Preparation of 4,5-bis-(trifluoromethylimino)-thiazolidines
    1.
    发明授权
    Preparation of 4,5-bis-(trifluoromethylimino)-thiazolidines 失效
    制备4,5-双(三氟甲基亚氨基) - 噻唑啉

    公开(公告)号:US3895020A

    公开(公告)日:1975-07-15

    申请号:US20615871

    申请日:1971-12-08

    申请人: BAYER AG

    摘要: 4,5-Bis-(trifluoromethylimino)-thiazolidines are prepared by reacting the thiol form of a thiourea or a thiocarboxylic acid amide having at least one hydrogen atom on each urea of amide nitrogen atom with perfluoro-2,5-diazahexa-2,4-diene in the presence of a hydrogen fluoride acceptor at a temperature of about -50* to 120*C, in accordance with the following formula

    in which Z is N-R or

    and R, R'', R'''' and R'''''' each is hydrogen or various optionally substituted hydrocarbon or heterocyclic radicals, several of them together possibly forming a heterocyclic ring. The invention also extends to compositions containing, and methods of using, the new compounds to combat fungi, insects and acarids.

    摘要翻译: 通过使酰胺氮原子的每个尿素上具有至少一个氢原子的硫脲或硫代羧酸酰胺的硫醇形式与全氟-2,5-二氮杂六-2反应制备4,5-双 - (三氟甲基亚氨基) 在氟化氢受体存在下,在约-50℃至120℃的温度下,根据下式计算:SH FC = N-CF 3 SC = N-CF 3 Z = C ANGLE + | - > Z = C ANGLE | NH F-C = N-CF 3 NC = N-CF 3 | | R“'R”,其中Z为= NR或} R'} = C ANGLE} R“',R,R ',R“和R”'各自为氢或各种任选取代的烃或杂环基,其中几个可能形成杂环。

    Substituted amidophenylguanidine fungicides
    2.
    发明授权
    Substituted amidophenylguanidine fungicides 失效
    取代氨基苯胍杀真菌剂

    公开(公告)号:US3881018A

    公开(公告)日:1975-04-29

    申请号:US33718373

    申请日:1973-03-01

    申请人: BAYER AG

    CPC分类号: C07D307/68 A01N47/44

    摘要: IN WHICH EACH X independently denotes a halogen atom, lower alkyl or lower alkoxy, n denotes 0, 1 or 2, R denotes a hydrogen atom, or lower alkyl, R'' denotes alkyl with 1-12 carbon atoms, and R'''' denotes a hydrogen atom, alkyl with 1-18 carbon atoms, which may be substituted, cycloalkyl with 5-8 ring carbon atoms, aralkyl, which may be substituted, aryl, which may be substituted, or 2-furyl, which possess fungicidal properties.

    Substituted amidophenylguanidines of the formula

    摘要翻译: 取代的式IN的苯基胍其中每个X独立地表示卤素原子,低级烷基或低级烷氧基,n表示0,1或2,R表示氢原子或低级烷基,R'表示具有1-12个碳原子的烷基, 并且R“表示氢原子,具有1-18个碳原子的烷基,其可被取代,具有5-8个环碳原子的环烷基,可被取代的芳烷基,可被取代的芳基,或2-呋喃基, 具有杀菌性。

    N-trityl-imidazoles as plant fungicides
    3.
    发明授权
    N-trityl-imidazoles as plant fungicides 失效
    作为植物杀真菌剂的N-三嗪基咪唑

    公开(公告)号:US3665079A

    公开(公告)日:1972-05-23

    申请号:US3665079D

    申请日:1970-09-02

    申请人: BAYER AG

    IPC分类号: A01N9/22

    CPC分类号: C07D233/56

    摘要: Plant fungicidal compositions are produced which comprises an amount of a compound of the formula:

    WHEREIN R is alkyl of one or two carbon atoms substituted by one to five fluoro moieties, sufficient to be effective for killing, combating or controlling plant fungi, in combination with a solid or liquid diluent or carrier. Methods for killing, combatting or controlling fungal diseases in plants comprise applying to the fungi or to the plant to be protected an effective or toxic amount of the above compound.

    1-trityl-1,2,4-triazoles
    6.
    发明授权
    1-trityl-1,2,4-triazoles 失效
    1-TRITYL-1,2,4-TRIAZOLES

    公开(公告)号:US3682950A

    公开(公告)日:1972-08-08

    申请号:US3682950D

    申请日:1969-08-08

    申请人: BAYER AG

    摘要: 1-Trityl-1,2,4-triazoles, i.e. 1-((optionally mono and di chloro-, fluoro-, cyano- and trifluoromethyl-substituted)(optionally mono and di chloro-, fluoro-, cyano- and trifluoromethyl- substituted)-(optionally mono and di chloro-, fluoro-, cyano- and trifluoromethyl- substituted)-trityl)-3(optionally chloro substituted)-5-(optionally chloro substituted)-1,2,4-triazoles, or 1-((optionally mono and di chloro, fluoro-, cyano- and trifluoromethyl- substituted phenyl)(optionally mono and di chloro-, fluoro-, cyano- and trifluoromethyl- substituted phenyl)-(optionally mono and di chloro-, fluoro-, cyano- and trifluoromethyl-substituted phenyl)methyl)-3-(optionally chloro-substituted)-5-(optionally chloro substituted)-1,2,4-triazoles, which possess fungicidal properties and which may be produced by conventional methods.

    摘要翻译: 1-三苯甲基-1,2,4-三唑,即1 - [(任选单和二氯 - ,氟 - ,氰基 - 和三氟甲基取代的) - (任选单和二氯 - ,氟 - ,氰基 - 和三氟甲基 - 取代的) - (任选单和二氯 - ,氟 - ,氰基 - 和三氟甲基取代的) - 三苯甲基] -3-(任选氯代取代的)-5-(任选氯取代的)-1,2,4-三唑, 或1 - [(任选单和二氯,氟 - ,氰基 - 和三氟甲基取代的苯基) - (任选单和二氯 - ,氟 - ,氰基 - 和三氟甲基取代的苯基) - (任选单和二 - ,氟 - ,氰基 - 和三氟甲基取代的苯基) - 甲基] -3-(任选氯取代的)-5-(任选氯取代的)-1,2,4-三唑,其具有杀真菌性并且可以产生 通过常规方法。

    N-({107 -cyano-alkyl)-carbamyl-benzimidazoles
    7.
    发明授权
    N-({107 -cyano-alkyl)-carbamyl-benzimidazoles 失效
    N - ({107-氰基 - 烷基) - 氨基甲酰苯胺

    公开(公告)号:US3673210A

    公开(公告)日:1972-06-27

    申请号:US3673210D

    申请日:1969-11-26

    申请人: BAYER AG

    摘要: N-( omega -cyano-alkyl)-carbamyl-benzimidazoles, i.e., 2(optionally alkoxy-carbonyl and alkyl-carbonyl)-3-(N-( omega cyano-alkyl)-carbamyl)-4,5,6 and/or 7-(optionally alkyl)benzimidazoles, which possess fungicidal, anti-bacterial, insecticidal, acaricidal and ovicidal properties and which may be produced by conventional methods.

    摘要翻译: N-(ω-氰基 - 烷基) - 氨基甲酰基 - 苯并咪唑,即2-(任选的烷氧羰基和羰基羰基)-3- [N-(ω-氰基 - 烷基) - 氨基甲酰基] -4,5,6 和/或7-(任选烷基) - 苯并咪唑,其具有杀真菌剂,抗细菌剂,杀虫剂,杀螨剂和杀卵剂的性质,并且可以通过常规方法制备。

    Fungicidal substituted ureidophenyl thioureas
    10.
    发明授权
    Fungicidal substituted ureidophenyl thioureas 失效
    杀真菌剂取代尿毒症

    公开(公告)号:US3920831A

    公开(公告)日:1975-11-18

    申请号:US39965373

    申请日:1973-09-21

    申请人: BAYER AG

    IPC分类号: C07C335/28 A01N9/12

    CPC分类号: C07C335/28

    摘要: Ureidophenyl thioureas of the formula:

    in which EACH INDEPENDENTLY STANDS FOR A HALOGEN ATOM, ALKYL WITH 1-4 CARBON ATOMS OR ALKOXY WITH 1-4 CARBON ATOMS, N STANDS FOR 0, 1 OR 2, R stands for alkyl with 1-12 carbon atoms, R'' and R'''' each stands independently for a hydrogen atom or alkyl with 1-4 carbon atoms, and R'''''' stands for a hydrogen atom, alkyl with 1 or 2 carbon atoms (which may carry at least one substituent selected from halogen, cyano, alkoxy with up to 4 carbon atoms and alkoxycarbonyl with up to 5 carbon atoms), alkyl with 3 to 18 carbon atoms (which carries at least one substituent selected from halogen, cyano, alkoxy with up to 4 carbon atoms and alkoxycarbonyl with up to 5 carbon atoms), cycloalkyl with 5 to 8 ring carbon atoms, aralkyl (the aryl moiety of which may carry at least one substituent selected from halogen, lower alkyl and lower alkoxy), phenyl (which may carry at least one substituent selected from halogen, lower alkyl and lower alkoxy), acyl with up to 18 carbon atoms (which may be substituted by halogen and/or lower alkyl), aroyl (which may carry at least one substituent selected from halogen, lower alkyl and lower alkoxy), alkylsulfonyl with up to 18 carbon atoms, arylsulfonyl (which may carry at least one substituent selected from halogen, amino, lower alkyl and lower alkoxy) or dialkylamino with up to 4 carbon atoms, possess fungicidal properties.