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公开(公告)号:US20170298093A1
公开(公告)日:2017-10-19
申请号:US15513719
申请日:2015-08-29
Applicant: Biophore India Pharmaceuticals Pvt. Ltd
Inventor: Manik Reddy Pullagurla , Jagadeesh Babu Rangisetty , Mecheril Valsan Nanda Kumar , Surya Bala Subrahmanyam Pendyala , Bhaskar Reddy Pitta
IPC: C07K5/107 , C07C237/20 , C07D303/36 , C07K1/14
CPC classification number: C07K5/1016 , C07C237/20 , C07D303/36 , C07K1/14 , C07K5/1008
Abstract: Novel methods for preparation of Carfilzomib and intermediates thereof with high stereo selection are reported. The synthetic procedures result in substantially pure Carfilzomib (I).
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公开(公告)号:US10329325B2
公开(公告)日:2019-06-25
申请号:US15513719
申请日:2015-08-29
Applicant: Biophore India Pharmaceuticals Pvt. Ltd
Inventor: Manik Reddy Pullagurla , Jagadeesh Babu Rangisetty , Mecheril Valsan Nanda Kumar , Surya Bala Subrahmanyam Pendyala , Bhaskar Reddy Pitta
IPC: C07K9/00 , C07K5/107 , C07K5/103 , C07C237/20 , C07D303/36 , C07K1/14
Abstract: Novel methods for preparation of Carfilzomib and intermediates thereof with high stereo selection are reported. The synthetic procedures result in substantially pure Carfilzomib (I).
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