发明授权
- 专利标题: Piperazine oxytocin receptor antagonists
- 专利标题(中): 哌嗪催产素受体拮抗剂
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申请号: US86107申请日: 1998-05-29
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公开(公告)号: US5968938A公开(公告)日: 1999-10-19
- 发明人: Peter D. Williams , Michelle A. Sparks , Ian Bell , James P. Guare, Jr. , Roger M. Freidinger
- 申请人: Peter D. Williams , Michelle A. Sparks , Ian Bell , James P. Guare, Jr. , Roger M. Freidinger
- 申请人地址: NJ Rahway
- 专利权人: Merck & Co., Inc.
- 当前专利权人: Merck & Co., Inc.
- 当前专利权人地址: NJ Rahway
- 主分类号: C07D211/46
- IPC分类号: C07D211/46 ; C07D211/96 ; C07D213/74 ; C07D235/06 ; C07D239/42 ; C07D241/20 ; C07D295/185 ; A61K31/495 ; C07D401/12 ; C07D403/12
摘要:
This invention relates to certain novel piperazine compounds and derivatives thereof, their synthesis, and their use as oxytocin receptor antagonists. One application of these compounds is in the treatment of preterm labor in mammals, especially humans. The ability of the compounds to relax uterine contractions in mammals also makes them useful for treating dysmenorrhea and stopping labor prior to cesarean delivery.
公开/授权文献
- USD406784S Identification bracelet 公开/授权日:1999-03-16
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