： C07D413/10 , C07D241/04 , C07D401/10 , C07D403/10 , Y02P20/55
摘要： The present invention is directed to a novel process for the preparation of piperazinyl and diazepanyl benzamide derivatives, useful for the treatment of disorders and conditions mediated by a histamine receptor, preferably the H3 receptor.
摘要翻译： 本发明涉及用于制备哌嗪基和二氮杂环庚烷基苯甲酰胺衍生物的新方法，其可用于治疗由组胺受体介导的病症和病症，优选H3受体。
-
公开(公告)号：US08309720B2
公开(公告)日：2012-11-13
申请号：US12459229
申请日：2009-06-29
申请人： Sergio Cesco-Cancian , Hongfeng Chen , Jeffrey S. Grimm , Neelakandha S. Mani , Christopher M. Mapes , David C. Palmer , Daniel J. Pippel , Kirk L. Sorgi , Tong Xiao
发明人： Sergio Cesco-Cancian , Hongfeng Chen , Jeffrey S. Grimm , Neelakandha S. Mani , Christopher M. Mapes , David C. Palmer , Daniel J. Pippel , Kirk L. Sorgi , Tong Xiao
IPC分类号： C07D211/06 , C07D211/30
CPC分类号： C07D401/12 , C07C211/22 , C07C211/26 , C07D211/22 , C07D211/26
摘要： The present invention is directed to processes for the preparation of substituted pyrimidine derivatives, useful as intermediates in the synthesis of histamine H4 receptor modulators, and to intermediates in H4 modulator synthesis.
摘要翻译： 本发明涉及制备用作合成组胺H 4受体调节剂的中间体的取代嘧啶衍生物的方法，以及H4调节剂合成中的中间体。
-
6.发明申请公开(公告)号：US20120178932A1
公开(公告)日：2012-07-12
申请号：US13427767
申请日：2012-03-22
申请人： Sergio CESCO-CANCIAN , Jeffrey S. GRIMM , Neelakandha S. MANI , Christopher M. MAPES , David C. PALMER , Daniel J. PIPPEL , Tong XIAO , Diego BROGGINI , Susanne LOCHNER
发明人： Sergio CESCO-CANCIAN , Jeffrey S. GRIMM , Neelakandha S. MANI , Christopher M. MAPES , David C. PALMER , Daniel J. PIPPEL , Tong XIAO , Diego BROGGINI , Susanne LOCHNER
IPC分类号： C07D401/14
CPC分类号： C07D403/04
摘要： The present invention is directed to benzoimidazol-2-yl pyrimidine derivatives useful as histamine H4 receptor modulators and processes for the preparation of such compounds.
摘要翻译： 本发明涉及可用作组胺H 4受体调节剂的苯并咪唑-2-基嘧啶衍生物及其制备方法。
-
7.发明申请PROCESS FOR THE PREPARATION OF PIPERAZINYL AND DIAZEPANYL BENZAMIDE DERIVATIVES 有权制备哌嗪和二氮茚衍生物衍生物的方法公开(公告)号：US20080171870A1
公开(公告)日：2008-07-17
申请号：US11953262
申请日：2007-12-10
申请人： Anusuya Choudhury , Jeffrey S. Grimm , Kirk L. Sorgi , David Palmer , Jing Liu
发明人： Anusuya Choudhury , Jeffrey S. Grimm , Kirk L. Sorgi , David Palmer , Jing Liu
IPC分类号： C07D413/00 , C07D295/00
CPC分类号： C07D413/10 , C07D241/04 , C07D401/10 , C07D403/10 , Y02P20/55
摘要： The present invention is directed to a novel process for the preparation of piperazinyl and diazepanyl benzamide derivatives, useful for the treatment of disorders and conditions mediated by a histamine receptor, preferably the H3 receptor.
摘要翻译： 本发明涉及用于制备哌嗪基和二氮杂环庚烷基苯甲酰胺衍生物的新方法，其可用于治疗由组胺受体介导的病症和病症，优选H3受体。
-
8.发明申请One-Pot Condensation-Reduction Methods for Preparing Substituted Allylic Alcohols 审中-公开用于制备取代的烯丙醇的一锅冷凝还原方法公开(公告)号：US20080009628A1
公开(公告)日：2008-01-10
申请号：US11762371
申请日：2007-06-13
申请人： Michael Reuman , Roger Faessler , Armin Roessler , Kirk Sorgi , Xun Li , Jeffrey S. Grimm
发明人： Michael Reuman , Roger Faessler , Armin Roessler , Kirk Sorgi , Xun Li , Jeffrey S. Grimm
IPC分类号： C07D401/02 , C07D209/48 , C07D211/06 , C07D211/96
CPC分类号： C07D209/48 , C07D401/04 , C07D401/06 , C07D401/14
摘要： One-pot condensation-reduction methods for preparing substituted allylic alcohols as well as highly selective extractive methods to separate isomeric alcohols produced in the one-pot condensation-reduction processes are provided for preparing, for example, a quinolone.
摘要翻译： 提供用于制备取代的烯丙醇的一锅缩合还原方法以及用于分离在一锅缩合还原方法中产生的异构醇的高选择性萃取方法用于制备例如喹诺酮。
-
9.发明授权Process for the preparation of piperazinyl and diazepanyl benzamide derivatives 有权制备哌嗪基和二氮杂环庚烷基苯甲酰胺衍生物的方法公开(公告)号：US07893257B2
公开(公告)日：2011-02-22
申请号：US11953262
申请日：2007-12-10
申请人： Anusuya Choudhury , Jeffrey S. Grimm , Kirk L. Sorgi , David Palmer , Jing Liu
发明人： Anusuya Choudhury , Jeffrey S. Grimm , Kirk L. Sorgi , David Palmer , Jing Liu
IPC分类号： C07D413/10
CPC分类号： C07D413/10 , C07D241/04 , C07D401/10 , C07D403/10 , Y02P20/55
摘要： The present invention is directed to a novel process for the preparation of piperazinyl and diazepanyl benzamide derivatives, useful for the treatment of disorders and conditions mediated by a histamine receptor, preferably the H3 receptor.
摘要翻译： 本发明涉及用于制备哌嗪基和二氮杂环庚烷基苯甲酰胺衍生物的新方法，其可用于治疗由组胺受体介导的病症和病症，优选H3受体。
-
10.发明申请公开(公告)号：US20100029942A1
公开(公告)日：2010-02-04
申请号：US12459224
申请日：2009-06-29
申请人： Sergio Cesco-Cancian , Jeffrey S. Grimm , Neelakandha S. Mani , Christopher M. Mapes , David C. Palmer , Daniel J. Pippel , Tong Xiao , Diego Broggini , Susanne Lochner
发明人： Sergio Cesco-Cancian , Jeffrey S. Grimm , Neelakandha S. Mani , Christopher M. Mapes , David C. Palmer , Daniel J. Pippel , Tong Xiao , Diego Broggini , Susanne Lochner
IPC分类号： C07D401/14
CPC分类号： C07D403/04
摘要： The present invention is directed to benzoimidazol-2-yl pyrimidine derivatives useful as histamine H4 receptor modulators and processes for the preparation of such compounds.
摘要翻译： 本发明涉及可用作组胺H 4受体调节剂的苯并咪唑-2-基嘧啶衍生物及其制备方法。
-
-
-
-
-
-
-
-
-
搜索结果
11 条记录 (耗时 0.023 秒)
