Invention Publication
- Patent Title: PEPTIDE-COMPOUND CYCLIZATION METHOD
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Application No.: US18460300Application Date: 2023-09-01
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Publication No.: US20240166689A1Publication Date: 2024-05-23
- Inventor: Shiori KARIYUKI , Takeo IIDA , Miki KOJIMA , Ryuichi TAKEYAMA , Mikimasa TANADA , Tetsuo KOJIMA , Hitoshi IIKURA , Atsushi MATSUO , Takuya SHIRAISHI , Takashi EMURA , Kazuhiko NAKANO , Koji TAKANO , Kousuke ASOU , Takuya TORIZAWA , Ryusuke TAKANO , Nozomi HISADA , Naoaki MURAO , Atsushi OHTA , Kaori KIMURA , Yusuke YAMAGISHI , Tatsuya KATO
- Applicant: Chugai Seiyaku Kabushiki Kaisha
- Applicant Address: JP Tokyo
- Assignee: Chugai Seiyaku Kabushiki Kaisha
- Current Assignee: Chugai Seiyaku Kabushiki Kaisha
- Current Assignee Address: JP Tokyo
- Priority: JP 11288865 2011.12.28 JP 12156943 2012.07.12
- Main IPC: C07K7/64
- IPC: C07K7/64 ; C07H21/04 ; C07K1/113 ; C07K5/087 ; C07K5/103 ; C07K7/06 ; C07K7/08 ; C07K11/00 ; C07K11/02 ; C07K19/00 ; C12P21/02

Abstract:
An object of the present invention is to provide methods of discovering drugs effective for tough targets, which have conventionally been discovered only with difficulty. The present invention relates to novel methods for cyclizing peptide compounds, and novel peptide compounds and libraries comprising the same, to achieve the above object.
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