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公开(公告)号：US20210009589A1
公开(公告)日：2021-01-14
申请号：US17034240
申请日：2020-09-28
发明人： Jérôme HERT , Daniel HUNZIKER , Patrizio MATTEI , Markus RUDOLPH , Petra SCHMITZ , Patrick DI GIORGIO
IPC分类号： C07D471/04 , A61K9/20 , A61K9/48 , C07D401/14 , C07D405/14 , C07D495/04 , C07D498/04 , C07D513/04 , C07D519/00
摘要： The invention provides novel compounds having the general formula (I) wherein R1, R2, Y, W, A, X, m and n are as defined herein, compositions including the compounds and methods of using the compounds.
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公开(公告)号：US20200223854A1
公开(公告)日：2020-07-16
申请号：US16832553
申请日：2020-03-27
发明人： Patrick DI GIORGIO , Jerome HERT , Daniel HUNZIKER , Patrizio MATTEI , Markus RUDOLPH , Petra SCHMITZ , Christoph ULLMER
IPC分类号： C07D487/04 , A61K31/5517 , A61K31/407 , C07D471/04 , A61K31/437 , A61P27/02
摘要： The invention provides novel compounds having the general formula (I) wherein R1, R2, Y, W, m, n, p and q are as defined herein, compositions including the compounds and methods of using the compounds.
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![OCTAHYDRO-CYCLOBUTA[1,2-c;3,4-c']DIPYRROL-2-YL](/abs-image/US/2021/01/21/US20210015792A1/abs.jpg.150x150.jpg)
公开(公告)号：US20210015792A1
公开(公告)日：2021-01-21
申请号：US17034323
申请日：2020-09-28
发明人： Patrizio MATTEI , Daniel HUNZIKER , Patrick DI GIORGIO , Jerome HERT , Markus RUDOLPH , Lisha WANG
IPC分类号： A61K31/407 , C07D209/56 , C07D487/04
摘要： The invention provides novel compounds having the general formula (I) wherein R1, Y and R2 are as described herein, compositions including the compounds and methods of using the compounds.
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公开(公告)号：US20190185426A1
公开(公告)日：2019-06-20
申请号：US16283640
申请日：2019-02-22
IPC分类号： C07D207/12 , C07D401/12 , C07D403/12 , C07D409/12
CPC分类号： C07D207/12 , C07D401/12 , C07D403/12 , C07D409/12
摘要： The invention provides novel compounds having the general formula (I) wherein R2, R3, R4, R5, R6, R7, R8, X, A and R11 are as described herein, compositions including the compounds and methods of using the compounds.
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公开(公告)号：US20230234939A1
公开(公告)日：2023-07-27
申请号：US18114959
申请日：2023-02-27
发明人： Sandra Marie Joseph GRALL-ULSEMER , Wolfgang GUBA , Christian LERNER , Mingming LI , Yongqiang LIU , Markus RUDOLPH , Sébastien SCHMITT , Lorenz URNER , Yongguang WANG , Min WANG , Jianhua WANG , Song YANG , Chengang ZHOU , Patrizio MATTEI
IPC分类号： C07D401/14 , C07D403/14 , A61P31/04
CPC分类号： C07D401/14 , C07D403/14 , A61P31/04
摘要： The invention provides novel imidazole pyrazole derivatives having the general formula (I), and pharmaceutically acceptable salts thereof, wherein A and R1-R7 are as described herein:
Further provided are pharmaceutical compositions including the compounds, processes of manufacturing the compounds and methods of using the compounds as medicaments, in particular methods of using the compounds as antibiotics for the treatment or prevention of bacterial infections and resulting diseases.-
公开(公告)号：US20200002336A1
公开(公告)日：2020-01-02
申请号：US16569459
申请日：2019-09-12
发明人： Jérôme HERT , Daniel HUNZIKER , Patrizio MATTEI , Markus RUDOLPH , Petra SCHMITZ , Patrick DI GIORGIO
IPC分类号： C07D471/04 , C07D405/14 , C07D498/04 , C07D401/14 , C07D519/00 , C07D513/04 , C07D495/04 , A61K9/20 , A61K9/48
摘要： The invention provides novel compounds having the general formula (I) wherein R1, R2, Y, W, A, X, m and n are as defined herein, compositions including the compounds and methods of using the compounds.
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公开(公告)号：US20200002297A1
公开(公告)日：2020-01-02
申请号：US16569475
申请日：2019-09-12
发明人： Patrizio MATTEI , Jérôme HERT , Daniel HUNZIKER , Markus RUDOLPH , Petra SCHMITZ , Patrick DI GIORGIO , Justin GOMME
IPC分类号： C07D257/04 , C07D405/14 , C07D401/12 , C07D401/14 , C07D405/12 , C07D401/10 , C07D403/10 , C07D417/14 , C07D401/06 , C07D409/14
摘要： The invention provides novel compounds having the general formula (I) wherein R1, R2, Y, X, W, m and n are as defined herein, compositions including the compounds and methods of using the compounds.
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公开(公告)号：US20190152895A1
公开(公告)日：2019-05-23
申请号：US16250905
申请日：2019-01-17
IPC分类号： C07C237/22 , C07D295/13 , C07D213/65 , C07C255/54
摘要： The invention provides novel compounds having the general formula (I) wherein R1, R2, R3, R4, R5, R6, R7, R3, R8, R9, R10 and R11 are as described herein, compositions including the compounds and methods of using the compounds.
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公开(公告)号：US20180148450A1
公开(公告)日：2018-05-31
申请号：US15850826
申请日：2017-12-21
发明人： Bernd BUETTELMANN , Buelent KOCER , Bernd KUHN , Marco PRUNOTTO , Hans RICHTER , Martin RITTER , Markus RUDOLPH , Alexander Lee SATZ
IPC分类号： C07D471/10 , C07D519/00 , A61P13/12 , A61P1/16 , A61P9/00 , A61P35/00 , A61P37/06
CPC分类号： C07D471/10 , A61P1/16 , A61P9/00 , A61P13/12 , A61P35/00 , A61P37/06 , C07D519/00
摘要： The present invention relates to compounds of formula (I): or pharmaceutically acceptable salts thereof, wherein L and R1 to R5 are as described herein, as well as processes for their manufacture, pharmaceutical compositions comprising them, and their use as medicaments.
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公开(公告)号：US20200339522A1
公开(公告)日：2020-10-29
申请号：US16811656
申请日：2020-03-06
发明人： Jerome HERT , Daniel HUNZIKER , Holger KUEHNE , Thomas LUEBBERS , Rainer E. MARTIN , Patrizio MATTEI , Werner NEIDHART , Hans RICHTER , Markus RUDOLPH , Emmanuel PINARD
IPC分类号： C07D249/08 , C07D487/04 , C07D249/12 , C07D409/12 , C07D413/12 , C07D231/12 , C07F7/08 , C07D401/12 , C07D407/12 , C07D407/04 , C07D471/04 , C07D237/14 , C07D403/12 , C07D417/12 , C07D231/56 , A61P27/02 , C07B41/04 , C07D231/20 , C07D249/04
摘要： The invention provides novel compounds having the general formula (I) wherein RA, RB, RC, RC1 and W are as defined herein, compositions including the compounds and methods of using the compounds.
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