Invention Grant
US09044518B2 Auristatin tyramine phosphate salts and auristatin aminoquinoline derivatives and prodrugs thereof
有权
Auristatin酪胺磷酸盐和auristatin氨基喹啉衍生物及其前体药物
- Patent Title: Auristatin tyramine phosphate salts and auristatin aminoquinoline derivatives and prodrugs thereof
- Patent Title (中): Auristatin酪胺磷酸盐和auristatin氨基喹啉衍生物及其前体药物
-
Application No.: US14007743Application Date: 2012-03-29
-
Publication No.: US09044518B2Publication Date: 2015-06-02
- Inventor: George R. Pettit , Fiona Hogan , Steven Toms
- Applicant: George R. Pettit , Fiona Hogan , Steven Toms
- Applicant Address: US AZ Scottsdale
- Assignee: ARIZONA BOARD OF REGENTS, A BODY CORPORATE OF THE STATE OF ARIZONA ACTING FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY
- Current Assignee: ARIZONA BOARD OF REGENTS, A BODY CORPORATE OF THE STATE OF ARIZONA ACTING FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY
- Current Assignee Address: US AZ Scottsdale
- Agency: Byrne Poh LLP
- Agent Nina R. Horan
- International Application: PCT/US2012/031118 WO 20120329
- International Announcement: WO2012/135440 WO 20121004
- Main IPC: A61K38/00
- IPC: A61K38/00 ; A61K47/48 ; C07D401/12 ; C07D207/12 ; C07K7/02 ; G01N33/50 ; C07K5/02 ; A61K45/06 ; A61K38/08 ; A61K31/4709 ; A61K31/472

Abstract:
The present invention relates to new auristatin compounds and prodrugs thereof, compositions comprising them and uses thereof.
Public/Granted literature
- US20140023666A1 AURISTATIN TYRAMINE PHOSPHATE SALTS AND AURISTATIN AMINOQUINOLINE DERIVATIVES AND PRODRUGS THEREOF Public/Granted day:2014-01-23
Information query
IPC分类: