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公开(公告)号:US20140038999A1
公开(公告)日:2014-02-06
申请号:US13946344
申请日:2013-07-19
Applicant: Bristol-Myers Squibb Company
Inventor: Vivekananda M. Vrudhula , Senliang Pan , Ramkumar Rajamani , Susheel Jethanand Nara , Maheswaran Sivasamban Karatholuvhu , Tarun Kumar Maishal , Jonathan L. Ditta , Carolyn Diane Dzierba , Joanne J. Bronson , John E. Macor
IPC: C07D471/04
CPC classification number: C07D471/04
Abstract: The present disclosure is generally directed to compounds which can inhibit AAK1 (adaptor associated kinase 1), compositions comprising such compounds, and methods for inhibiting AAK1.
Abstract translation: 本公开一般涉及可以抑制AAK1(衔接子相关激酶1),包含这些化合物的组合物和抑制AAK1的方法的化合物。
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公开(公告)号:US20160222021A1
公开(公告)日:2016-08-04
申请号:US14917306
申请日:2013-09-11
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Vivekananda M. Vrudhula , Senliang Pan , Ramkumar Rajamani , John E. Macor , Joanne J. Bronson , Carolyn Diane Dzierba , Susheel Jethanand Nara , Maheswaran Sivasamban Karatholuvhu
IPC: C07D491/052 , C07D491/20
CPC classification number: C07D491/052 , C07D491/04 , C07D491/20
Abstract: The present disclosure is generally directed to compounds which can inhibit AAK1 (adaptor associated kinase 1), compositions comprising such compounds, and methods for inhibiting AAK1.
Abstract translation: 本公开一般涉及可以抑制AAK1(衔接子相关激酶1),包含这些化合物的组合物和抑制AAK1的方法的化合物。
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公开(公告)号:US08703953B2
公开(公告)日:2014-04-22
申请号:US13777144
申请日:2013-02-26
Applicant: Bristol-Myers Squibb Company
Inventor: Vivekananda M. Vrudhula , Senliang Pan , Ramkumar Rajamani , John E. Macor , Joanne J. Bronson , Carolyn Diane Dzierba , Susheel Jethanand Nara , Maheswaran Sivasamban Karatholuvhu
IPC: A61K31/44 , C07D491/00
CPC classification number: C12N9/99 , C07D491/04 , C07D491/052 , C07D491/20
Abstract: The present disclosure is generally directed to compounds which can inhibit AAK1 (adaptor associated kinase 1), compositions comprising such compounds, and methods for inhibiting AAK1.
Abstract translation: 本公开一般涉及可以抑制AAK1(衔接子相关激酶1),包含这些化合物的组合物和抑制AAK1的方法的化合物。
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公开(公告)号:US20130237555A1
公开(公告)日:2013-09-12
申请号:US13777144
申请日:2013-02-26
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Vivekananda M. Vrudhula , Senliang Pan , Ramkumar Rajamani , John E. Macor , Joanne J. Bronson , Carolyn Diane Dzierba , Susheel Jethanand Nara , Maheswaran Sivasamban Karatholuvhu
IPC: C07D491/052 , C12N9/99 , C07D491/20
CPC classification number: C12N9/99 , C07D491/04 , C07D491/052 , C07D491/20
Abstract: The present disclosure is generally directed to compounds which can inhibit AAK1 (adaptor associated kinase 1), compositions comprising such compounds, and methods for inhibiting AAK1.
Abstract translation: 本公开一般涉及可以抑制AAK1(衔接子相关激酶1),包含这些化合物的组合物和抑制AAK1的方法的化合物。
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公开(公告)号:US10174044B2
公开(公告)日:2019-01-08
申请号:US15563697
申请日:2016-04-04
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Susheel Jethanand Nara , Carolyn Diane Dzierba , John E. Macor , Joanne J. Bronson , Rajamani Ramkumar , Tarun Kumar Maishal , Maheswaran Sivasamban Karatholuvhu , Soodamani Thangavel , Kamalraj Thiyagarajan
IPC: A61K31/436 , C07D491/052 , C07D471/04 , C07D491/04 , A61P25/28 , A61P25/02 , A61P25/04 , A61P25/18 , A61P25/16 , C07B59/00
Abstract: The present disclosure is generally directed to compounds which can inhibit AAK1 (adaptor associated kinase 1), compositions comprising such compounds, and methods for inhibiting AAK1.
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公开(公告)号:US20160333006A1
公开(公告)日:2016-11-17
申请号:US15111416
申请日:2014-01-29
Applicant: Bristol-Myers Squibb Company
Inventor: Vivekananda M. Vrudhula , Senliang Pan , Ramkumar Rajamani , Susheel Jethanand Nara , Maheswaran Sivasamban Karatholuvhu , Tarun Kumar Maishal , Jonathan L. Ditta , Carolyn Diane Dzierba , Joanne J Bronson , John E. Macor
IPC: C07D471/04
CPC classification number: C07D471/04
Abstract: The present disclosure is generally directed to compounds which can inhibit AAK1 (adaptor associated kinase 1), compositions comprising such compounds, and methods for inhibiting AAK1.
Abstract translation: 本公开一般涉及可以抑制AAK1(衔接子相关激酶1),包含这些化合物的组合物和抑制AAK1的方法的化合物。
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公开(公告)号:US08969564B2
公开(公告)日:2015-03-03
申请号:US14188141
申请日:2014-02-24
Applicant: Bristol-Myers Squibb Company
Inventor: Vivekananda M. Vrudhula , Senliang Pan , Ramkumar Rajamani , John E. Macor , Joanne J. Bronson , Carolyn Diane Dzierba , Susheel Jethanand Nara , Maheswaran Sivasamban Karatholuvhu
IPC: A61K31/44 , C07D491/00 , C12N9/99 , C07D491/052 , C07D491/20 , C07D491/04
CPC classification number: C12N9/99 , C07D491/04 , C07D491/052 , C07D491/20
Abstract: The present disclosure is generally directed to compounds which can inhibit AAK1 (adaptor associated kinase 1), compositions comprising such compounds, and methods for inhibiting AAK1.
Abstract translation: 本公开一般涉及可以抑制AAK1(衔接子相关激酶1),包含这些化合物的组合物和抑制AAK1的方法的化合物。
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公开(公告)号:US20160332985A1
公开(公告)日:2016-11-17
申请号:US15112294
申请日:2015-01-23
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Richard A. Hartz , Vijay T. Ahuja , John E. Macor , Joanne J. Bronson , Bireshwar Dasgupta , Carolyn Diane Dzierba , Susheel Jethanand Nara , Maheswaran Sivasamban Karatholuvhu
IPC: C07D401/04 , C07D401/14 , C07D215/12 , C07D413/04 , C07D471/04
CPC classification number: C07D401/04 , C07D215/12 , C07D215/18 , C07D401/14 , C07D413/04 , C07D471/04
Abstract: The present disclosure is generally directed to compounds of formula (I) which can inhibit AAKI (adaptor associated kinase 1), compositions comprising such compounds, and methods for inhibiting AAKI.
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公开(公告)号:US20160016967A1
公开(公告)日:2016-01-21
申请号:US14767952
申请日:2014-02-06
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Vivekananda M. Vrudhula , Carolyn Diane Dzierba , Joanne J. Bronson , John E. Macor , Susheel Jethanand Nara , Ramkumar Rajamani , Maheswaran Sivasamban Karatholuvhu
IPC: C07D491/052
CPC classification number: C07D491/052
Abstract: The present disclosure is generally directed to compounds which can inhibit AAK1 (adaptor associated kinase 1), compositions comprising such compounds, and methods for inhibiting AAK1.
Abstract translation: 本公开一般涉及可以抑制AAK1(衔接子相关激酶1),包含这些化合物的组合物和抑制AAK1的方法的化合物。
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公开(公告)号:US08901305B2
公开(公告)日:2014-12-02
申请号:US13946344
申请日:2013-07-19
Applicant: Bristol-Myers Squibb Company
Inventor: Vivekananda M. Vrudhula , Senliang Pan , Ramkumar Rajamani , Susheel Jethanand Nara , Maheswaran Sivasamban Karatholuvhu , Tarun Kumar Maishal , Jonathan L. Ditta , Carolyn Diane Dzierba , Joanne J. Bronson , John E. Macor
IPC: A61K31/44 , C07D471/00 , C07D471/04
CPC classification number: C07D471/04
Abstract: The present disclosure is generally directed to compounds which can inhibit AAK1 (adaptor associated kinase 1), compositions comprising such compounds, and methods for inhibiting AAK1.
Abstract translation: 本公开一般涉及可抑制AAK1(衔接子相关激酶1),包含这些化合物的组合物和抑制AAK1的方法的化合物。
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