公开(公告)号：US07585891B2

公开(公告)日：2009-09-08

申请号：US10554347

申请日：2004-04-28

申请人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  John W. Lyga ,  Matthew P. Whiteside ,  Frank J. Zawacki

发明人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  John W. Lyga ,  Matthew P. Whiteside ,  Frank J. Zawacki

IPC分类号： A61K31/343 ,  A61K31/353 ,  C07D307/83 ,  C07D311/04

CPC分类号： A01N43/30 ,  A01N43/32 ,  A01N43/40 ,  A01N43/60 ,  A01N47/16 ,  C07D211/22 ,  C07D307/79 ,  C07D307/83 ,  C07D311/04 ,  C07D401/04 ,  C07D495/10

摘要： Certain novel (dihalopropenyl)phenylalkyl substituted benzodioxolane and benzodioxane derivatives have provided unexpected insecticidal activity. These compounds are represented by formula I: where R through R10, inclusively, x, A, B, y, D, E, G and M are fully described herein. Preferred compounds of the present invention are those wherein the benzofused ring moiety is attached to the remainder of the molecule at the positions designated as 1- or 2-. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 某些新的（二卤代丙烯基）苯基烷基取代的苯并二氧杂环戊烷和苯并二恶烷衍生物提供了意想不到的杀虫活性。 这些化合物由式I表示：其中R至R10，包括x，A，B，y，D，E，G和M在本文中完整描述。 本发明优选的化合物是其中苯并稠环部分在指定为1-或2-的位置连接到分子的其余部分的化合物。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US07576224B2

公开(公告)日：2009-08-18

申请号：US11292023

申请日：2005-12-01

申请人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  David M. Roush ,  Stephen F. Donovan ,  Frank J. Zawacki ,  Walter H. Yeager ,  John W. Lyga ,  Daniel H. Cohen

发明人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  David M. Roush ,  Stephen F. Donovan ,  Frank J. Zawacki ,  Walter H. Yeager ,  John W. Lyga ,  Daniel H. Cohen

IPC分类号： C07D307/80 ,  C07D495/10

CPC分类号： A01N43/30 ,  A01N43/32 ,  A01N43/40 ,  A01N43/60 ,  A01N47/16 ,  C07D211/22 ,  C07D307/79 ,  C07D307/83 ,  C07D311/04 ,  C07D401/04 ,  C07D495/10

摘要： Insecticidal (dihalopropenyl) phenylalkyl substituted dihydrobenzofuran and dihydrobenzopyran derivatives of Formula I are disclosed. These compounds provide unexpected insecticidal activity across a spectrum of insect pests combined with desirable physical properties including improved photostability. wherein x and y are integers independently selected from 0 or 1; and B is a bridging group *—(CR16R17)q—(CR18R19)r—(CR20R21)s-Lt-(CR22R23)u—(CR24R25)v—(CR26R27)w—, where the asterisk denotes attachment at A; and q, r, s, u, v and w are integers independently selected from 0, 1 and 2; and t is an integer selected from 0 and 1. A, D, E, G, M, R through R11, and R16 through R27, inclusively, are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I and methods of controlling insects by applying said compositions to a locus where insects are present or are expected to be present are also disclosed.

摘要翻译： 公开了杀虫（二卤代丙烯基）苯基烷基取代的二氢苯并呋喃和式I的二氢苯并吡喃衍生物。 这些化合物在一系列昆虫害虫中提供了意想不到的杀虫活性，并结合所需的物理性质，包括改善的光稳定性。 其中x和y是独立地选自0或1的整数; * - （CR16R17）q-（CR18R19）r-（CR20R21）s-Lt-（CR22R23），而B是桥接基团<？in-line-formula description =“In-line Formulas”end =“lead” u-（CR24R25）v-（CR26R27）w - ，<？在线公式描述=“在线公式”end =“tail”？>其中星号表示在A附近; q，r，s，u，v和w是独立地选自0,1和2的整数; 并且t是选自0和1的整数。本文充分描述了A，D，E，G，M，R至R 11和R 16至R 27。 此外，还公开了包含杀虫有效量的至少一种式I化合物的组合物和通过将所述组合物施用于存在昆虫或预期存在的场所来控制昆虫的方法。

公开(公告)号：US07208450B2

公开(公告)日：2007-04-24

申请号：US10510331

申请日：2004-04-28

申请人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  John W. Lyga ,  Matthew P. Whiteside

发明人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  John W. Lyga ,  Matthew P. Whiteside

IPC分类号： A01N43/76 ,  A01N43/78 ,  C07D263/54 ,  C07D277/62

CPC分类号： A01N43/30 ,  A01N43/32 ,  A01N43/40 ,  A01N43/60 ,  A01N47/16 ,  C07D211/22 ,  C07D307/79 ,  C07D307/83 ,  C07D311/04 ,  C07D401/04 ,  C07D495/10

摘要： Certain novel (dihalopropenyl)phenylalkyl substituted benzoxazole and benzothiazole derivatives have unexpected insecticidal activity. These compounds are represented by formula (I): where R through R11, inclusively. x, A, B, y, D, E and G are fully described herein. Preferred compounds of the present invention are those wherein the benzo-fused ring moiety is attached to the remainder of the molecule at the positions designated as (5) or (6) and where R11 is either C1–C3 alkyl or halo C1–C3 alkyl. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula (I), and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 某些新的（二卤代丙烯基）苯基烷基取代的苯并恶唑和苯并噻唑衍生物具有出人意料的杀虫活性。 这些化合物由式（I）表示：其中R 1至R 11包括。 这里完整地描述了x，A，B，y，D，E和G。 本发明优选的化合物是其中苯并稠环部分在（5）或（6）表示的位置连接到分子的其余部分，其中R 11是C < C 1 -C 3烷基或卤素C 1 -C 3烷基。 此外，还公开了包含杀虫有效量的至少一种式（I）化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US06987194B2

公开(公告)日：2006-01-17

申请号：US10832624

申请日：2004-04-27

申请人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  David M. Roush ,  Stephen F. Donovan ,  Frank J. Zawacki ,  Walter H. Yeager ,  John W. Lyga ,  Daniel H. Cohen

发明人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  David M. Roush ,  Stephen F. Donovan ,  Frank J. Zawacki ,  Walter H. Yeager ,  John W. Lyga ,  Daniel H. Cohen

IPC分类号： C07D307/83 ,  C07D311/04 ,  A61K31/343 ,  A61K31/353

CPC分类号： A01N43/30 ,  A01N43/32 ,  A01N43/40 ,  A01N43/60 ,  A01N47/16 ,  C07D211/22 ,  C07D307/79 ,  C07D307/83 ,  C07D311/04 ,  C07D401/04 ,  C07D495/10

摘要： Insecticidal (dihalopropenyl) phenylalkyl substituted dihydrobenzofuran and dihydrobenzopyran derivatives of Formula I are disclosed. These compounds provide unexpected insecticidal activity across a spectrum of insect pests combined with desirable physical properties including improved photostability. wherein x and y are integers independently selected from 0 or 1; and B is a bridging group *—(CR16R17)q—(CR18R19)r—(CR20R21)s—Lt—(CR22R23)u—(CR24R25)v—(CR26R27)w—, where the asterisk denotes attachment at A; and q, r, s, u, v and w are integers independently selected from 0, 1 and 2; and t is an integer selected from 0 and 1. A, D, E, G, M, R through R11, and R16 through R27, inclusively, are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I and methods of controlling insects by applying said compositions to a locus where insects are present or are expected to be present are also disclosed.

摘要翻译： 公开了杀虫（二卤代丙烯基）苯基烷基取代的二氢苯并呋喃和式I的二氢苯并吡喃衍生物。 这些化合物在一系列昆虫害虫中提供了意想不到的杀虫活性，并结合所需的物理性质，包括改善的光稳定性。 其中x和y是独立地选自0或1的整数; 并且B是桥接基团<？in-line-formula description =“In-line Formulas”end =“lead”？> * - （CR ^{16 17 ） - （CR 20） - （CR 20） - （CR 20） - （CR 20） - （CR 22）23 - - - （CR 22）23 （CR 26）25（ - ） - （CR 26）25 ） q，r，s，u，v和w是独立地选自0,1和2的整数; A，D，E，G，M，R至R 11和R 16至R 27中的一个整数。 / SUP>，包括这里完全描述。 此外，还公开了包含杀虫有效量的至少一种式I化合物的组合物和通过将所述组合物施用于存在昆虫或预期存在的场所来控制昆虫的方法。}