Invention Application
- Patent Title: Thiazolopyrimidine modulators of TRPV1
- Patent Title (中): TRPV1的噻唑并嘧啶调节剂
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Application No.: US11824202Application Date: 2007-06-28
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Publication No.: US20080004253A1Publication Date: 2008-01-03
- Inventor: Bryan James Branstetter , James Guy Breitenbucher , Alec D. Lebsack , Wei Xiao
- Applicant: Bryan James Branstetter , James Guy Breitenbucher , Alec D. Lebsack , Wei Xiao
- Main IPC: A61K31/55
- IPC: A61K31/55 ; A61K31/541 ; A61K31/5377 ; A61K31/519 ; C07D498/02

Abstract:
Certain TRPV1-modulating thiazolopyrimidine compounds are described. The compounds may be used in pharmaceutical compositions and methods for treating disease states, disorders, and conditions mediated by TRPV1 activity, such as pain, arthritis, itch, cough, asthma, or inflammatory bowel disease.
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