Invention Grant
US5489604A 2-saccharinylmethyl aryl and aryloxy acetates useful as proteolytic
enzyme inhibitors and compositions and method of use thereof
失效
可用作蛋白水解酶抑制剂的2-糖基甲基芳基和芳氧基乙酸酯及其组合物及其使用方法
- Patent Title: 2-saccharinylmethyl aryl and aryloxy acetates useful as proteolytic enzyme inhibitors and compositions and method of use thereof
- Patent Title (中): 可用作蛋白水解酶抑制剂的2-糖基甲基芳基和芳氧基乙酸酯及其组合物及其使用方法
-
Application No.: US287372Application Date: 1994-08-08
-
Publication No.: US5489604APublication Date: 1996-02-06
- Inventor: Lee H. Latimer , Richard P. Dunlap
- Applicant: Lee H. Latimer , Richard P. Dunlap
- Applicant Address: NY New York
- Assignee: Sterling Winthrop, Inc.
- Current Assignee: Sterling Winthrop, Inc.
- Current Assignee Address: NY New York
- Main IPC: A61K9/48
- IPC: A61K9/48 ; A61K31/425 ; A61K31/428 ; A61K31/44 ; A61P1/00 ; A61P11/00 ; A61P35/00 ; A61P43/00 ; C07D275/06 ; C07D417/04 ; C07D417/12 ; C07D513/04
Abstract:
4-R.sup.4 -R.sup.5 -2-Saccharinylmethyl aryl and aryloxy acetates, useful in the treatment of degenerative diseases, are prepared by reacting a 4-R.sup.4 -R.sup.5 -2-halomethylsaccharin with an aryl or aryloxyacetic acid in the presence of an acid-acceptor.
Information query
