公开(公告)号：US20070135453A1

公开(公告)日：2007-06-14

申请号：US10579395

申请日：2004-12-14

Applicant: Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

Inventor： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC: A01N43/90 ,  C07D487/04

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: The present invention relates to 6-(2,4,6-trihalophenyl)triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-member saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R1 and/or R2 may be substituted as defined in the description; L1, L2, L3 are chlorine or fluorine, where at least one group is chlorine; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

Abstract translation: 本发明涉及式I的6-（2,4,6-三卤代苯基）三唑并嘧啶，其中取代基如下：R 1是烷基，卤代烷基，环烷基，卤代环烷基，烯基， 卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或五或六元饱和的部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 2 R 1是氢或R 1，R 2和R 2中所提及的基团之一，与它们的氮原子一起 还可以形成通过N连接的五元或六元杂环基或杂芳基，并且可以含有一个至三个其它由O，N和S组成的组的杂原子作为环成员; R 1和/或R 2可以如说明书中所定义的取代; L 1，L 2，L 3 3是氯或氟，其中至少一个基团是氯; X是氰基，烷基，烷氧基，烯氧基，卤代烷氧基或卤代烯氧基; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20060241128A1

公开(公告)日：2006-10-26

申请号：US10532719

申请日：2003-11-04

Applicant: Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

Inventor： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC: A01N43/90 ,  C07D487/04

CPC classification number: C07C69/65 ,  A01N43/90 ,  C07D487/04

Abstract: Substituted 6-(2-halogenphenyl)-triazolopyrimidines of formula I in which R1 denote alkyl, alkenyl, alkynyl, alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or a 5- or 6-membered saturated, unsaturated, or aromatic heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, wherein R1 and R2 radicals may be substituted as defined in the description, R2 denote hydrogen, or a group mentioned for R1; or R1 and R2 together with the interjacent nitrogen atom represent a 5- or 6-membered heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which ring may be substituted as defined in the description; Hal is halogen; L1, L3 independently denote hydrogen, halogen, or alkyl; L2 is hydrogen, halogen, haloalkyl, or NH2, NHRb, or N(Rb)2, wherein Rb is as defined in the description, wherein at least one from L1, L2, and L3 is not hydrogen; X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy. processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

Abstract translation: 其中R 1表示烷基，烯基，炔基，链二烯基，卤代烷基，卤代烯基，环烷基，苯基，萘基或5-或6-元的取代的6-（2-卤代苯基） - 三唑并嘧啶， 含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的饱和，不饱和或芳族杂环，其中R 1和R 2可以是 如说明书中所定义，R 2表示氢或R 1所提及的基团; 或R 1和R 2连同中间的氮原子代表含有1-4个氮原子或一至三个氮原子的一个或多个六元杂环，一个 硫或氧原子，该环可以如说明书中所定义取代; 卤素是卤素; L 1，L 3独立地表示氢，卤素或烷基; L 2是氢，卤素，卤代烷基或NH 2，NHR b或/或N（R b） 其中R b如描述中所定义，其中至少一个L 1，L 2， ，而L 3不是氢; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基。 其制备方法，含有它们的组合物及其用于对抗植物病原真菌的用途。

公开(公告)号：US20060102600A1

公开(公告)日：2006-05-18

申请号：US11281265

申请日：2005-11-17

Applicant: Peter Schafer ,  Frank Faisst ,  Martin Huonker ,  Richard Petersen

Inventor： Peter Schafer ,  Frank Faisst ,  Martin Huonker ,  Richard Petersen

IPC: B23K26/20 ,  B23K26/14

CPC classification number: B23K26/0648 ,  B23K26/123 ,  B23K26/142 ,  B23K26/1436 ,  B23K26/1437 ,  B23K26/1464 ,  B23K26/16 ,  B23K26/21 ,  B23K26/702

Abstract: A laser welding device includes a laser that generates a laser beam, an optics, and a limiting apparatus. The optics has a focal length of at least 200 nm and being configured to focus the laser beam onto a processing zone of a workpiece. The limiting apparatus limits a mixture of welding gases and heated ambient air, produced during laser welding, within the laser beam to a region that is less than the focal length from a surface of the workpiece.

Abstract translation: 激光焊接装置包括产生激光束的激光器，光学器件和限制装置。 光学元件具有至少200nm的焦距，并被配置为将激光束聚焦到工件的处理区域上。 限制装置将激光焊接期间产生的焊接气体和加热的环境空气的混合物限制在小于来自工件表面的焦距的区域内。

公开(公告)号：US20060079537A1

公开(公告)日：2006-04-13

申请号：US10531898

申请日：2003-11-14

Applicant: Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

Inventor： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC: A61K31/519 ,  C07D487/04

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: 2-Substituted triazolopyrimidines of the formula I, in which the substituents are as defined below: L are halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, —C(═O)-A or S(═O)pA′; A and A′ are as defined in the description; p is 0, 1 or 2; m is 0, 1, 2, 3, 4 or 5; X is cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered ring which may be interrupted by an atom from the group consisting of O, N and S, where R1 and/or R2 may be substituted as defined in the description; and R3 is cyano, hydroxyl, alkoxy, alkenyloxy, haloalkoxy, haloalkenyloxy, NR1R2 or S(O)nR31, where n and R31 are as defined in the description; Processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

Abstract translation: 氰基，硝基，烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基，烯氧基，炔氧基，卤代烷氧基，-C（ - O） - 取代的取代基如下： -A或S（-O） A'; A和A'如说明书所定义; p为0,1或2; m为0,1,2,3,4或5; X是氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，链二烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，苯基，萘基或五 - 至十元饱和的，部分不饱和的或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 1和R 2连同 它们所连接的氮原子也可以形成可被来自O，N和S的原子间隔的五元或六元环，其中R 1和/或 R 2可以如说明书中定义的取代; 和R 3是氰基，羟基，烷氧基，烯氧基，卤代烷氧基，卤代烯氧基，NR 1 R 2或S（O）n 其中n和R 31如在说明书中所定义的; 描述了制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20050272749A1

公开(公告)日：2005-12-08

申请号：US10531981

申请日：2003-11-04

Applicant: Jordi Tormo Blasco ,  Carsten Bletner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

Inventor： Jordi Tormo Blasco ,  Carsten Bletner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC: C07D487/04 ,  A61K31/519

CPC classification number: C07D487/04

Abstract: 5-Alkyl-7-aminotriazolopyrimidines of the formula I, where: R1, R2 are hydrogen, alkyl, alkenyl, alkynyl, haloalkyl, cycloalkyl, phenyl, naphthyl; 5- or 6-membered saturated, unsaturated or aromatic heterocyclyl which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or R1 and R2 together with the bridging nitrogen atom can form a 5- or 6-membered ring which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R3 is cycloalkyl or bicycloalkyl; where R1, R2 and R3 may be substituted as outlined in the description; X is alkyl or haloalkyl; and their salts; processes and intermediates for their preparation, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

Abstract translation: 式I的5-烷基-7-氨基三唑并嘧啶，其中：R 1，R 2是氢，烷基，烯基，炔基，卤代烷基，环烷基，苯基，萘基; 含有1-4个氮原子或一至三个氮原子和一个硫或氧原子的5-或6-元饱和，不饱和或芳族杂环基; 或R 1和R 2与桥连氮原子一起可以形成含有1-4个氮原子或一至三个氮原子的5-或6-元环，并且 一个硫或氧原子; R 3是环烷基或双环烷基; 其中R 1，R 2和R 3可以如说明书中概述的那样被取代; X是烷基或卤代烷基; 和它们的盐; 描述了其制备方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20050143344A1

公开(公告)日：2005-06-30

申请号：US11022075

申请日：2004-12-23

Applicant: Jerome Zeldis ,  Herbert Faleck ,  Peter Schafer

Inventor： Jerome Zeldis ,  Herbert Faleck ,  Peter Schafer

IPC: A61K31/00 ,  A61K31/454 ,  A61K31/724

CPC classification number: A61K31/454 ,  A61K31/00

Abstract: Methods of treating, preventing and/or managing central nervous system disorders, such as Amyotrophic Lateral Sclerosis (ALS or Lou Gehrig's Disease) and related syndromes are disclosed. Specific methods encompass the administration of an immunomodulatory compound of the invention, or a pharmaceutically acceptable salt, solvate, hydrate, stereoisomer, clathrate, or prodrug thereof, alone or in combination with a second active ingredient. Pharmaceutical compositions, single unit dosage forms, and kits suitable for use in methods of the invention are also disclosed.

Abstract translation: 公开了治疗，预防和/或控制中枢神经系统疾病如肌萎缩性侧索硬化症（ALS或Lou Gehrig's disease）及相关综合征的方法。 具体方法包括单独或与第二活性成分组合施用本发明的免疫调节化合物或其药学上可接受的盐，溶剂合物，水合物，立体异构体，包合物或前药。 还公开了适用于本发明方法的药物组合物，单一单位剂型和试剂盒。

公开(公告)号：US6150303A

公开(公告)日：2000-11-21

申请号：US463246

申请日：2000-01-21

Applicant: Olaf Menke ,  Markus Menges ,  Gerhard Hamprecht ,  Robert Reinhard ,  Peter Schafer ,  Cyrill Zagar ,  Karl-Otto Westphalen ,  Ulf Misslitz ,  Helmut Walter

Inventor： Olaf Menke ,  Markus Menges ,  Gerhard Hamprecht ,  Robert Reinhard ,  Peter Schafer ,  Cyrill Zagar ,  Karl-Otto Westphalen ,  Ulf Misslitz ,  Helmut Walter

IPC: A01N43/80 ,  C07D261/04 ,  A01N43/72

CPC classification number: C07D261/04

Abstract: Substituted 3-phenylisoxazolines I, and their salts and enol ethers, are described as herbicides ##STR1## where X.dbd.--O--, --S--, --N(R.sup.9)--;R.sup.1 .dbd.CN, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -haloalkoxy, C.sub.1 -C.sub.4 -alkylsulfonyl;R.sup.2 .dbd.H or unsubstituted or substituted C.sub.1 -C.sub.6 -alkyl, (C.sub.1 -C.sub.6 -alkyl)carbonyl, C.sub.1 -C.sub.6 -alkylsulfonyl, C.sub.2 -C.sub.6 -alkenyl, (C.sub.2 -C.sub.6 -alkenyl)carbonyl, C.sub.2 -C.sub.6 -alkynyl, (C.sub.2 -C.sub.6 -alkynyl)carbonyl;R.sup.3 .dbd.H, halogen;R.sup.4 .dbd.CN, halogen, C.sub.1 -C.sub.3 -haloalkyl;R.sup.5 .dbd.H, CN, halogen, C.sub.1 -C.sub.3 -haloalkyl;R.sup.6 .dbd.H, CN, halogen, C.sub.1 -C.sub.3 -haloalkyl or unsubstituted or substituted C.sub.1 -C.sub.6 -alkoxy;R.sup.7 .dbd.CN, halogen;R.sup.8 in position .alpha., R.sup.7 in this case being in position .beta., or in position .beta., R.sup.7 in this case being in position .alpha., is1) H, OH, SH, CN, NO.sub.2, halogen, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl, C.sub.1 -C.sub.6 -haloalkoxy, C.sub.1 -C.sub.6 -haloalkylthio, C.sub.1 -C.sub.6 -alkylthio-(C.sub.1 -C.sub.6 -alkyl)carbonyl, (C.sub.1 -C.sub.6 -alkyl)iminooxycarbonyl, C.sub.1 -C.sub.6 -alkoxy-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -alkoxyamino-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -alkoxy-C.sub.1 -C.sub.6 -alkylamino-C.sub.1 -C.sub.6 -alkyl,2) unsubstituted or substituted C.sub.1 -C.sub.6 -alkoxy, C.sub.1 -C.sub.6 -alkylthio, C.sub.3 -C.sub.6 -cycloalkoxy, C.sub.3 -C.sub.6 -cycloalkylthio, C.sub.2 -C.sub.6 -alkenyloxy, C.sub.2 -C.sub.6 -alkenylthio, C.sub.2 -C.sub.6 -alkynyloxy, C.sub.2 -C.sub.6 -alkynylthio, (C.sub.1 -C.sub.6 -alkyl)carbonyloxy, (C.sub.1 -C.sub.6 -alkyl)carbonylthio, (C.sub.1 -C.sub.6 -alkoxy)carboxyloxy, (C.sub.2 -C.sub.6 -alkenyl)carbonyloxy, (C.sub.2 -C.sub.6 -alkenyl)carbonylthio, (C.sub.2 -C.sub.6 -alkynyl)carbonyloxy, (C.sub.2 -C.sub.6 -alkynyl)carbonylthio, C.sub.1 -C.sub.6 -alkylsulfonyloxy or C.sub.1 -C.sub.6 -alkylsulfonyl,3) 29 further radicals;R.sup.9 .dbd.H, C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, C.sub.1 -C.sub.6 -alkoxy-C.sub.1 -C.sub.6 -alkyl, (C.sub.1 -C.sub.6 -alkoxy)carbonyl-C.sub.1 -C.sub.6 -alkyl, (C.sub.3 -C.sub.6 -alkenyloxy)carbonyl-C.sub.1 -C.sub.6 -alkyl, unsubstituted or substituted phenyl or phenyl-C.sub.1 -C.sub.6 -alkyl.

公开(公告)号：US6031106A

公开(公告)日：2000-02-29

申请号：US142767

申请日：1998-09-14

Applicant: Albrecht Harreus ,  Norbert Gotz ,  Michael Rack ,  Heinz Isak ,  Peter Schafer

Inventor： Albrecht Harreus ,  Norbert Gotz ,  Michael Rack ,  Heinz Isak ,  Peter Schafer

IPC: B01J23/42 ,  C07D213/61 ,  C07D213/38 ,  C07D213/42

CPC classification number: C07D213/61

Abstract: A process for preparing pyridyl-substituted N-phenylhydroxylamines by catalytic hydrogenation of the corresponding nitro compounds in the presence of an N-substituted morpholine compound and rearrangement of the hydroxylamine compounds obtained to pyridyl-4-fluoraniline compounds is described.

Abstract translation: PCT No.PCT / EP97 / 01336 Sec。 371日期：1998年9月14日 102（e）1998年9月14日PCT PCT 1997年3月17日PCT公布。 公开号WO97 / 34872 日期：1997年9月25日描述了在N-取代的吗啉化合物存在下，通过相应的硝基化合物的催化氢化制备吡啶基取代的N-苯基羟胺的方法，以及所得的羟胺化合物的重排反应到吡啶基-4-氟苯胺化合物。

公开(公告)号：US6013606A

公开(公告)日：2000-01-11

申请号：US765180

申请日：1997-06-30

Applicant: Ralf Klintz ,  Gerhard Hamprecht ,  Elisabeth Heistracher ,  Peter Schafer ,  Christoph-Sweder von dem Bussche-Hunnefeld ,  Peter Munster ,  Reinhard Kirstgen ,  Albrecht Harreus ,  Karl-Otto Westphalen ,  Matthias Gerber ,  Helmut Walter

Inventor： Ralf Klintz ,  Gerhard Hamprecht ,  Elisabeth Heistracher ,  Peter Schafer ,  Christoph-Sweder von dem Bussche-Hunnefeld ,  Peter Munster ,  Reinhard Kirstgen ,  Albrecht Harreus ,  Karl-Otto Westphalen ,  Matthias Gerber ,  Helmut Walter

IPC: C07D239/52 ,  A01N37/32 ,  A01N37/50 ,  A01N43/38 ,  A01N43/54 ,  C07C251/40 ,  C07C259/06 ,  C07C265/14 ,  C07C271/28 ,  C07C271/58 ,  C07C331/28 ,  C07D209/48 ,  C07D239/54 ,  C07D239/56 ,  C07D239/58 ,  C07D413/10 ,  A01N43/50 ,  C07D223/10 ,  C07D235/26

CPC classification number: C07D209/48 ,  A01N37/32 ,  A01N37/50 ,  A01N43/54 ,  C07C251/40 ,  C07C259/06 ,  C07C265/14 ,  C07C271/28 ,  C07C271/58 ,  C07C331/28 ,  C07D239/54

Abstract: Substituted cinnamic oxime derivatives I and cinnamic hydroxamide derivatives II ##STR1## (R.sup.1= halogen, NO.sub.2, CN, CF.sub.3 ; R.sup.2 =H, halogen; R.sup.3= H, halogen, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, hydroxy-C.sub.1 -C.sub.6 -alkyl;R.sup.4= H, halogen, CN, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl orR.sup.3 +R.sup.4 =chemical bond;Y=--O--, --S--, --O--CO--, --O--SO.sub.2 -- or chemical bond;Y'=--O-- or --S--;R.sup.5= unsubst. or subst. C.sub.1 -C.sub.6 -alkyl or C.sub.1 -C.sub.6 -haloalkyl; C.sub.3 -C.sub.6 -cycloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, unsubst. or subst. phenyl or phenyl-C.sub.1 -C.sub.6 -alkyl, or, if Y is --O--, --S-- or a chemical bond, is (C.sub.1 -C.sub.6 -alkyl)carbonyl or (C.sub.1 -C.sub.6 -alkoxy)carbonyl; or, if Y is a chemical bond, is hydrogen or halogen;R.sup.5 '=R.sup.5, H or (C.sub.1 -C.sub.6 -haloalkyl)carbonyl;R.sup.6= H, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, hydroxy-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -alkoxy-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -alkylthio-C.sub.1 -C.sub.6 -alkyl, cyano-C.sub.1 -C.sub.6 -alkyl, (C.sub.1 -C.sub.6 -alkoxy) carbonyl-C.sub.1 -C.sub.6 -alkyl, (C.sub.1 -C.sub.6 -alkyl) carbonyl-C.sub.1 -C.sub.6 -alkyl, (C.sub.1 -C.sub.6 -alkyl)carbonyloxy-C.sub.1 -C.sub.6 -alkyl or unsubst. or subst. phenyl-C.sub.1 -C.sub.6 -alkyl;or, if Y is oxygen or sulfur, R.sup.5 +R.sup.6 together=unsubst. or subst. C.sub.1 -C.sub.3 -alkylene;Cyc=N-(3,4,5,6-tetrahydrophthalimido) or ##STR2## X.sup.1, X.sup.2 =oxygen or sulfur; R.sup.7 =H, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl, NH.sub.2 ;R.sup.8, R.sup.9 =H, halogen, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl or unsubst. or subst. phenyl);and salts of I and II.Use: herbicides; desiccation/defoliation of plants.

Abstract translation: PCT No.PCT / EP95 / 02584第 371日期：1997年6月30日 102（e）日期1997年6月30日PCT提交1995年7月4日PCT公布。 第WO96 / 02518号公报 日期1996年2月1日取代肉桂肟衍生物I和肉桂酸羟基酰胺衍生物II（R1 =卤素，NO2，CN，CF3; R2 = H，卤素; R3 = H，卤素，C1-C6-烷基，C1-C6-卤代烷基， C3-C6-环烷基，C3-C6-烯基，C3-C6-炔基，羟基-C1-C6-烷基; R4 = H，卤素，CN，C1-C6-烷基，C1-C6-卤代烷基或R3 + R4 = 化学键; Y = -O-，-S-，-O-CO-，-O-SO2-或化学键; Y'= -O-或-S-; R5 =未取代或未取代的C1-C6- 烷基或C 1 -C 6 - 卤代烷基; C 3 -C 6 - 环烷基，C 3 -C 6 - 烯基，C 3 -C 6炔基，未取代或取代的苯基或苯基-C 1 -C 6烷基，或者如果Y是-O- （C 1 -C 6烷基）羰基或（C 1 -C 6 - 烷氧基）羰基;或者如果Y是化学键，则是氢或卤素; R 5'= R 5，H或（C 1 -C 6 - -C 6 - 卤代烷基）羰基; R 6 = H，C 1 -C 6烷基，C 1 -C 6卤代烷基，C 3 -C 6环烷基，C 3 -C 6 - 烯基，C 3 -C 6炔基，羟基-C 1 -C 6烷基， C 1 -C 6烷氧基-C 1 -C 6烷基，C 1 -C 6烷硫基-C 1 -C 6烷基，氰基-C 1 -C 6烷基，（C 1 -C 6 - 烷氧基）羰基-C 1 -C 6烷基，（C 1 -C 6 - 烷基）羰基-C 1 -C 6 - 烷基，（C 1 -C 6 - 烷基）羰基氧基 -C 1 -C 6 - 烷基或未取代基。 或subst。 苯基-C 1 -C 6 - 烷基; 或者如果Y是氧或硫，则R5 + R6一起=不成立。 或subst。 C1-C3-亚烷基; Cyc = N-（3,4,5,6-四氢邻苯二甲酰亚氨基）或X1，X2 =氧或硫; R7 = H，C1-C6-烷基，C1-C6-卤代烷基，NH2; R8，R9 = H，卤素，C1-C6-烷基，C1-C6-卤代烷基或未取代基。 或subst。 苯基）; 和I和II的盐。 用途：除草剂; 植物的干燥/脱叶。

公开(公告)号：US5962694A

公开(公告)日：1999-10-05

申请号：US068306

申请日：1998-05-07

Applicant: Cyrill Zagar ,  Albrecht Harreus ,  Christoph-Sweder von dem Bussche-Hunnefeld ,  Gerhard Hamprecht ,  Elisabeth Heistracher ,  Peter Schafer ,  Olaf Menke ,  Karl-Otto Westphalen ,  Ulf Misslitz ,  Helmut Walter

Inventor： Cyrill Zagar ,  Albrecht Harreus ,  Christoph-Sweder von dem Bussche-Hunnefeld ,  Gerhard Hamprecht ,  Elisabeth Heistracher ,  Peter Schafer ,  Olaf Menke ,  Karl-Otto Westphalen ,  Ulf Misslitz ,  Helmut Walter

IPC: A01N43/56 ,  C07D231/18 ,  C07D231/20

CPC classification number: A01N43/56 ,  C07D231/18 ,  C07D231/20

Abstract: Substituted 1-methyl-3-phenylpyrazoles I and their agriculturally useful acid addition salts ##STR1## where R.sup.1 =C.sub.1 -C.sub.4 -haloalkoxy or C.sub.1-C.sub.4 -haloalkylthio;R.sup.2 =halogen; R.sup.3 =F or Cl;R.sup.4 =CN, C.sub.1 -C.sub.4 -fluoroalkyl, C.sub.2 -C.sub.4 -fluoroalkenyl or --C(R.sup.5)(X-R.sup.6)(Y-R.sup.7);R.sup.5 =H or C.sub.1 -C.sub.4 -alkyl; X and Y=--O-- or --S--;R.sup.6, R.sup.7 =C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.3 -C.sub.4 -alkenyl, C.sub.3 -C.sub.4 -haloalkenyl or C.sub.3 -C.sub.4 -alkynyl;are used as herbicides; for the desiccation/defoliation of plants.

Abstract translation: PCT No.PCT / EP96 / 04819 Sec。 371日期1998年5月7日 102（e）日期1998年5月7日PCT提交1996年11月5日PCT公布。 公开号WO97 / 18195 PCT 日期1997年5月22日取代的1-甲基-3-苯基吡唑I及其农业上可用的酸加成盐，其中R 1 = C 1 -C 4 - 卤代烷氧基或C 1 -C 4 - 卤代烷硫基; R2 =卤素; R3 = F或Cl; R4 = CN，C1-C4-氟烷基，C2-C4-氟链烯基或-C（R5）（X-R6）（Y-R7）; R5 = H或C1-C4-烷基; X和Y = -O-或-S-; R6，R7 = C1-C4-烷基，C1-C4-卤代烷基，C3-C4-烯基，C3-C4-卤代烯基或C3-C4-炔基; 用作除草剂; 用于植物的干燥/脱叶。