公开(公告)号：US20090235467A1

公开(公告)日：2009-09-24

申请号：US12341453

申请日：2008-12-22

Applicant: Laurent VIDAL ,  Eric Metais ,  Aziz Fadli ,  Alan Katritzky

Inventor： Laurent VIDAL ,  Eric Metais ,  Aziz Fadli ,  Alan Katritzky

IPC: A61K8/49 ,  C07D221/00 ,  A61Q5/10

CPC classification number: C07D471/04 ,  A61K8/4926 ,  A61K2800/88 ,  A61Q5/10

Abstract: A new class of chemical entities chosen from aminoindolizines of formula (I), acid addition salts thereof, and solvates thereof: their use for dyeing keratin fibers, including human keratin fibers such as the hair; dyeing compositions comprising such chemical entities; and to kits containing compositions comprising those chemical entities.

Abstract translation: 一类选自式（I）的氨基吲哚啉，其酸加成盐及其溶剂化物的化学物质：它们用于染色角蛋白纤维，包括人角蛋白纤维如毛发; 包含这些化学实体的染色组合物; 以及含有包含那些化学实体的组合物的试剂盒。

公开(公告)号：US08034124B2

公开(公告)日：2011-10-11

申请号：US12666123

申请日：2008-06-19

Applicant: Aziz Fadli ,  Eric Metais

Inventor： Aziz Fadli ,  Eric Metais

IPC: A61Q5/10 ,  C07D231/00

CPC classification number: C07D487/04 ,  C07D213/77 ,  C07D231/04 ,  C07D231/44 ,  C07D233/88 ,  C07D235/30 ,  C07D277/04 ,  C07D277/50 ,  C07D277/82 ,  C07D401/12 ,  C07D417/12

Abstract: The subject of the present invention is azo derivatives containing a pyrazolinone unit having the following formula (I), their mesomeric forms, their addition salts with an acid and their solvates and their use for dyeing keratin fibers. The subject of the invention is also a composition for dying keratin fibers comprising at least one azo derivative containing a pyrazolinone unit of formula (I) as direct dye, and the method for dyeing keratin fibers using this composition. The present invention makes it possible in particular to obtain chromatic colors that are resistant to the various attacks to which the hair may be subjected, in particular to shampoos and to light.

Abstract translation: 本发明的主题是含有具有下式（I）的吡唑啉酮单元，它们的内消旋形式，它们与酸的加成盐及其溶剂化物的偶氮衍生物及其用于染色角蛋白纤维的用途。 本发明的主题还是一种用于染色角蛋白纤维的组合物，其包含至少一种含有式（I）的吡唑啉酮单元作为直接染料的偶氮衍生物，以及使用该组合物染色角蛋白纤维的方法。 本发明特别是可以获得耐受头发可能经受的各种攻击的彩色，特别是洗发剂和光。

公开(公告)号：US20090044348A1

公开(公告)日：2009-02-19

申请号：US12213441

申请日：2008-06-19

Applicant: Aziz Fadli ,  Eric Metais

Inventor： Aziz Fadli ,  Eric Metais

IPC: A61K8/49 ,  C07D231/08 ,  A61Q5/00 ,  C07D487/02

CPC classification number: C07D231/48 ,  A61K8/494 ,  A61Q5/06 ,  A61Q5/065 ,  C07D231/54 ,  C07D231/56 ,  C07D401/12 ,  C07D487/04

Abstract: The present disclosure relates to a composition for coloring keratin fibers which comprises, in an appropriate dyeing medium, at least one compound chosen from leuco compounds of formula (I), azomethine dyes with a pyrazolinone unit of formula (II), their mesomeric forms, acid addition salts and solvates thereof: and dyeing methods and multicompartment devices for use thereof.

公开(公告)号：US07776107B2

公开(公告)日：2010-08-17

申请号：US12341453

申请日：2008-12-22

Applicant: Laurent Vidal ,  Eric Metais ,  Aziz Fadli ,  Alan Katritzky

Inventor： Laurent Vidal ,  Eric Metais ,  Aziz Fadli ,  Alan Katritzky

IPC: A61Q5/10 ,  C07D221/02

CPC classification number: C07D471/04 ,  A61K8/4926 ,  A61K2800/88 ,  A61Q5/10

Abstract: A new class of chemical entities chosen from aminoindolizines of formula (I), acid addition salts thereof, and solvates thereof: their use for dyeing keratin fibers, including human keratin fibers such as the hair; dyeing compositions comprising such chemical entities; and to kits containing compositions comprising those chemical entities.

Abstract translation: 一类选自式（I）的氨基吲哚啉，其酸加成盐及其溶剂化物的化学物质：它们用于染色角蛋白纤维，包括人角蛋白纤维如毛发; 包含这些化学实体的染色组合物; 以及含有包含这些化学实体的组合物的试剂盒。

公开(公告)号：US07582123B2

公开(公告)日：2009-09-01

申请号：US12213441

申请日：2008-06-19

Applicant: Aziz Fadli ,  Eric Metais

Inventor： Aziz Fadli ,  Eric Metais

IPC: A61Q5/10 ,  C07D231/44

CPC classification number: C07D231/48 ,  A61K8/494 ,  A61Q5/06 ,  A61Q5/065 ,  C07D231/54 ,  C07D231/56 ,  C07D401/12 ,  C07D487/04

Abstract: The present disclosure relates to a composition for coloring keratin fibers which comprises, in an appropriate dyeing medium, at least one compound chosen from leuco compounds of formula (I), azomethine dyes with a pyrazolinone unit of formula (II), their mesomeric forms, acid addition salts and solvates thereof: and dyeing methods and multicompartment devices for use thereof.

Abstract translation: 本公开涉及一种着色角蛋白纤维的组合物，其在合适的染色介质中包含至少一种选自式（I）的无色化合物，偶氮甲碱染料与式（II）的吡唑啉酮单元，其介体形式， 酸加成盐和溶剂合物：和用于其的染色方法和多室装置。

公开(公告)号：US20100269269A1

公开(公告)日：2010-10-28

申请号：US12666123

申请日：2008-06-19

Applicant: Aziz Fadli ,  Eric Metais

Inventor： Aziz Fadli ,  Eric Metais

IPC: A61K8/40 ,  C09B39/00 ,  A61Q5/10

CPC classification number: C07D487/04 ,  C07D213/77 ,  C07D231/04 ,  C07D231/44 ,  C07D233/88 ,  C07D235/30 ,  C07D277/04 ,  C07D277/50 ,  C07D277/82 ,  C07D401/12 ,  C07D417/12

Abstract: The subject of the present invention is azo derivatives containing a pyrazolinone unit having the following formula (I), their mesomeric forms, their addition salts with an acid and their solvates and their use for dyeing keratin fibers. The subject of the invention is also a composition for dying keratin fibers comprising at least one azo derivative containing a pyrazolinone unit of formula (I) as direct dye, and the method for dyeing keratin fibers using this composition. The present invention makes it possible in particular to obtain chromatic colours that are resistant to the various attacks to which the hair may be subjected, in particular to shampoos and to light.

Abstract translation: 本发明的主题是含有具有下式（I）的吡唑啉酮单元，它们的内消旋形式，它们与酸的加成盐及其溶剂化物的偶氮衍生物及其用于染色角蛋白纤维的用途。 本发明的主题还是一种用于染色角蛋白纤维的组合物，其包含至少一种含有式（I）的吡唑啉酮单元作为直接染料的偶氮衍生物，以及使用该组合物染色角蛋白纤维的方法。 本发明特别是可以获得耐受头发可能经受的各种攻击的彩色，特别是洗发剂和光。

公开(公告)号：US20140352081A1

公开(公告)日：2014-12-04

申请号：US14345103

申请日：2012-09-13

Applicant: Aziz Fadli

Inventor： Aziz Fadli

IPC: A61K8/41 ,  C09B69/00 ,  C07C217/84 ,  C07D295/135 ,  A61Q5/10 ,  A61K8/49

CPC classification number: A61K8/415 ,  A61K8/41 ,  A61K8/49 ,  A61K8/4913 ,  A61K8/4926 ,  A61K8/494 ,  A61K8/4946 ,  A61K2800/10 ,  A61K2800/4324 ,  A61K2800/88 ,  A61Q5/10 ,  C07C215/80 ,  C07C217/08 ,  C07C217/84 ,  C07D295/088 ,  C07D295/135 ,  C09B69/001

Abstract: The present invention relates to a para-aminophenol compound of formula (I) the addition salts thereof with an acid and the solvates thereof, dye composition comprising the latter and a dyeing process.

Abstract translation: 本发明涉及式（I）的对氨基苯酚化合物，其与酸及其溶剂化物的加成盐，包含其的染料组合物和染色方法。

公开(公告)号：US08623100B2

公开(公告)日：2014-01-07

申请号：US13994288

申请日：2011-12-14

Applicant: Aziz Fadli ,  Fatima Makhlouf

Inventor： Aziz Fadli ,  Fatima Makhlouf

IPC: A61Q5/10 ,  C07D209/04

CPC classification number: A61K8/492 ,  A61K8/4946 ,  A61K2800/882 ,  A61Q5/10 ,  C07D209/40 ,  C07D401/12 ,  C07D403/12 ,  C07D413/12

Abstract: The invention relates to 4-aminoindole derivatives of formula (I), and the addition salts thereof, mesomers thereof, isomers thereof and solvates thereof: and to their use for the oxidation dyeing of keratin fibers, and in particular of human keratin fibers such as the hair. The present invention makes it possible to achieve dark shades, natural shades and dark natural shades. The present invention also makes it possible to obtain powerful, chromatic, aesthetic, sparingly selective coloration of keratin fibers in varied shades, which is resistant to the various attacking factors to which the hair may be subjected. In particular, when the 4-aminoindole derivatives are combined with one or more heterocyclic oxidation bases, they make it possible to obtain a wide range of colors and coloration of keratin fibers that shows good chromaticity and good selectivity.

Abstract translation: 本发明涉及式（I）的4-氨基吲哚衍生物及其加成盐，其介体，其异构体和溶剂化物，以及它们用于角蛋白纤维，特别是人角蛋白纤维如 头发。 本发明可以实现暗色调，天然色调和暗色的天然色调。 本发明还使得可以以各种色调获得强大的，有色的，美观的，谨慎的选择性着色的角蛋白纤维，其耐受头发可能经受的各种攻击因素。 特别地，当4-氨基吲哚衍生物与一个或多个杂环氧化碱组合时，它们可以获得显示良好色度和良好选择性的角蛋白纤维的宽范围颜色和着色。

公开(公告)号：US20130263390A1

公开(公告)日：2013-10-10

申请号：US13994288

申请日：2011-12-14

Applicant: Aziz Fadli ,  Fatima Makhlouf

Inventor： Aziz Fadli ,  Fatima Makhlouf

IPC: A61K8/49 ,  A61Q5/10

CPC classification number: A61K8/492 ,  A61K8/4946 ,  A61K2800/882 ,  A61Q5/10 ,  C07D209/40 ,  C07D401/12 ,  C07D403/12 ,  C07D413/12

Abstract: The invention relates to 4-aminoindole derivatives of formula (I), and the addition salts thereof, mesomers thereof, isomers thereof and solvates thereof: and to their use for the oxidation dyeing of keratin fibres, and in particular of human keratin fibres such as the hair. The present invention makes it possible to achieve dark shades, natural shades and dark natural shades. The present invention also makes it possible to obtain powerful, chromatic, aesthetic, sparingly selective coloration of keratin fibres in varied shades, which is resistant to the various attacking factors to which the hair may be subjected. In particular, when the 4-aminoindole derivatives are combined with one or more heterocyclic oxidation bases, they make it possible to obtain a wide range of colours and coloration of keratin fibres that shows good chromaticity and good selectivity.

Abstract translation: 本发明涉及式（I）的4-氨基吲哚衍生物及其加成盐，其介体，其异构体和溶剂化物，以及它们用于角蛋白纤维，特别是人角蛋白纤维如 头发。 本发明可以实现暗色调，天然色调和暗色的天然色调。 本发明还使得可以以各种色调获得强大的，有色的，美观的，谨慎选择性的角蛋白纤维的着色，其耐受头发可能经受的各种攻击因素。 特别地，当4-氨基吲哚衍生物与一个或多个杂环氧化碱组合时，它们可以获得显示良好色度和良好选择性的角蛋白纤维的宽范围颜色和着色。

公开(公告)号：US20120278997A1

公开(公告)日：2012-11-08

申请号：US13389832

申请日：2010-08-11

Applicant: Anne-Marie Couroux ,  Aziz Fadli

Inventor： Anne-Marie Couroux ,  Aziz Fadli

IPC: A61K8/49 ,  A61Q5/10

CPC classification number: A61Q5/10 ,  A61K8/49 ,  A61K8/4913 ,  A61K8/494 ,  A61K8/4946 ,  A61K2800/88

Abstract: The subject of the present invention is dye composition for keratin fibres, comprising, in suitable dyeing medium, a coupler of formula (I) or addition salts thereof with an acid a particular cationic or noncationic aminopyrazolopyridine derivative. The composition of the present invention makes it possible in particular to obtain a colouring with varied, intense and/or chromatic, aesthetic and relatively nonselective shades which are highly resistant to the various attacks to which the hair may be subjected.

Abstract translation: 本发明的主题是用于角蛋白纤维的染料组合物，其在合适的染色介质中包含式（I）的成色剂或其加成盐与酸，特别是阳离子或非阳离子型氨基吡唑并吡啶衍生物。 本发明的组合物特别可以获得对于头发可能经受的各种攻击具有高度抗性的变化，强烈和/或有色，美观和相对非选择性色调的着色。