发明申请
US20160122340A1 HISTONE DEACETYLASE INHIBITORS BASED ON DERIVATIVES OF TRICYCLIC POLYHYDROACRIDINE AND ANALOGS POSSESSING FUSED SATURATED FIVE-AND-SEVEN-MEMBERED RINGS
审中-公开
基于TRICYCLIC聚羟基吡啶衍生物的组蛋白脱乙酰壳多糖抑制剂和受损的饱和饱和五元配合环的模拟物
- 专利标题： HISTONE DEACETYLASE INHIBITORS BASED ON DERIVATIVES OF TRICYCLIC POLYHYDROACRIDINE AND ANALOGS POSSESSING FUSED SATURATED FIVE-AND-SEVEN-MEMBERED RINGS
- 专利标题（中）： 基于TRICYCLIC聚羟基吡啶衍生物的组蛋白脱乙酰壳多糖抑制剂和受损的饱和饱和五元配合环的模拟物
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申请号： US14890031申请日： 2014-05-09
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公开(公告)号： US20160122340A1公开(公告)日： 2016-05-05
- 发明人: Fernando Pedro COSSÍO MORA , Yosu Ion VARA SALAZAR , María del Carmen MASDEU MARGALEF , María Remedios ALCALÁ CAFFARENA , Sergio VILLAFRUELA CÁNEVA , Dorleta OTAEGUI ANSA , Eneko ALDABA ARÉVALO , Aizpea ZUBIA OLASCOAGA , Eider SAN SEBASTIÁN LARZABAL
- 申请人： QUIMATRYX, S.L. , UNIVERSIDAD DEL PAÍS VASCO
- 优先权： EP13382170.2 20130509
- 国际申请： PCT/EP2014/059554 WO 20140509
- 主分类号： C07D471/04
- IPC分类号： C07D471/04 ; C07D401/12 ; C07D219/04 ; C07D219/10 ; C07D221/16
摘要：
The present invention refers to compounds of formula (I): as well as to a method for their preparation, pharmaceutical compositions comprising the same, and use thereof for the treatment and/or chemoprevention of cancer hematological malignancy, proliferative diseases, neurological disorders and immunological disorders.
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