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1.发明申请Synthetic Rigidin Analogues as Anticancer Agents, Salts, Solvates and Prodrugs Thereof, and Method of Producing Same 有权合成菱镁苷类似物作为抗癌剂，盐，溶剂化物和前体药物及其生产方法公开(公告)号：US20140142125A1
公开(公告)日：2014-05-22
申请号：US13678987
申请日：2012-11-16
IPC分类号： C07D487/04
CPC分类号： C07D487/04
摘要： A compound having the Formula I as follows: wherein R1 and R2 are selected from hydrogen, aryl, fused aryl, heteroaryl, saturated carbocylclic, partially saturated carbocyclic, saturated heterocyclic, partially saturated heterocyclic, C1-10 alkyl, haloalkyl, alkenyl, alkynyl, arylalkyl, arylalkenyl, arylalkynyl, heteroarylalkyl, heteroarylalkenyl, carbocycloalkyl, heterocycloalkyl, hydroxyalkyl, aminoalkyl, carboxyalkyl, nitroalkyl, cyanoalkyl, acetamidoalkyl, and acyloxyalkyl. A process for the preparation thereof is also provided.
摘要翻译： 具有式I的化合物如下：其中R 1和R 2选自氢，芳基，稠合芳基，杂芳基，饱和碳环，部分饱和碳环，饱和杂环，部分饱和杂环，C 1-10烷基，卤代烷基，烯基，炔基， 芳基烷基，芳基烯基，芳基炔基，杂芳基烷基，杂芳基烯基，碳环烷基，杂环烷基，羟基烷基，氨基烷基，羧基烷基，硝基烷基，氰基烷基，乙酰氨基烷基和酰氧基烷基。 还提供了其制备方法。
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2.发明授权Synthetic rigidin analogues as anticancer agents, salts, solvates and prodrugs thereof, and method of producing same 有权作为抗癌剂，其盐，溶剂化物和前体药物的合成嘧啶类似物及其制备方法公开(公告)号：US09334280B2
公开(公告)日：2016-05-10
申请号：US14584929
申请日：2014-12-29
IPC分类号： A01N43/90 , A61K31/519 , C07D487/00 , C07D487/04
CPC分类号： C07D487/04 , A61K31/519
摘要： A compound having the Formula as follows: wherein R, R1 and R2 are selected from hydrogen, aryl, fused aryl, heteroaryl, saturated carbocylclic, partially saturated carbocyclic, saturated heterocyclic, partially saturated heterocyclic, C1-10 alkyl, haloalkyl, alkenyl, alkynyl, arylalkyl, arylalkenyl, arylalkynyl, heteroarylalkyl, heteroarylalkenyl, alkenylalkyl, alkynylalkyl, carbocycloalkyl, heterocycloalkyl, hydroxyalkyl, aminoalkyl, carboxyalkyl, nitroalkyl, cyanoalkyl, acetamidoalkyl, and acyloxyalkyl. A process for the preparation thereof is also provided.
摘要翻译： 具有下式的化合物：其中R 1，R 2和R 2选自氢，芳基，稠合芳基，杂芳基，饱和碳环，部分饱和碳环，饱和杂环，部分饱和杂环，C 1-10烷基，卤代烷基，烯基，炔基 芳基烷基，芳基烯基，芳基炔基，杂芳基烷基，杂芳基烯基，烯基烷基，炔基烷基，碳环烷基，杂环烷基，羟基烷基，氨基烷基，羧基烷基，硝基烷基，氰基烷基，乙酰氨基烷基和酰氧基烷基。 还提供了其制备方法。
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3.发明申请Synthetic Rigidin Analogues as Anticancer Agents, Salts, Solvates and Prodrugs Thereof, and Method of Producing Same 有权合成菱镁苷类似物作为抗癌剂，盐，溶剂化物和前体药物及其生产方法公开(公告)号：US20150111906A1
公开(公告)日：2015-04-23
申请号：US14584929
申请日：2014-12-29
IPC分类号： C07D487/04
CPC分类号： C07D487/04 , A61K31/519
摘要： A compound having the Formula as follows: wherein R, R1 and R2 are selected from hydrogen, aryl, fused aryl, heteroaryl, saturated carbocylclic, partially saturated carbocyclic, saturated heterocyclic, partially saturated heterocyclic, C1-10 alkyl, haloalkyl, alkenyl, alkynyl, arylalkyl, arylalkenyl, arylalkynyl, heteroarylalkyl, heteroarylalkenyl, alkenylalkyl, alkynylalkyl, carbocycloalkyl, heterocycloalkyl, hydroxyalkyl, aminoalkyl, carboxyalkyl, nitroalkyl, cyanoalkyl, acetamidoalkyl, and acyloxyalkyl. A process for the preparation thereof is also provided.
摘要翻译： 具有下式的化合物：其中R 1，R 2和R 2选自氢，芳基，稠合芳基，杂芳基，饱和碳环，部分饱和碳环，饱和杂环，部分饱和杂环，C 1-10烷基，卤代烷基，烯基，炔基 芳基烷基，芳基烯基，芳基炔基，杂芳基烷基，杂芳基烯基，烯基烷基，炔基烷基，碳环烷基，杂环烷基，羟基烷基，氨基烷基，羧基烷基，硝基烷基，氰基烷基，乙酰氨基烷基和酰氧基烷基。 还提供了其制备方法。
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4.发明授权Synthetic rigidin analogues as anticancer agents, salts, solvates and prodrugs thereof, and method of producing same 有权作为抗癌剂，其盐，溶剂化物和前体药物的合成嘧啶类似物及其制备方法公开(公告)号：US08946246B2
公开(公告)日：2015-02-03
申请号：US13678987
申请日：2012-11-16
IPC分类号： A01N43/90 , A61K31/519 , C07D487/00 , C07D487/04
CPC分类号： C07D487/04
摘要： A compound having the Formula I as follows: wherein R1 and R2 are selected from hydrogen, aryl, fused aryl, heteroaryl, saturated carbocylclic, partially saturated carbocyclic, saturated heterocyclic, partially saturated heterocyclic, C1-10 alkyl, haloalkyl, alkenyl, alkynyl, arylalkyl, arylalkenyl, arylalkynyl, heteroarylalkyl, heteroarylalkenyl, carbocycloalkyl, heterocycloalkyl, hydroxyalkyl, aminoalkyl, carboxyalkyl, nitroalkyl, cyanoalkyl, acetamidoalkyl, and acyloxyalkyl. A process for the preparation thereof is also provided.
摘要翻译： 具有式I的化合物如下：其中R 1和R 2选自氢，芳基，稠合芳基，杂芳基，饱和碳环，部分饱和碳环，饱和杂环，部分饱和杂环，C 1-10烷基，卤代烷基，烯基，炔基， 芳基烷基，芳基烯基，芳基炔基，杂芳基烷基，杂芳基烯基，碳环烷基，杂环烷基，羟基烷基，氨基烷基，羧基烷基，硝基烷基，氰基烷基，乙酰氨基烷基和酰氧基烷基。 还提供了其制备方法。
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