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发明授权
CN105246866B 合成巨大戟醇及其中间体的方法 失效 - 权利终止

合成巨大戟醇及其中间体的方法
摘要：
本发明大体上涉及合成二萜杂环化合物的方法。更具体地，本发明涉及从式(1)化合物合成巨大戟醇(式(21)，CAS 30220‑46‑3)的有效方法。本发明还提供沿着巨大戟醇的合成路线的各种有利中间体。巨大戟醇的有效合成在设计和合成相关类似物，诸如巨大戟醇‑3‑当归酸酯中是重要的。
摘要（英）：

The present invention relates generally to methods of synthesis of diterpene heterocylic compounds. More particularly, the present invention relates to efficient methods of synthesis of ingenol (Formula (21), CAS 30220-46-3), from a compound of formula (1). The present invention also provides for various advantageous intermediates along the synthetic route of ingenol. Efficient synthesis of ingenol is important in the design and synthesis of related analogues, such as ingenol-3-angelate.

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