Invention Application
- Patent Title: ARYLAMIDE DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN
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Application No.: US16090403Application Date: 2017-04-12
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Publication No.: US20190127357A1Publication Date: 2019-05-02
- Inventor: Pilar GOYA , Antoni TORRENS-JOVER , Carmen ALMANSA-ROSALES , Joser-Luis DIAZ-FERNÁNDEZ , Ana-Maria CAAMAÑO-MOURE
- Applicant: ESTEVE PHARMACEUTICALS , S.A.
- Priority: EP16382166.3 20160412
- International Application: PCT/EP2017/058736 WO 20170412
- Main IPC: C07D413/10
- IPC: C07D413/10 ; C07D413/14 ; C07D401/14 ; C07D401/12 ; C07D409/12 ; C07D409/14 ; C07D405/14 ; C07D417/14
Abstract:
The present invention relates to arylamide derivatives having dual pharmacological activity towards both the α2δ subunit, in particular the α2δ-1 subunit, of the voltage-gated calcium channel and the μ-opioid receptor, to processes of preparation of such compounds, to pharmaceutical compositions comprising them, and to their use in therapy, in particular for the treatment of pain.
Public/Granted literature
- US10577360B2 Arylamide derivatives having multimodal activity against pain Public/Granted day:2020-03-03
Information query
