Invention Grant
- Patent Title: Pyrazole compositions useful as inhibitors of ERK
- Patent Title (中): 吡唑组合物可用作ERK的抑制剂
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Application No.: US09971497Application Date: 2001-10-05
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Publication No.: US06784195B2Publication Date: 2004-08-31
- Inventor: Michael Hale , James Janetka , Francois Maltais , Jingrong Cao
- Applicant: Michael Hale , James Janetka , Francois Maltais , Jingrong Cao
- Main IPC: A61K314196
- IPC: A61K314196

Abstract:
Described herein are compounds that are useful as protein kinase inhibitors having the formula: where R1, R2, T and Ht are described in the specification. The compounds are useful for treating disease states in mammals that are alleviated by a protein kinase inhibitor, particularly diseases such as cancer, inflammatory disorders, restenosis, and cardiovascular disease.
Public/Granted literature
- US20020151574A1 Pyrazole compositions useful as inhibitors of ERK Public/Granted day:2002-10-17
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