公开(公告)号：US3740401A

公开(公告)日：1973-06-19

申请号：US3740401D

申请日：1970-11-18

申请人： BOEHRINGER SOHN INGELHEIM

发明人： KUMMER W ,  STOCKHAUS K ,  STAHLE H ,  KOPPE H

IPC分类号： C07D233/50 ,  C07D49/34 ,  C07D57/48

CPC分类号： C07D233/50

摘要： COMPOUND OF THE FORMULA

2-((CYCLOPENTYL)-N(-Y)-)-2-IMIDAZOLINE, OR 2-((CYCLO-

HEPTYL)-N(-Z)-)-2-IMIDAZOLINE

WHEREIN 1 IS 2,6-DICHLORO-PHENYL, 2-CHLORO-L-METHY6-PHENYL, 2CHLORO-4-METHYL-PHENYL, 2-METHYL-4-CHLORO-PHENYL,2CHLORO-PHENYL, 2,4-DICHLORO-PHENYL, 2-METHYL-PHENYL. 2,6-DIETHYL-PHENYL, 4-BROMO-PHENYL, 2,6- DICHLORO-4BROMO-PHENYL, 4-CYANO-PHENYL, 4-FLUORO-PHENYL OR 2-TRI FLUOROMETHYL-PHENYL, 2-METHOXY-4-CHLORO-PHENYL OR 2CHLORO-3-METHYL-PHENYL, AND Z IS

(2-CL,6-R7-PHENYL)-

WHERE R7 IS CHLORINE OR METHYL, AND THEIR NON-TOXIC, PHARMACOLOGICALLY ACCEPTABLE ACID ADDITION SALTS, THE COMPOUNDS AS WELL AS THEIR SALTS ARE USEFUL AS ANALGESICS.