公开(公告)号：US20110282070A1

公开(公告)日：2011-11-17

申请号：US13188402

申请日：2011-07-21

申请人： Hiroshi SHIMOHARADA ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

发明人： Hiroshi SHIMOHARADA ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

IPC分类号： C07D413/10 ,  C07C317/46 ,  C07C51/60 ,  C07D231/20 ,  C07D405/10

CPC分类号： C07D231/20 ,  C07D405/12 ,  C07D413/12

摘要： A benzoylpyrazole compound represented by the formula (I) or its salt: wherein R1 is alkyl or cycloalkyl, R2 is a hydrogen atom or alkyl, R3 is alkyl; cycloalkyl; haloalkyl; alkoxyalkyl; alkoxycarbonylalkyl; alkenyl; or arylalkyl which may be substituted by R8, R4 is alkyl; haloalkyl; alkoxy; halogen; nitro; cyano; alkylthio; alkylsulfinyl; or alkylsulfonyl, R5 is a hydrogen atom; alkyl; alkenyl; alkynyl; halogen; cyano; cyanoalkyl; cyanoalkeny; haloalkyl; alkoxyalkyl; haloalkoxyalkyl; amino(thiocarbonyl)alkyl which may be substituted by at least one substituent selected from alkyl, cyano, is cyanoalkyl, (alkylthio)carbonylalkyl, alkyl(thiocarbonyl)alkyl, —C(O)OR7 and —C(O)SR7; thiocyanatoalkyl; alkoxy; alkenyloxy; alkynyloxy; haloalkoxy; alkoxyalkoxy; haloalkoxyalkoxy; alkoxyhaloalkoxy; haloalkoxyhaloalkoxy; alkoxyalkoxyalkyl; alkylthio; alkoxyalkylthio; haloalkoxyalkylthio; alkoxyhaloalkylthio; haloalkoxyhaloalkylthio; alkylthioalkylthio; haloalkylthioalkylthio; alkylthiohaloalkylthio; haloalkylthiohaloalkylthio; alkylthioalkoxy; alkylsulfonyl; alkylsulfonylalkyl; alkoxycarbonylalkyl; alkoxycarbonylalkoxy; heterocyclylalkyl; heterocyclyloxy; heterocyclylalkoxy; heterocyclylalkoxyalkyl; heterocyclyloxyalkyl; cycloalkyloxy; —OC(O)SR7; —OC(O)OR7; —C(O)OR7; —C(O)SR7; —C(S)OR7; —C(S)SR7; aminoalkyl which may be substituted by at least one substituent selected from alkyl, cyano, cyanoalkyl, (alkylthio)carbonylalkyl, alkyl(thiocarbonyl)alkyl, —C(O)OR7 and —C(O)SR7; or 4,5-dihydroisoxazol-3-yl which may be substituted by R9, R6 is haloalkyl; halogen; nitro; cyano; alkylthio; alkylsulfinyl; or alkylsulfonyl, R7 is alkyl; haloalkyl; alkoxyalkyl; alkenyl; haloalkenyl; alkynyl; or arylalkyl which may be substituted by R10, and each of R8, R9 and R10 which are independent of one another, is halogen; alkyl; or alkoxy.

公开(公告)号：US20100317528A1

公开(公告)日：2010-12-16

申请号：US12521649

申请日：2007-12-27

申请人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Souichiro Nagayama ,  Makiko Sano ,  Yoshinori Kitahara ,  Tatsuya Okita ,  Hiroshi Hata

发明人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Souichiro Nagayama ,  Makiko Sano ,  Yoshinori Kitahara ,  Tatsuya Okita ,  Hiroshi Hata

IPC分类号： A01N43/56 ,  C07D231/20 ,  A01P13/00

CPC分类号： A01N43/56 ,  C07C317/22 ,  C07D231/20 ,  C07D405/10 ,  C07D413/10

摘要： To provide a novel herbicide which has a wide range of applications to agricultural or non-agricultural fields and various methods for application such as soil treatment and foliage treatment and which exhibits excellent herbicidal effects.A herbicide containing a benzoylpyrazole compound represented by the formula (I) or its salt, as an active ingredient: wherein R1 is alkyl or cycloalkyl, R2 is a hydrogen atom or alkyl, R3 is hydroxy, R4 is alkyl, haloalkyl or the like, R5 is halogen, cyano, cyanoalkyl or the like, and R6 is haloalkyl, halogen or the like.

摘要翻译： 提供一种广泛应用于农业或非农业领域的新型除草剂和各种施用方法如土壤处理和叶面处理，并且具有优异的除草效果。 一种除草剂，其含有式（I）表示的苯甲酰基吡唑化合物或其盐作为活性成分：其中R1是烷基或环烷基，R2是氢原子或烷基，R3是羟基，R4是烷基，卤代烷基等， R5是卤素，氰基，氰基烷基等，R6是卤代烷基，卤素等。

公开(公告)号：US20050245399A1

公开(公告)日：2005-11-03

申请号：US10834028

申请日：2004-04-29

申请人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Hiroshi Kikugawa ,  Yoshinori Kitahara

发明人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Hiroshi Kikugawa ,  Yoshinori Kitahara

IPC分类号： A01N43/40 ,  A01N43/56 ,  A01N47/20 ,  A01N47/22 ,  A01N47/30 ,  C07D231/20 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12

CPC分类号： A01N47/30 ,  A01N43/56 ,  A01N47/20 ,  A01N47/22 ,  C07D231/20 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12

摘要： The present invention relates to novel pyrazole derivatives of the formula (I) or its salt: wherein X, Y, R1, R2, R3, R4 and R5 each have one of the meanings given in the description, a process for producing them, and their use as herbicides, desiccants or defoliants.

摘要翻译： 本发明涉及式（I）的新型吡唑衍生物或其盐：其中X，Y，R 1，R 2，R 3， R 4，R 4和R 5各自具有说明书中给出的含义之一，其制备方法及其作为除草剂，干燥剂或脱叶剂的用途。

公开(公告)号：US08030498B2

公开(公告)日：2011-10-04

申请号：US12094734

申请日：2006-12-13

申请人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

发明人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

IPC分类号： C07D231/20 ,  A61K31/415

CPC分类号： C07D231/20 ,  C07D405/12 ,  C07D413/12

摘要： A benzoylpyrazole compound represented by the formula (I) or its salt, useful as herbicides and intermediates thereof.

摘要翻译： 由式（I）表示的苯甲酰基吡唑化合物或其盐，可用作除草剂及其中间体。

公开(公告)号：US20090286683A1

公开(公告)日：2009-11-19

申请号：US12094734

申请日：2006-12-13

申请人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

发明人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

IPC分类号： A01N43/56 ,  C07D231/18 ,  C07D405/10 ,  A01P13/00

CPC分类号： C07D231/20 ,  C07D405/12 ,  C07D413/12

摘要： A benzoylpyrazole compound represented by the formula (I) or its salt, useful as herbicides and intermediates thereof.

摘要翻译： 由式（I）表示的苯甲酰基吡唑化合物或其盐，可用作除草剂及其中间体。

公开(公告)号：US4790869A

公开(公告)日：1988-12-13

申请号：US9924

申请日：1987-02-02

申请人： Fumio Kimura ,  Takahiro Haga ,  Kazuyuki Maeda ,  Hiroshi Shimoharada ,  Tsunezo Yoshida ,  Masahiko Ikeguchi

发明人： Fumio Kimura ,  Takahiro Haga ,  Kazuyuki Maeda ,  Hiroshi Shimoharada ,  Tsunezo Yoshida ,  Masahiko Ikeguchi

IPC分类号： A01N47/36 ,  C07D275/02 ,  C07D275/03 ,  C07D521/00 ,  A01N43/54 ,  C07D239/47 ,  C07D417/12

CPC分类号： C07D275/03 ,  A01N47/36 ,  C07D521/00

摘要： A sulfonamide compound and a salt thereof is represented by the following general formula: ##STR1## wherein each of X.sub.1, X.sub.2, and X.sub.3 independently represents a hydrogen atom or a halogen atom, each of Y.sub.1, Y.sub.2, and Y.sub.3 independently represents a halogen atom, and R represents a methyl group or a methoxy group, and is effective as an active ingredient of a herbicidal composition.

摘要翻译： 磺酰胺化合物及其盐由以下通式表示：其中X1，X2和X3各自独立地表示氢原子或卤素原子，Y1，Y2和Y3各自独立地表示卤素原子 R表示甲基或甲氧基，作为除草组合物的有效成分是有效的。

公开(公告)号：US08466088B2

公开(公告)日：2013-06-18

申请号：US12525554

申请日：2008-02-01

申请人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Souichiro Nagayama ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

发明人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Souichiro Nagayama ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

IPC分类号： A01N63/00

CPC分类号： A01N43/56 ,  A01N33/18 ,  A01N37/20 ,  A01N37/22 ,  A01N37/36 ,  A01N37/40 ,  A01N39/04 ,  A01N41/10 ,  A01N43/10 ,  A01N43/40 ,  A01N43/653 ,  A01N43/70 ,  A01N43/707 ,  A01N43/80 ,  A01N43/82 ,  A01N43/88 ,  A01N47/06 ,  A01N47/30 ,  A01N47/36 ,  A01N57/20 ,  A01N2300/00

摘要： Provided is an herbicidal composition which can be applied at a low dose as compared with individual application, and thus is effective to reduce the environmental load on a place where the composition is applied or a periphery thereof, of which the herbicidal spectrum is enlarged, and of which the herbicidal effects last over a long period of time. The herbicidal composition has as active ingredients (a) a herbicidal benzoylpyrazole compound represented by the formula (I) or its salt: wherein Q is —C(O)SR3 or a hydrogen atom, R1 is alkyl or cycloalkyl, R2 is a hydrogen atom or alkyl, R3 is alkyl, cycloalkyl or the like, R4 is alkyl, haloalkyl or the like, R5 is a hydrogen atom, alkyl or the like, R6 is haloalkyl, halogen or the like, and (b) a further herbicidal compound.

摘要翻译： 本发明提供了与单独使用相比可以以低剂量施用的除草组合物，因此有效地降低施用组合物的地方或其周边，增加除草频谱的环境负荷，以及 其除草效果持续很长时间。 除草组合物具有（a）式（I）表示的除草酰苯并吡唑化合物或其盐：其中Q为-C（O）SR 3或氢原子，R 1为烷基或环烷基，R 2为氢原子 或烷基，R 3是烷基，环烷基等，R 4是烷基，卤代烷基等，R 5是氢原子，烷基等，R 6是卤代烷基，卤素等，和（b）另外的除草化合物。

公开(公告)号：US20100099563A1

公开(公告)日：2010-04-22

申请号：US12525554

申请日：2008-02-01

申请人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Souichiro Nagayama ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

发明人： Hiroshi Shimoharada ,  Masamitsu Tsukamoto ,  Masahiko Ikeguchi ,  Hiroshi Kikugawa ,  Souichiro Nagayama ,  Makiko Sano ,  Yoshinori Kitahara ,  Hidemasa Kominami ,  Tatsuya Okita

IPC分类号： A01N43/56 ,  A01N43/66 ,  A01N43/40

CPC分类号： A01N43/56 ,  A01N33/18 ,  A01N37/20 ,  A01N37/22 ,  A01N37/36 ,  A01N37/40 ,  A01N39/04 ,  A01N41/10 ,  A01N43/10 ,  A01N43/40 ,  A01N43/653 ,  A01N43/70 ,  A01N43/707 ,  A01N43/80 ,  A01N43/82 ,  A01N43/88 ,  A01N47/06 ,  A01N47/30 ,  A01N47/36 ,  A01N57/20 ,  A01N2300/00

摘要： To provide a herbicidal composition which can be applied at a low dose as compared with individual application, and thus is effective to reduce the environmental load on a place where the composition is applied or a periphery thereof, of which the herbicidal spectrum is enlarged, and of which the herbicidal effects last over a long period of time.A herbicidal composition which comprises as active ingredients (a) a herbicidal benzoylpyrazole compound represented by the formula (I) or its salt: wherein Q is —C(O)SR3 or a hydrogen atom, R1 is alkyl or cycloalkyl, R2 is a hydrogen atom or alkyl, R3 is alkyl, cycloalkyl or the like, R4 is alkyl, haloalkyl or the like, R5 is a hydrogen atom, alkyl or the like, R6 is haloalkyl, halogen or the like, and (b) other herbicidal compound.

摘要翻译： 提供与单独施用相比可以以低剂量施用的除草组合物，因此有效地减少施用组合物的地方或其周边，其除草频谱扩大的环境负荷，以及 其除草效果持续很长时间。 一种除草组合物，其包含作为活性成分的（a）由式（I）表示的除草酰苯并吡唑化合物或其盐：其中Q为-C（O）SR 3或氢原子，R 1为烷基或环烷基，R 2为氢 原子或烷基，R3是烷基，环烷基等，R4是烷基，卤代烷基等，R5是氢原子，烷基等，R6是卤代烷基，卤素等，和（b）其它除草化合物。

公开(公告)号：US06479435B1

公开(公告)日：2002-11-12

申请号：US09779674

申请日：2001-02-09

申请人： David A. Pulman ,  Bai-Ping Ying ,  Shao-Yong Wu ,  Sandeep Gupta ,  Hiroshi Shimoharada ,  Masamitsu Tsukamoto

发明人： David A. Pulman ,  Bai-Ping Ying ,  Shao-Yong Wu ,  Sandeep Gupta ,  Hiroshi Shimoharada ,  Masamitsu Tsukamoto

IPC分类号： C07D40312

CPC分类号： C07D401/12 ,  A01N31/14 ,  A01N33/22 ,  A01N37/48 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/66 ,  A01N43/713 ,  A01N43/80 ,  A01N43/90 ,  A01N47/06 ,  C07D403/12 ,  C07D471/04 ,  C07D487/04 ,  C07D513/04

摘要： Diaryl ether compounds useful in the control of weeds are described. An exemplary compound is represented by the general formula (I): In this formula Q is represented by Q1 X and Y represent a hydrogen atom, halogen atom, cyano group, nitro group or (C1-6)haloalkyl group; R1 is halogen; R2 and R3 represent a hydrogen atom, a (C1-6)alkyl group or a (C1-6)haloalkyl group . Methods of making the compounds are also described.

摘要翻译： 描述了可用于控制杂草的二芳基醚化合物。 示例性化合物由通式（I）表示：在该式中Q由Q1X表示，Y表示氢原子，卤素原子，氰基，硝基或（C1-6）卤代烷基; R1是卤素; R2和R3表示氢原子，（C1-6）烷基或（C1-6）卤代烷基。 还描述了制备化合物的方法。

公开(公告)号：US06333296B1

公开(公告)日：2001-12-25

申请号：US09380830

申请日：1999-09-10

申请人： David A. Pulman ,  Bai-Ping Ying ,  Shao-Yong Wu ,  Sandeep Gupta ,  Hiroshi Shimoharada ,  Masamitsu Tsukamoto

发明人： David A. Pulman ,  Bai-Ping Ying ,  Shao-Yong Wu ,  Sandeep Gupta ,  Hiroshi Shimoharada ,  Masamitsu Tsukamoto

IPC分类号： C07D23946

CPC分类号： C07D401/12 ,  A01N31/14 ,  A01N33/22 ,  A01N37/48 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/66 ,  A01N43/713 ,  A01N43/80 ,  A01N43/90 ,  A01N47/06 ,  C07D403/12 ,  C07D471/04 ,  C07D487/04 ,  C07D513/04

摘要： Diaryl ether compounds useful in the control of weeds are described. An exemplary compound is represented by the general formula (I): In this formula Q is represented by Q9: X and Y represent a hydrogen atom, halogen atom, cyano group, nitro group or (C1-6)haloalkyl group. A1 and A2 are independently oxygen or sulfur atoms. R9 and R10 represent a hydrogen atom, a (C1-6)alkyl group, an acyl group, or a (C1-6)alkylsulfonyl group; or R9 and R10 may form a ring consisting of polymethylene, (CH2)m groups, where m is an integer of 2, 3, 4 or 5, together with the nitrogen atom of NR9R10, which may or may not have a (C1-6)alkyl substituent. Methods of making the compounds are also described.

摘要翻译： 描述了可用于控制杂草的二芳基醚化合物。 示例性化合物由通式（I）表示：在该式中Q由Q 9表示：X，Y表示氢原子，卤素原子，氰基，硝基或（C 1-6）卤代烷基。 A1和A2独立地是氧或硫原子。 R9和R10表示氢原子，（C1-6）烷基，酰基或（C1-6）烷基磺酰基; 或R 9和R 10可以形成由多亚甲基，（CH 2）m基团组成的环，其中m是2,3,4或5的整数，以及NR 9 R 10的氮原子，其可以具有或不具有（C1- 6）烷基取代基。 还描述了制备化合物的方法。