Triazine derivatives, their production and use
    1.
    发明授权
    Triazine derivatives, their production and use 失效
    三嗪衍生物,其生产和使用

    公开(公告)号:US06294536B1

    公开(公告)日:2001-09-25

    申请号:US09445159

    申请日:2000-03-01

    IPC分类号: A61K3153

    摘要: The present invention relates to compounds represented by the formula: wherein ring H represents an optionally substituted aromatic heterocyclic group or an optionally substituted alicyclic hydrocarbon group; X and Y independently represent a single bond, —O—, a group of the formula: —S(O)m— wherein m is 0, 1 or 2, a group of the formula: —NR8— wherein R8 represents a hydrogen atom, an alkyl group or an acyl group, —CO— or an optionally substituted methylene group; —A—B— represents —N═CH—, —CH═N—, —N═N— or —CH═CH—; R1 represents a hydrogen atom, a halogen atom, an optionally substituted alkyl group which may be bonded through a hetero atom or an acyl group; R2 and R3 independently represent a hydrogen atom, a halogen atom or an optionally substituted alkyl group; R4 represents a hydrogen atom or a halogen atom; R5 represents a hydrogen atom, an optionally substituted alkyl group or an acyl group; R6 and R7 independently represent a hydrogen atom or R6 and R7 may form a chemical bond together with each other; and D represents —CH2— or —CO—; or a salt thereof. These compounds and salts thereof are useful as anti-protozoal agents.

    摘要翻译: 本发明涉及由下式表示的化合物:其中环H表示任选取代的芳族杂环基或任选取代的脂环族烃基; X和Y独立地表示单键,-O-,下式-S(O)m - 的基团,其中m为0,1或2,式-NR8-的基团,其中R8表示氢原子 ,烷基或酰基,-CO-或任选取代的亚甲基; -A-B-表示-N = CH-,-CH = N-,-N = N-或-CH = CH-; R1表示氢原子,卤素原子,可以通过杂原子或酰基键合的任意取代的烷基; R2和R3独立地表示氢原子,卤素原子或任选取代的烷基; R4表示氢原子或卤素原子; R5代表氢原子,任选取代的烷基或酰基; R6和R7独立地表示氢原子或R6,R7可以彼此形成化学键; 和D表示-CH 2 - 或-CO-; 或其盐。 这些化合物及其盐可用作抗原生动物剂。

    Thioether derivatives, their method for production and use
    4.
    发明授权
    Thioether derivatives, their method for production and use 有权
    硫醚衍生物,其生产和使用方法

    公开(公告)号:US06630578B2

    公开(公告)日:2003-10-07

    申请号:US09988774

    申请日:2001-11-20

    IPC分类号: C07C24500

    摘要: Novel dendritic molecules are provided which respond immediately by emission of light when stimulated with light or electric energy, and are useful, for example, as switching material of memory. The dendritic molecules have a core, a branch structure composed of Unit 1 represented by the following formula: wherein, ring A stands for a homo or heterocyclic six membered ring, optionally other branched structures, and surface functional groups as essential constituents.

    摘要翻译: 提供了当用光或电能刺激时,通过发出光而立即响应的新型树枝状分子,并且例如用作存储器的切换材料是有用的。 树枝状分子具有核心,由下式表示的单元1构成的支链结构:其中环A代表同价或杂环六元环,任选其它支链结构和表面官能团作为必要成分。

    Process of producing sulfonylurea derivatives
    6.
    发明授权
    Process of producing sulfonylurea derivatives 失效
    磺酰脲衍生物的制备方法

    公开(公告)号:US4994571A

    公开(公告)日:1991-02-19

    申请号:US237231

    申请日:1988-08-26

    IPC分类号: A01N47/36 C07D521/00

    CPC分类号: C07D521/00 A01N47/36

    摘要: This invention relates to a process for producing a compound of the formula (I) as shown below. ##STR1## wherein Q is a condensed heterocyclic group having a nitrogen atom in the bridgehead position which may optionally be substituted, R.sub.1 and R.sub.2 each are an alkyl group, an alkoxy group or halogen and Z is CH or N, or a salt thereof.The compound (I) or a salt thereof is novel and of value as agricultural chemicals.According to the process of this invention the compound (I) or a salt thereof can be produced in good yield and high purity.

    Molecular bonding method and molecular bonding device
    8.
    发明申请
    Molecular bonding method and molecular bonding device 审中-公开
    分子键合方法和分子键合装置

    公开(公告)号:US20070172600A1

    公开(公告)日:2007-07-26

    申请号:US10554059

    申请日:2004-04-23

    摘要: External energy is fed to N-[3-{3,5-bis{3,5-bis[3,5-bis(4-mercaptobenzylthio)benzylthio]benzylthio}benzyloxy}-propionyl-4-nitro-1-naphthylamine (18a) being a molecule capable of photosensitization as an intermediate excitation medium, fixed on support (12) of a metal, so as to photosensitized molecule of excited triplet state (18b), thereby inducing an excited triplet energy transfer from this photosensitized molecule to first molecule (28a) having a residue capable of bonding. The first molecule (28b) having thus been excited by the excited triplet energy transfer is bonded with second molecule (30) having a residue capable of bonding which is a bonding object to be bonded with the first molecule.

    摘要翻译: 将外部能量加入到N- [3- {3,5-双{3,5-双[3,5-二(4-巯基苄硫基)苄硫基]苄硫基}苄氧基} - 丙酰基-4-硝基-1-萘胺( 18 a)作为中和激发介质的能够光敏化的分子,固定在金属的载体(12)上,以便激发三重态的光敏化分子(18b),从而诱导来自该光敏化分子的激发的三线态能量转移 涉及具有能够键合的残基的第一分子(28a)。 由激发的三线态能量转移激发的第一分子(28b)与具有能够键合的残基的第二分子(30)结合,该第二分子(30)是与第一分子键合的结合对象。

    Probe
    9.
    发明申请
    Probe 审中-公开
    探测

    公开(公告)号:US20070114400A1

    公开(公告)日:2007-05-24

    申请号:US10554203

    申请日:2004-04-23

    IPC分类号: G21K7/00

    CPC分类号: G01Q70/18

    摘要: Abstract: A probe comprising support (12) of a gold wire and, fixed thereon, intermediate excited medium (18a) having been excited to an excited triplet state by supply of external energy thereto, wherein transfer of excited triplet energy is effected from the intermediate excited medium toward a first molecule having a residue with bonding capability. The first molecule having thus been excited by the transfer of excited triplet energy is bonded with a second molecule having a residue with bonding capability as a bonding target to be bonded with the first molecule.

    摘要翻译: 摘要:一种探针,其包括金线的支撑体(12),并且固定在其上,通过向其施加外部能量而被激发到激发三重态的中间激发介质(18a),其中激发的三线态能量的转移从 中等激发介质朝着具有结合能力的残基的第一分子。 通过激发的三线态能量的转移而激发的第一分子与具有键合能力的残基的第二分子键合作为与第一分子结合的键合靶。

    Triazine derivative, production and use thereof
    10.
    发明授权
    Triazine derivative, production and use thereof 失效
    三嗪衍生物,其生产和使用

    公开(公告)号:US06211178B1

    公开(公告)日:2001-04-03

    申请号:US09335918

    申请日:1999-06-18

    IPC分类号: A61K3153

    摘要: The present invention provides a novel triazine derivative of the formula wherein ring A is an optionally substituted aromatic group which be; X is an oxygen or sulfur atom; R1 and R6 are each a hydrogen atom or an optionally substituted hydrocarbon residue or heterocyclic group which may bound through a hetero-atom; R2 and R3 are each independently a hydrogen atom, a halogen atom, or a group bound through a carbon, oxygen or sulfur atom, or taken together, represent ═S; R4 and R5 are each independently a hydrogen atom, a halogen atom, or a group bound through a carbon, oxygen, nitrogen or sulfur atom; R1 and R2, and R5 and R6, may each bind together to form a chemical bond; provided that where ring A is a phenyl group having at least a halogen atom in position-2 or 4 and X is an oxygen atom, R4 and R5 do not conjoinedly represent a chemical bond and an antiprotozoan composition containing the same or salt thereof.

    摘要翻译: 本发明提供了一种新的三氟乙烯衍生物,其中A为任选取代的芳基,X为氧或硫原子; R 1和R 6各自为氢原子或任选取代的烃残基或可结合的杂环基 通过杂原子; R 2和R 3各自独立地为氢原子,卤素原子或通过碳,氧或硫原子结合的基团,或一起表示= S; R 4和R 5各自独立地为氢原子 卤素原子或通过碳,氧,氮或硫原子结合的基团; R 1和R 2以及R 5和R 6可以各自键合在一起形成化学键; 条件是当环A为至少具有2或4位的卤素原子且X为氧原子的苯基时,R 4和R 5不连结地表示化学键,而含有该化合键的抗原生动物组合物或其盐。