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1.Process for the preparation of temsirolimus and its intermediates 失效
Title translation: 制备替西罗莫司及其中间体的方法公开(公告)号:US08524893B2
公开(公告)日:2013-09-03
申请号:US13016235
申请日:2011-01-28
Applicant: Nitin Gupta , Vishal Handa , Abir Kumar Pal , Hemant Kumar Singh , Saswata Lahiri , Sushil Kumar Dubey
Inventor: Nitin Gupta , Vishal Handa , Abir Kumar Pal , Hemant Kumar Singh , Saswata Lahiri , Sushil Kumar Dubey
IPC: C07D498/00
CPC classification number: C07D498/18 , C07D319/06
Abstract: Novel intermediates, process for their preparation and their use in the preparation of therapeutically effective antineoplastic agents, in particular Temsirolimus of formula (I).
Abstract translation: 新型中间体,其制备方法及其在制备治疗有效的抗肿瘤药物中的用途,特别是式(I)的替西罗莫司。
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2.PROCESS FOR THE PREPARATION OF TEMSIROLIMUS AND ITS INTERMEDIATES 失效
Title translation: 制备纤维素及其中间体的方法公开(公告)号:US20110184167A1
公开(公告)日:2011-07-28
申请号:US13016235
申请日:2011-01-28
Applicant: Nitin Gupta , Vishal Handa , Abir Kumar Pal , Hemant Kumar Singh , Saswata Lahiri , Sushil Kumar Dubey
Inventor: Nitin Gupta , Vishal Handa , Abir Kumar Pal , Hemant Kumar Singh , Saswata Lahiri , Sushil Kumar Dubey
IPC: C07D498/12 , C07D407/12
CPC classification number: C07D498/18 , C07D319/06
Abstract: Novel intermediates, process for their preparation and their use in the preparation of therapeutically effective antineoplastic agents, in particular Temsirolimus of formula (I).
Abstract translation: 新型中间体,其制备方法及其在制备治疗有效的抗肿瘤药物中的用途,特别是式(I)的替西罗莫司。
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