-
1.1,6- DIAZABICYCLO [3,2,1] OCTAN-7-ONE DERIVATIVES AND THEIR USE IN THE TREATMENT OF BACTERIAL INFECTIONS 审中-公开
标题翻译: 1,6-二氮杂双环[3,2,1] OCT-7-ONE衍生物及其在治疗细菌感染中的用途公开(公告)号:US20150203503A1
公开(公告)日:2015-07-23
申请号:US14365064
申请日:2013-04-19
申请人: Vijaykumar Jagdishwar Patil , Ravikumar Tadiparthi , Bharat Dond , Amol Kale , Loganathan Velupillai , Deepak Dekhane , Satish Shrimant Birajdar , Mohammad Usman Shaikh , Sushilkumar Maurya , Piyush Ambalal Patel , Prasad Dixit , Mangesh Pawar , Mahesh Vithalbhai Patel , Sachin Bhagwat
发明人: Vijaykumar Jagdishwar Patil , Ravikumar Tadiparthi , Bharat Dond , Amol Kale , Loganathan Velupillai , Deepak Dekhane , Satish Shrimant Birajdar , Mohammad Usman Shaikh , Sushilkumar Maurya , Piyush Ambalal Patel , Prasad Dixit , Mangesh Pawar , Mahesh Vithalbhai Patel , Sachin Bhagwat
IPC分类号: C07D487/08 , A61K45/06 , A61K31/55 , A61K31/496 , A61K31/439 , A61K31/4545
CPC分类号: C07D471/08 , A61K31/407 , A61K31/439 , A61K31/4545 , A61K31/496 , A61K31/546 , A61K31/55 , A61K45/06 , A61P31/04 , C07C211/63 , C07D487/08
摘要: Compounds of Formula (I), their preparation and use in preventing or treating bacterial infections are disclosed.
摘要翻译: 公开了式(I)化合物及其制备和用于预防或治疗细菌感染的方法。
-
2.1,6-Diazabicyclo [3,2,1] octan-7-one derivatives and their use in the treatment of bacterial infections 有权
标题翻译: 1,6-二氮杂双环[3,2,1]辛-7-酮衍生物及其在细菌感染治疗中的应用公开(公告)号:US20140088068A1
公开(公告)日:2014-03-27
申请号:US14113980
申请日:2012-08-24
申请人: Sachin Bhagwat , Prasad Keshav Deshpande , Satish Bhawsar , Vijaykumar Jagdishwar Patil , Ravikumar Tadiparthi , Shivaji Sampatrao Pawar , Sunil Bhaginath Jadhav , Sanjay Kisan Dabhade , Vikas Vitthalrao Deshmukh , Bharat Dond , Satish Birajdar , Mohammad Usman Shaikh , Deepak Dekhane , Piyush Ambalal Patel
发明人: Sachin Bhagwat , Prasad Keshav Deshpande , Satish Bhawsar , Vijaykumar Jagdishwar Patil , Ravikumar Tadiparthi , Shivaji Sampatrao Pawar , Sunil Bhaginath Jadhav , Sanjay Kisan Dabhade , Vikas Vitthalrao Deshmukh , Bharat Dond , Satish Birajdar , Mohammad Usman Shaikh , Deepak Dekhane , Piyush Ambalal Patel
IPC分类号: C07D471/08 , A61K31/43 , A61K31/424 , A61K31/496 , A61K31/439 , C07D519/00 , A61K31/5383 , A61K31/5377 , A61K31/4545 , A61K31/546
CPC分类号: C07D471/08 , A61K31/424 , A61K31/43 , A61K31/431 , A61K31/439 , A61K31/4545 , A61K31/46 , A61K31/496 , A61K31/5377 , A61K31/5383 , A61K31/546 , A61K45/06 , C07D498/04 , C07D519/00 , A61K2300/00
摘要: Compounds of Formula (I), their preparation and use in preventing or treating bacterial infections are disclosed.
摘要翻译: 公开了式(I)化合物及其制备和用于预防或治疗细菌感染的方法。
-
公开(公告)号:US08288416B2
公开(公告)日:2012-10-16
申请号:US12311243
申请日:2007-09-22
申请人: Vijaykumar Jadgishwar Patil , Mahesh Vithalbhai Patel , Bharat Kalidas Trivedi , Deepak Vijaykumar Dekhane , Mohammad Usman Shaikh , Yati Chugh , Rajesh Prabhakar Chavan , Mohammad Alam Jafri
发明人: Vijaykumar Jadgishwar Patil , Mahesh Vithalbhai Patel , Bharat Kalidas Trivedi , Deepak Vijaykumar Dekhane , Mohammad Usman Shaikh , Yati Chugh , Rajesh Prabhakar Chavan , Mohammad Alam Jafri
IPC分类号: A61K31/445 , C07D413/14
CPC分类号: C07D413/10 , C07F9/65583
摘要: The present invention relates to oxazolidinones of Formula I and pharmaceutically acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof. The invention also relates to processes for the preparation of the compound of Formula I and pharmaceutically acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof, and to pharmaceutical compositions containing the compounds of Formula I and pharmaceutically acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof and to methods for treating or preventing microbial infections using the compounds of Formula I and pharmaceutically acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof.
摘要翻译: 本发明涉及式I的恶唑烷酮及其药学上可接受的盐,药学上可接受的溶剂化物或其多晶型物。 本发明还涉及制备式I化合物及其药学上可接受的盐,药学上可接受的溶剂合物或多晶型物的方法,以及含有式I化合物及其药学上可接受的盐,药学上可接受的溶剂化物或多晶型物的药物组合物,以及 使用式I化合物及其药学上可接受的盐,药学上可接受的溶剂合物或多晶型物治疗或预防微生物感染的方法。
-
4.1,6-diazabicyclo [3,2,1] octan-7-one derivatives and their use in the treatment of bacterial infections 有权
标题翻译: 1,6-二氮杂双环[3,2,1]辛-7-酮衍生物及其在细菌感染治疗中的应用公开(公告)号:US09006230B2
公开(公告)日:2015-04-14
申请号:US14113980
申请日:2012-08-24
申请人: Sachin Bhagwat , Prasad Keshav Deshpande , Satish Bhawsar , Vijaykumar Jagdishwar Patil , Ravikumar Tadiparthi , Shivaji Sampatrao Pawar , Sunil Bhaginath Jadhav , Sanjay Kisan Dabhade , Vikas Vitthalrao Deshmukh , Bharat Dond , Satish Birajdar , Mohammad Usman Shaikh , Deepak Dekhane , Piyush Ambalal Patel
发明人: Sachin Bhagwat , Prasad Keshav Deshpande , Satish Bhawsar , Vijaykumar Jagdishwar Patil , Ravikumar Tadiparthi , Shivaji Sampatrao Pawar , Sunil Bhaginath Jadhav , Sanjay Kisan Dabhade , Vikas Vitthalrao Deshmukh , Bharat Dond , Satish Birajdar , Mohammad Usman Shaikh , Deepak Dekhane , Piyush Ambalal Patel
IPC分类号: A61K31/00 , C07D233/10 , C07D243/00 , C07D471/08 , A61K31/424 , A61K31/43 , A61K31/439 , A61K31/4545 , A61K31/496 , A61K31/5377 , A61K31/5383 , A61K31/546 , C07D519/00 , C07D498/04
CPC分类号: C07D471/08 , A61K31/424 , A61K31/43 , A61K31/431 , A61K31/439 , A61K31/4545 , A61K31/46 , A61K31/496 , A61K31/5377 , A61K31/5383 , A61K31/546 , A61K45/06 , C07D498/04 , C07D519/00 , A61K2300/00
摘要: Compounds of Formula (I), their preparation and use in preventing or treating bacterial infections are disclosed.
摘要翻译: 公开了式(I)化合物及其制备和用于预防或治疗细菌感染的方法。
-
公开(公告)号:US09127004B2
公开(公告)日:2015-09-08
申请号:US14298182
申请日:2014-06-06
申请人: Sachin Bhagwat , Prasad Keshav Deshpande , Satish Bhawsar , Vijaykumar Jagdishwar Patil , Ravikumar Tadiparthi , Shivaji Sampatrao Pawar , Sunil Bhaginath Jadhav , Sanjay Kisan Dabhade , Vikas Vitthalrao Deshmukh , Bharat Dhond , Satish Birajdar , Mohammad Usman Shaikh , Deepak Dekhane , Piyush Ambalal Patel
发明人: Sachin Bhagwat , Prasad Keshav Deshpande , Satish Bhawsar , Vijaykumar Jagdishwar Patil , Ravikumar Tadiparthi , Shivaji Sampatrao Pawar , Sunil Bhaginath Jadhav , Sanjay Kisan Dabhade , Vikas Vitthalrao Deshmukh , Bharat Dhond , Satish Birajdar , Mohammad Usman Shaikh , Deepak Dekhane , Piyush Ambalal Patel
IPC分类号: C07D487/00 , A61K31/44 , C07D471/08 , A61K31/424 , A61K31/43 , A61K31/439 , A61K31/4545 , A61K31/496 , A61K31/5377 , A61K31/5383 , A61K31/546 , C07D519/00 , C07D498/04
CPC分类号: C07D471/08 , A61K31/424 , A61K31/43 , A61K31/431 , A61K31/439 , A61K31/4545 , A61K31/46 , A61K31/496 , A61K31/5377 , A61K31/5383 , A61K31/546 , A61K45/06 , C07D498/04 , C07D519/00 , A61K2300/00
摘要: Compounds of Formula (I), their preparation and use in preventing or treating bacterial infections are disclosed.
摘要翻译: 公开了式(I)化合物及其制备和用于预防或治疗细菌感染的方法。
-
公开(公告)号:US20140288064A1
公开(公告)日:2014-09-25
申请号:US14298182
申请日:2014-06-06
申请人: Sachin BHAGWAT , Prasad Keshav DESHPANDE , Satish BHAWSAR , Vijaykumar Jagdishwar PATIL , Ravikumar TADIPARTHI , Shivaji Sampatrao PAWAR , Sunil Bhaginath JADHAV , Sanjay Kisan DABHADE , Vikas Vitthalrao DESHMUKH , Bharat DHOND , Satish BIRAJDAR , Mohammad Usman SHAIKH , Deepak DEKHANE , Piyush Ambalal PATEL
发明人: Sachin BHAGWAT , Prasad Keshav DESHPANDE , Satish BHAWSAR , Vijaykumar Jagdishwar PATIL , Ravikumar TADIPARTHI , Shivaji Sampatrao PAWAR , Sunil Bhaginath JADHAV , Sanjay Kisan DABHADE , Vikas Vitthalrao DESHMUKH , Bharat DHOND , Satish BIRAJDAR , Mohammad Usman SHAIKH , Deepak DEKHANE , Piyush Ambalal PATEL
IPC分类号: C07D471/08 , C07D498/04
CPC分类号: C07D471/08 , A61K31/424 , A61K31/43 , A61K31/431 , A61K31/439 , A61K31/4545 , A61K31/46 , A61K31/496 , A61K31/5377 , A61K31/5383 , A61K31/546 , A61K45/06 , C07D498/04 , C07D519/00 , A61K2300/00
摘要: Compounds of Formula (I), their preparation and use in preventing or treating bacterial infections are disclosed.
摘要翻译: 公开了式(I)化合物及其制备和用于预防或治疗细菌感染的方法。
-
公开(公告)号:US20100120721A1
公开(公告)日:2010-05-13
申请号:US12311243
申请日:2007-09-22
申请人: Vijaykumar Jadgishwar Patil , Mahesh Vithalbhai Patel , Bharat Kalidas Trivedi , Deepak Vijaykumar Dekhane , Mohammad Usman Shaikh , Yati Chugh , Rajesh Prabhakar Chavan , Mohammad Alam Jafri
发明人: Vijaykumar Jadgishwar Patil , Mahesh Vithalbhai Patel , Bharat Kalidas Trivedi , Deepak Vijaykumar Dekhane , Mohammad Usman Shaikh , Yati Chugh , Rajesh Prabhakar Chavan , Mohammad Alam Jafri
IPC分类号: A61K31/454 , C07F9/117 , C07D413/14 , C07D413/10 , A61K31/661 , A61P31/04 , A61P31/00
CPC分类号: C07D413/10 , C07F9/65583
摘要: The present invention relates to oxazolidinones of Formula I and pharmaceutically acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof. The invention also relates to processes for the preparation of the compound of Formula I and pharmaceutically acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof, and to pharmaceutical compositions containing the compounds of Formula I and pharmaceutically acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof and to methods for treating or preventing microbial infections using the compounds of Formula I and pharmaceutically acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof.
摘要翻译: 本发明涉及式I的恶唑烷酮及其药学上可接受的盐,药学上可接受的溶剂化物或其多晶型物。 本发明还涉及制备式I化合物及其药学上可接受的盐,药学上可接受的溶剂合物或多晶型物的方法,以及含有式I化合物及其药学上可接受的盐,药学上可接受的溶剂化物或多晶型物的药物组合物,以及 使用式I化合物及其药学上可接受的盐,药学上可接受的溶剂合物或多晶型物治疗或预防微生物感染的方法。
-
-
-
-
-
-